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Cat. No. Product Name Target Signaling Pathways
TN1121 Evocarpine

Apoptosis; cAMP; Anti-infection; Calcium Channel; Antibacterial Apoptosis; GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Evocarpine 是从 Evodiae fructus 分离得到的一种喹诺酮类生物碱,有抗细菌活性。它可通过电压依赖性钙通道抑制 Ca2+内流。
TN1099 Dihydroevocarpine

MAO; P-gp; Antifection Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience
Dihydroevocarpine shows potent anti-Helicobacter pylori activity with the minimum inhibitory concentration (MIC) value of 10-20 microg/ml. Dihydroevocarpine is a moderate modulator of p-glycoprotein (p-gp) activity; it shows more potent inhibitory effects against MAO-B compared to MAO-A.

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Evocarpine
Cat.No: TN1121
Synonym:
Target: Apoptosis, cAMP, Anti-infection, Calcium Channel, Antibacterial
Dihydroevocarpine
Cat.No: TN1099
Synonym:
Target: MAO, P-gp, Antifection
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