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Cat. No. Product Name Target Signaling Pathways
T8523 ILK-IN-3

Integrin Cytoskeletal Signaling
ILK-IN-3 是一种整合素连接激酶抑制剂,具有抗肿瘤活性。
T5488 ILK-IN-2

OSU-T315

Integrin Cytoskeletal Signaling
ILK-IN-2 (OSU-T315) 是一种新型强效口服活性的整合素连接激酶(ILK)抑制剂,IC50 为 0.6 μM。
T5485 OSU-T315

OSU-T315 (1,5-regioisomer),ILK-IN-2

Apoptosis; Integrin; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling
OSU-T315 (OSU-T315 (1,5-regioisomer)) 是一种整联蛋白连接激酶抑制剂,通过去磷酸化 AKT-Ser473 和其他 ILK 靶标抑制 PI3K/AKT 信号传导。它阻止 AKT 转位到脂筏消除 AKT 的活化,并以 ILK 非依赖性方式触发 Caspase 依赖性细胞凋亡。它通过自噬和凋亡导致细胞死亡。
T80610 Romilkimab

SAR156597

Romilkimab (SAR156597),一种特异性结合IL-4与IL-13的嵌合人源化IG抗体。
T37953 Sphingomyelins (buttermilk)

Sphingomyelins (SMs) are bioactive sphingolipids found in mammalian cell membranes.1SMs make up 2-15% of the total organ phospholipid population but are found at higher concentrations in the brain and myelin sheaths surrounding peripheral nerves. They interact with cholesterol to control its distribution within cellular membranes and maintain cholesterol homeostasis in cells. SMs undergo hydrolysis by sphingomyelinase to form ceramides, which are sphingolipid mediators of intracellular signaling...
T76181 Human milk lysozyme

Human milk lysozyme,一种在人乳中发现的溶菌酶,被认为是保护新生儿胃肠道免受细菌感染的关键防御因子。
T35796 Lactosylceramides (bovine buttermilk)

LacCer (bovine buttermilk)

ROS Immunology/Inflammation
Lactosylceramides (bovine buttermilk) (LacCer (bovine buttermilk)) 是从牛酪乳中分离出来的神经酰胺,抑制细胞增殖,可用于研究肿瘤和肝脏病变。

化合物

ILK-IN-3
Cat.No: T8523
Synonym:
Target: Integrin
ILK-IN-2
Cat.No: T5488
Synonym: OSU-T315
Target: Integrin
OSU-T315
Cat.No: T5485
Synonym: OSU-T315 (1,5-regioisomer),ILK-IN-2
Target: Apoptosis, Integrin, Autophagy
Romilkimab
Cat.No: T80610
Synonym: SAR156597
Target:
Sphingomyelins (buttermilk)
Cat.No: T37953
Synonym:
Target:
Human milk lysozyme
Cat.No: T76181
Synonym:
Target:
Lactosylceramides (bovine buttermilk)
Cat.No: T35796
Synonym: LacCer (bovine buttermilk)
Target: ROS
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