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抑制剂 & 化合物

1

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Cat. No. Product Name Target Signaling Pathways
T7447 Adefovir

HBV; Reverse Transcriptase; Telomerase DNA Damage/DNA Repair; Microbiology/Virology
Adefovir 是一种单磷酸腺苷类似物抗病毒剂,在细胞内转化为 Adefovir diphosphate 后可抑制HBVDNA 聚合酶。它在 HepG2.2.15 细胞系中对HBV 的IC50为 0.7 μM。它对多种病毒(包括HBV 和疱疹病毒)具有良好的抗病毒活性。
T0863 Idoxuridine

IDU,碘苷,SKF 14287,5-Iodo-2′-deoxyuridine,NSC 39661,5-IUdR,Dendrid

Antifection; HSV Microbiology/Virology
Idoxuridine (Dendrid) 是一种抑制病毒 DNA 合成的脱氧尿苷类似物,用作抗病毒剂。
T0220 Foscarnet sodium

Phosphonoformate,膦甲酸钠

Virus Protease; Reverse Transcriptase; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Foscarnet sodium (Phosphonoformate) 是一种病毒 DNA 聚合酶活性抑制剂,可逆地抑制病毒复制。它是一种用于治疗巨细胞病毒性视网膜炎的抗病毒剂。
T31659 Eprociclovir

AV10,AV-10,A-5021,A 5021,A5021,AV 10

Antifection Microbiology/Virology
Eprociclovir (A-5021) 是一种新型阿昔洛韦类似物,是 EHV1 复制的强效抑制剂,可能用于治疗和/或预防该病毒感染。Eprociclovir 对大多数人类疱疹病毒都有很强的抗疱疹活性。
T80672 1,4-Dihydroxynaphthalene

Naphthalene-1,4-diol

HSV Microbiology/Virology
1,4-Dihydroxynaphthalene 一种有效的 HSV-1蛋白酶抑制剂,对HCMV蛋白酶有抑制作用,可用于研究疱疹病毒。
TQ0095 Brincidofovir

CMX001,HDP-CDV

Others; Antiviral; HSV Immunology/Inflammation; Microbiology/Virology; Others
Brincidofovir (HDP-CDV) 是 Cidofovir 的一种具有口服活性的亲脂性形式的前体药物,是一种口服长效的抗病毒药物,有广泛的抗 DNA 病毒活性。
T29093 Valomaciclovir stearate

A-174606.0,RP-606,EPB-348,ABT-606,MIV-606

Valomaciclovir stearate is a DNA polymerase inhibitor. Valomaciclovir stearate is an orally available drug with broad-spectrum antiviral activity against a variety of important herpesviruses, including Epstein-Barr virus, or EBV (the first virus to be dir
T70027 Eprociclovir potassium

Eprociclovir potassium is a new acyclovir analogue and a potent inhibitor of EHV1 replication and may have potential for the treatment and/or prophylaxis of infections with this virus. Eprociclovir possess potent anti-herpetic activity against most human herpesviruses. A-5021 proved to be about 15-fold more potent than acyclovir in inhibiting viral replication. Eprociclovir inhibits murine herpetic keratitis. A-5021 eyedrops, which are easily applied onto the affected cornea, ameliorated clinica...
T69817 Eprociclovir Na

Eprociclovir Na is the salt form of Eprociclovir, also known as A-5021, a new acyclovir analogue and a potent inhibitor of EHV1 replication and may have potential for the treatment and/or prophylaxis of infections with this virus. Eprociclovir possess potent anti-herpetic activity against most human herpesviruses. A-5021 proved to be about 15-fold more potent than acyclovir in inhibiting viral replication. Eprociclovir inhibits murine herpetic keratitis. A-5021 eyedrops, which are easily applie...
T68957 Eprociclovir dihydrate

Eprociclovir dihydrate is a new acyclovir analogue and a potent inhibitor of EHV1 replication and may have potential for the treatment and/or prophylaxis of infections with this virus. Eprociclovir possess potent anti-herpetic activity against most human herpesviruses. A-5021 proved to be about 15-fold more potent than acyclovir in inhibiting viral replication. Eprociclovir inhibits murine herpetic keratitis. A-5021 eyedrops, which are easily applied onto the affected cornea, ameliorated clinica...

化合物

Adefovir
Cat.No: T7447
Synonym:
Target: HBV, Reverse Transcriptase, Telomerase
Idoxuridine
Cat.No: T0863
Synonym: IDU,碘苷,SKF 14287,5-Iodo-2′-deoxyuridine,NSC 39661,5-IUdR,Dendrid
Target: Antifection, HSV
Foscarnet sodium
Cat.No: T0220
Synonym: Phosphonoformate,膦甲酸钠
Target: Virus Protease, Reverse Transcriptase, DNA/RNA Synthesis
Eprociclovir
Cat.No: T31659
Synonym: AV10,AV-10,A-5021,A 5021,A5021,AV 10
Target: Antifection
1,4-Dihydroxynaphthalene
Cat.No: T80672
Synonym: Naphthalene-1,4-diol
Target: HSV
Brincidofovir
Cat.No: TQ0095
Synonym: CMX001,HDP-CDV
Target: Others, Antiviral, HSV
Valomaciclovir stearate
Cat.No: T29093
Synonym: A-174606.0,RP-606,EPB-348,ABT-606,MIV-606
Target:
Eprociclovir potassium
Cat.No: T70027
Synonym:
Target:
Eprociclovir Na
Cat.No: T69817
Synonym:
Target:
Eprociclovir dihydrate
Cat.No: T68957
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T75643 Isoxanthohumol

HSV Microbiology/Virology
Isoxanthohumol 是一种从啤酒花和啤酒中提取的一种前黄酮类化合物,对几种人类癌细胞株具有抗增殖活性。Isoxanthohumol对肿瘤细胞肺转移灶的转移或侵袭有抑制作用。Isoxanthohumol具有抗病毒活性,对疱疹病毒(HSV1和HSV2)和牛病毒性腹泻病毒(BVDV)具有抑制作用。

天然产物

Isoxanthohumol
Cat.No: T75643
Synonym:
Target: HSV
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