首页 工具
登录
购物车

搜索结果

Search Results for " hsps "

4

抑制剂 & 化合物

1

天然产物

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T7661 SD-169

SD 169,1H-吲哚-5-甲酰胺

p38 MAPK MAPK
SD-169 (SD 169) 是一种可口服的 ATP 竞争性MAPK p38α抑制剂,IC50值为 3.2 nM。它对p38β MAPK 的IC50值为 122 nM。它通过抑制 T 细胞的浸润和活化阻止糖尿病的发展。
T5008 Teprenone

Tetraprenylacetone,Geranylgeranylacetone,替普瑞酮

HSP Cytoskeletal Signaling; Metabolism
Teprenone (Geranylgeranylacetone) 是一种热休克蛋白诱导剂,有抗溃疡作用。
T2444 KNK437

Heat Shock Protein Inhibitor I

HSP Cytoskeletal Signaling; Metabolism
KNK437 (Heat Shock Protein Inhibitor I) 是一种 HSP 抑制剂,抑制 HSP40,HSP70 和 HSP105 的活化。
T36865 Heat Shock Protein Inhibitor II

Heat shock protein (Hsp) inhibitor II is the active form of Hsp inhibitor I and a benzylidene lactam compound that prevents the synthesis of inducible Hsps, such as Hsp105, Hsp72, and Hsp40. Hsp inhibitor II decreases Hsp72 synthesis in vivo and reduces thermotolerance of tumors in SCC VII tumor-containing mice. At 100 μM, it inhibits the development of thermotolerance in COLO 320 DM cells. Inhibition of Hsp70 with Hsp inhibitor II in combination with amphotericin B increases susceptibility of A...

化合物

SD-169
Cat.No: T7661
Synonym: SD 169,1H-吲哚-5-甲酰胺
Target: p38 MAPK
Teprenone
Cat.No: T5008
Synonym: Tetraprenylacetone,Geranylgeranylacetone,替普瑞酮
Target: HSP
KNK437
Cat.No: T2444
Synonym: Heat Shock Protein Inhibitor I
Target: HSP
Heat Shock Protein Inhibitor II
Cat.No: T36865
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T1153 Trimethoprim

NIH 204,BW 56-72,甲氧苄啶,NSC-106568

DHFR; DNA/RNA Synthesis; Antifolate; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Trimethoprim (NSC-106568) 是抑菌抗生素,也是具有口服活性的二氢叶酸还原酶抑制剂。它对多种革兰氏阳性和革兰氏阴性需氧细菌具有活性,可用于尿路感染,肺孢子菌肺炎和志贺氏菌病的研究。

天然产物

Trimethoprim
Cat.No: T1153
Synonym: NIH 204,BW 56-72,甲氧苄啶,NSC-106568
Target: DHFR, DNA/RNA Synthesis, Antifolate, Antibacterial, Antibiotic
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