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Cat. No. | Product Name | Target | Signaling Pathways |
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T11191 |
EN6
|
Proton pump; Autophagy | Autophagy; Membrane transporter/Ion channel |
EN6 是一种小分子体内自噬激活剂,其共价靶向溶酶体v-ATP 酶的 ATP6V1A 亚基中的半胱氨酸 277。它以溶酶体依赖性方式清除 TDP-43 聚集体,这是额颞叶痴呆的病原体。它介导的 ATP6V1A 修饰使 v-ATP 酶与 Rags 分离,从而抑制 mTORC1 信号传导、增加溶酶体酸化和激活自噬。 | |||
T25150 |
BI-69A11
BI 69A11,(E)-3-(1H-Benzo[d]imidazol-2-yl)-1-(6-chloro-2-hydroxy-4-phenylquinolin-3-yl)prop-2-en-1-one |
NF-κB; Akt | Cytoskeletal Signaling; NF-κB; PI3K/Akt/mTOR signaling |
BI-69A11 ((E)-3-(1H-Benzo[d]imidazol-2-yl)-1-(6-chloro-2-hydroxy-4-phenylquinolin-3-yl)prop-2-en-1-one) 是一种双重 AKT 和 NFkB 通路抑制剂。它通过靶向 Akt 增强结肠癌细胞对 mda-7/IL-24 诱导的生长抑制的敏感性。 | |||
T124161 |
5α,8α-Epidioxyergost-6-en-3β-ol
|
||
5α,8α-Epidioxyergost-6-en-3β-ol 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124161。 | |||
T126063 |
8-Oxoeremophil-6-en-12-oic aicd
|
||
8-Oxoeremophil-6-en-12-oic aicd 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126063。 | |||
T123873 |
6-(4-Hydroxyphenyl)-2-methylhept-2-en-4-one
|
||
6-(4-Hydroxyphenyl)-2-methylhept-2-en-4-one 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T123873。 | |||
TNU0739 | (-)-(1S,5R)-cis-Bicyclo[3.2.0]hept-2-en-6-one | ||
Building block - others | |||
TNU0847 |
6-[[(3b)-Cholest-5-en-3-yl]oxy]-1-hexanol
|
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Intermediate and Building Blocks - Nucleophile; Scaffolds and Templates | |||
T130192 |
3,5,7-Trihydroxy-p-menth-1-en-6-one, 5-Tigloyl, 3
|
||
3,5,7-Trihydroxy-p-menth-1-en-6-one, 5-Tigloyl, 3 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T130192。 | |||
T125520 |
(S,E)-2-Methyl-6-(p-tolyl)hept-3-en-2-ol
|
||
(S,E)-2-Methyl-6-(p-tolyl)hept-3-en-2-ol 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125520。 | |||
T65075 |
(3S,8S,9S,10R,13R,14S,17R)-10,13-Dimethyl-17-((R)-6-methylheptan-2-yl)-2,3,4,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-3-yl (Z)-octadec-9-en-1-yl carbonate
|
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(3S,8S,9S,10R,13R,14S,17R)-10,13-Dimethyl-17-((R)-6-methylheptan-2-yl)-2,3,4,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-3-yl (Z)-octadec-9-en-1-yl carbonate 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65075,CAS号为 17110-51-9。 | |||
TNU0846 |
Chlolest-5-en-3β-tosylate; Cholest-5-en-3-ol (3β)-(4-methylbenzenesulfonate)
|
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Chlolest-5-en-3β-tosylate; Cholest-5-en-3-ol (3β)-(4-methylbenzenesulfonate) 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TNU0846,CAS号为 1182-65-6。 | |||
T69766 |
Gusacitinib HCl
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||
