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Cat. No.	Product Name	Target	Signaling Pathways
T7389	G15	Estrogen Receptor/ERR	Endocrinology/Hormones
	G15 是一种高亲和力的、选择性的 G 蛋白偶联雌激素受体(GPER/GPR30)拮抗剂(Ki:20 nM)。
T2034	AG1557 AG-1557,AG 1557	EGFR; HER	Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
	AG1557 (AG-1557) 是一种表皮生长因子受体(EGFR) 酪氨酸激酶抑制剂，pIC50值为 8.194。
T11344	G150	DNA; cGAS	DNA Damage/DNA Repair; Immunology/Inflammation
	G150 是高选择性h-cGAS 抑制剂，IC50值为 10.2 nM，用于抑制 dsDNA 引发的干扰素表达。
T17414	Amino-PEG15-amine H2N-PEG15-CH2CH2NH2	Others	Others
	Amino-PEG15-amine is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
T70391	AMG151 HCl
	ARRY-403, also known as AMG-151, is an orally available allosteric glucokinase (GK) activator developed for the treatment of type 2 diabetes mellitus (T2DM). ARRY-403 has many favorable physicochemical characteristics and ADME properties (low potential to cause drug–drug interactions (DDIs). ARRY-403 potently activates human glucokinase (GK) in vitro (EC50 = 79 nM at 5 mM glucose), with an S0.5 = 0.93 mM glucose (ARRY-403 at 5 mM) and Vmax = 134% compared to the no activator control. It possesse...
T17968	Fmoc-NH-PEG15-CH2CH2COOH	Others	Others
	Fmoc-NH-PEG15-CH2CH2COOH is a PEG-based PROTAC linker utilized for PROTAC synthesis[1].
T17488	Azido-PEG15-t-butyl ester	Others	Others
	Azido-PEG15-t-butyl ester is a polyethylene glycol (PEG) derived linker, specifically designed for the synthesis of proteolysis-targeting chimeras (PROTACs)[1].
T17715	Cbz-N-PEG15-amine	Others	Others
	Cbz-N-PEG15-amine is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
T18150	m-PEG15-NHS ester	Others	Others
	m-PEG15-NHS ester is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
T17670	Boc-NH-PEG15-azide	Others	Others
	Boc-NH-PEG15-azide is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
T17487	Azido-PEG15-azide	Others	Others
	Azido-PEG15-azide is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
T15490	HO-PEG15-OH	Others	Others
	HO-PEG15-OH is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
T18149	m-PEG15-alcohol	Others	Others
	m-PEG15-alcohol is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
T17620	Bis-PEG15-acid	Others	Others
	Bis-PEG15-acid is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
T17671	Boc-NH-PEG15-NH2	Others	Others
	Boc-NH-PEG15-NH2 is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.

化合物

Cat.No: T7389

Target: Estrogen Receptor/ERR

Cat.No: T2034

Synonym: AG-1557,AG 1557

Target: EGFR, HER

Cat.No: T11344

Target: DNA, cGAS

Amino-PEG15-amine

Cat.No: T17414

Synonym: H2N-PEG15-CH2CH2NH2

Target: Others

Cat.No: T70391

Fmoc-NH-PEG15-CH2CH2COOH

Cat.No: T17968

Target: Others

Azido-PEG15-t-butyl ester

Cat.No: T17488

Target: Others

Cbz-N-PEG15-amine

Cat.No: T17715

Target: Others

m-PEG15-NHS ester

Cat.No: T18150

Target: Others

Boc-NH-PEG15-azide

Cat.No: T17670

Target: Others

Azido-PEG15-azide

Cat.No: T17487

Target: Others

Cat.No: T15490

Target: Others

m-PEG15-alcohol

Cat.No: T18149

Target: Others

Cat.No: T17620

Target: Others

Boc-NH-PEG15-NH2

Cat.No: T17671

Target: Others

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