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Search Results for " deoxycorticosterone acetate "

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抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T11394 GFB-8438

TRP/TRPV Channel Membrane transporter/Ion channel
GFB-8438 是有效的TRPC5选择性抑制剂,对 hTRPC5 和 hTRPC4 的IC50分别为 0.18 和 0.29 μM。它对 TRPC6、其他 TRP 家族成员、NaV1.5 具有良好的选择性,对 hERG 通道的活性也有限。它对小鼠足细胞的保护作用。
T26841 BMS 182874

BMS182874,BMS-182874

Endothelin Receptor GPCR/G Protein
BMS 182874 是一种口服有效的高选择性内皮素受体 endothelin receptor ETA 拮抗剂,对 ETA 的 IC50 值为0.150 μM,对 ETA 的 Ki 值为0.055 μM。BMS 182874 能够在大鼠高血压模型中降低 Deoxycorticosterone acetate 诱导的动脉压,可用于研究心血管疾病。
T35876 Chlorthalidone Impurity G

Chlorthalidone impurity G is a potential impurity found in commercial preparations of chlorthalidone that has moderate antihypertensive effects. Chlorthalidone is a thiazide-like diuretic that inhibits the Na+/Cl- cotransporter in the distal convoluted tubule of the kidney, which prevents reabsorption of sodium and chloride leading to a reduction in plasma volume and cardiac output. It also inhibits carbonic anhydrase (CA), including the isoforms CAVB, VII, IX, XII, and XIII (Kis = 2.8-23 nM) an...

化合物

GFB-8438
Cat.No: T11394
Synonym:
Target: TRP/TRPV Channel
BMS 182874
Cat.No: T26841
Synonym: BMS182874,BMS-182874
Target: Endothelin Receptor
Chlorthalidone Impurity G
Cat.No: T35876
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T3033 Deoxycorticosterone acetate

醋酸去氧皮质酮,DOC acetate,Cortexone acetate,11-Deoxycorticosterone acetate,醋酸脱氧皮质酮

Glucocorticoid Receptor; Endogenous Metabolite; Adrenergic Receptor Endocrinology/Hormones; GPCR/G Protein; Metabolism; Neuroscience
Deoxycorticosterone acetate (Cortexone acetate) 是肾上腺产生的类固醇激素,具有盐皮质激素活性,并作为醛固酮的前体。

天然产物

Deoxycorticosterone acetate
Cat.No: T3033
Synonym: 醋酸去氧皮质酮,DOC acetate,Cortexone acetate,11-Deoxycorticosterone acetate,醋酸脱氧皮质酮
Target: Glucocorticoid Receptor, Endogenous Metabolite, Adrenergic Receptor
TargetMol Loading
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