Gusacitinib, also known as ASN-002 and EN-3351, is a potent dual inhibitor of SYK/JAK kinases. ASN002 showed strong antitumor activity in both hematological and solid tumor xenograft models. ASN002 strongly suppressed the SYK and JAK family kinase signaling pathways as measured in pLAT and pSTAT assays, respectively. When profiled in a panel of 178 cell lines, ASN002 showed strong anti-proliferative activity in many lymphoid/leukemia cell lines, including SU-DHL-6, SU-DHL-4, OCI-LY10, H929 and... | |||
T37419 | Zetomipzomib | ||
KZR-616, a first-in-class inhibitor of the immunoproteasome, selectively targets the LMP7 (IC50: 39/57 nM=hLMP7/mLMP7) and LMP2 (IC50: 131/179 nM=hLMP7/mLMP7) subunits of the immunoproteasome. KZR-616 has the potential for the research of multiple autoimmune diseases[1][2]. KZR-616 also inhibits MECL-1 subunit (IC50=623 nM) and constitutive proteasome β5 subunit (IC50=688 nM). KZR-616 maintains LMP7 and LMP2 selective inhibition in MOLT-4 cells. KZR-616 (250 nM) shows a comparable cytokine inhib... |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN6832 |
Sulcatone
6-甲基-5-庚烯-2-酮,6-methylhept-5-en-2-one,6-Methyl-5-hepten-2-one |
Endogenous Metabolite | Metabolism |
Sulcatone (6-Methyl-5-hepten-2-one) 是内源性代谢产物的一种。 | |||
TN2584 |
11-Hydroxydrim-7-en-6-one
|
Others | Others |
11-Hydroxydrim-7-en-6-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2584,CAS号为 74635-87-3。 | |||
TN3332 | 9alpha,11-Dihydroxydrim-7-en-6-one | Others | Others |
9alpha,11-Dihydroxydrim-7-en-6-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3332,CAS号为 127681-58-7。 | |||
TN3331 |
9alpha,11,12-Trihydroxydrim-7-en-6-one
|
Others | Others |
9alpha,11,12-Trihydroxydrim-7-en-6-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3331,CAS号为 192566-65-7。 | |||
TN6357 |
5-Hydroxy-1,7-diphenylhept-6-en-3-one
|
||
5-Hydroxy-1,7-diphenylhept-6-en-3-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6357,CAS号为 155239-30-8。 | |||
TN5861 |
3-Hydroxy-p-menth-1-en-6-one
(3R,4S)-3-Hydroxy-p-menth-1-en-6-one |
||
3-Hydroxy-p-menth-1-en-6-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5861,CAS号为 61570-82-9。 | |||
TN2513 |
1,7-Bis(4-hydroxyphenyl)hept-6-en-3-ol
|
Others | Others |
1,7-Bis(4-hydroxyphenyl)hept-6-en-3-ol is a natural product from Alpinia galanga. | |||
TN2514 |
1,7-Bis(4-hydroxyphenyl)hept-6-en-3-one
|
Others | Others |
1,7-Bis(4-hydroxyphenyl)hept-6-en-3-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2514,CAS号为 1251830-57-5。 | |||
TN1214 |
2-Methoxy-5-acetoxy-fruranogermacr-1(10)-en-6-one
2-Methoxy-5-acetoxy-furanogermacr-1(10)-en-6-one |
Others | Others |
2-Methoxy-5-acetoxy-furanogermacr-1(10)-en-6-one is a natural product | |||
TN2994 |
4-(6-Methyl-4-oxohept-5-en-2-yl)cyclohex-2-en-1-one
|
Others | Others |
4-(6-Methyl-4-oxohept-5-en-2-yl)cyclohex-2-en-1-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2994,CAS号为 170380-68-4。 | |||
TN3068 |
4|A,6|A-Dihydroxyeudesm-11(13)-en-12,8|A-olide
4alpha,6alpha-Dihydroxyeudesm-11(13)-en-12,8beta-olide |
Others | Others |
4|A,6|A-Dihydroxyeudesm-11(13)-en-12,8|A-olide 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3068,CAS号为 35001-19-5。 | |||
TN3141 |
6-(4-Hydroxy-3-methylphenyl)-2-methylhept-2-en-4-one
|
Others | Others |
6-(4-Hydroxy-3-methylphenyl)-2-methylhept-2-en-4-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3141,CAS号为 949081-05-4。 | |||
TN2471 |
1-(3,4-Dihydroxyphenyl)-7-(4-hydroxyphenyl)hept-6-en-3-ol
|
Others | Others |
1-(3,4-Dihydroxyphenyl)-7-(4-hydroxyphenyl)hept-6-en-3-ol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2471,CAS号为 1206788-61-5。 | |||
TN6909 |
Polyporusterone B
猪苓酮B,(1R,2R,4S,5R,7R,11R,14S,15R)-14-[(2R,3R)-2,3-dihydroxy-6-methyl-5-methylideneheptan-2-yl]-4,5,11-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,?.011,1?]heptadec-9-en-8-one |
Others | Others |
Polyporusterone B ((1R,2R,4S,5R,7R,11R,14S,15R)-14-[(2R,3R)-2,3-dihydroxy-6-methyl-5-methylideneheptan-2-yl]-4,5,11-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,?.011,1?]heptadec-9-en-8-one) 是一种三萜羧酸,从Polyporus umbellatusFries 中分离得到。它对自由基诱导的红细胞裂解 (溶血) 具有抑制作用。 | |||
TN5870 |
1,8-Dihydroxy-p-menth-3-en-2-one
6-Hydroxy-3-(2-hydroxypropan-2-yl)-6-methylcyclohex-2-en-1-one |
||
1,8-Dihydroxy-p-menth-3-en-2-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5870,CAS号为 1392224-56-4。 | |||
TN6864 |
Prosaikogenin F
(2R,3R,4S,5R,6R)-2-{[(1S,2R,4S,5R,8R,9S,10R,13S,14R,17S,18R)-2-hydroxy-9-(hydroxymethyl)-4,5,9,13,20,20-hexamethyl-24-oxahexacyclo[15.5.2.01,1?.0?,1?.0?,1?.0?,13]tetracos-15-en-10-yl]oxy}-6-methyloxane-3,4,5-triol,前柴胡皂苷F |
Others | Others |
Prosaikogenin F ((2R,3R,4S,5R,6R)-2-{[(1S,2R,4S,5R,8R,9S,10R,13S,14R,17S,18R)-2-hydroxy-9-(hydroxymethyl)-4,5,9,13,20,20-hexamethyl-24-oxahexacyclo[15.5.2.01,1?.0?,1?.0?,1?.0?,13]tetracos-15-en-10-yl]oxy}-6-methyloxane-3,4,5-triol) 是一种单糖苷,具有溶血和抗癌特性。 | |||
TN6498 |
Stevia impurity (13-[(2-O-6-deoxy-β-D-glucopyranosyl-3-O-β-D-glucopyranosyl-β-D-glucopyranosyl)oxy]ent-kaur-16-en-19-oic acid β-D-glucopyranosyl ester)
|
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Stevia impurity (13-[(2-O-6-deoxy-β-D-glucopyranosyl-3-O-β-D-glucopyranosyl-β-D-glucopyranosyl)oxy]ent-kaur-16-en-19-oic acid β-D-glucopyranosyl ester) 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6498,CAS号为 1309929-72-3。 | |||
TN1201 |
25(S)-Ruscogenin-1-O-α-L-rhamnopyranosyl (1→2)-β-D-xylopyranoside
25(S)-鲁斯可皂苷元-1-O-Α-L-吡喃鼠李糖基-(1→2)-Β-D-吡喃木糖苷,山麦冬皂苷C,(1beta,3beta,25S)-3-Hydroxyspirost-5-en-1-yl 2-O-(6-deoxy-alpha-L-mannopyranosyl)-beta-D-xylopyranoside |
Others | Others |
(1beta,3beta,25S)-3-Hydroxyspirost-5-en-1-yl 2-O-(6-deoxy-alpha-L-mannopyranosyl)-beta-D-xylopyranoside is a natural product | |||
TN2512 |
1,7-Bis(4-hydroxyphenyl)hept-1-en-3-one
|
Others | Others |
1,7-Bis(4-hydroxyphenyl)hept-1-en-3-one是一种天然产物,属于姜科山姜属,其产品编号为 TN2512,CAS号为 1083200-79-6。1,7-Bis(4-hydroxyphenyl)hept-1-en-3-one可用作对照参考。 | |||
TN3755 |
Dammar-20(21)-en-3,24,25-triol
|
Others | Others |
Dammar-20(21)-en-3,24,25-triol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3755,CAS号为 55050-69-6。 |