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Search Results for " cyclic 3',5'-monophosphate adenosine "

6

抑制剂 & 化合物

3

天然产物

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Cat. No. Product Name Target Signaling Pathways
T31931L Gizzerosine HCl

Gizzerosine HCl(89238-78-8 Free base)

Others Others
Gizzerosine 2HCl是鱼粉热处理过程中产生的一种物质,可诱导的肉鸡雏鸡组织病理学病变,可提高离体鸡原产鸡的细胞内环腺苷-3',5'-单磷酸水平。
T1024 Roflumilast

罗氟司特,B9302-107,BYK 20869,APTA 2217,BY 217

PDE; RSV Metabolism; Microbiology/Virology
Roflumilast (APTA 2217) 是一种口服的长效 4 型磷酸二酯酶抑制剂 (PDE4),具有抗炎和潜在的抗肿瘤活性,作用于PDE4A1,PDEA4,PDEB1和PDEB2,IC50分别为 0.7,0.9,0.7 和 0.2 nM。
T1139 Salbutamol

Albuterol,沙丁胺醇,AH-3365

Adrenergic Receptor GPCR/G Protein; Neuroscience
Salbutamol (Albuterol) 是短效的 β2 肾上腺素受体激动剂,用于哮喘和慢性阻塞性肺疾病(COPD) 引发的支气管痉挛的研究。
T25463 Griseolic acid

Griseolic acid is a cyclic adenosine 3',5'-monophosphate phosphodiesterase II inhibitor.
T32156 Indimilast

Indimilast is used to inhibit phosphodiesterase IV that regulates lung inflammation and causes bronchiectasis by increasing intracellular cyclic adenosine 3', 5'-monophosphate in airway smooth muscle and inflammatory cells. Potential to treat chronic obst
T63776 PDE1-IN-4

PDE1-IN-4 是有效的、选择性的 PDE1 (磷酸二酯酶 -1) 抑制剂,能够作用于 PDE1C (IC50: 10 nM)、PDE1A (IC50: 145 nM) 和 PDE1B (IC50: 354 nM)。PDE1-IN-4 能够调控 cAMP (3′,5′- 环磷酸腺苷) 和 cGMP (3′,5′- 环磷酸鸟苷),表现出抗纤维化效果。PDE1-IN-4 能够抑制 TGF-β1 诱导的人肺成纤维细胞分化。PDE1-IN-4 能够用于研究特发性肺纤维化 (IPF)。

化合物

Gizzerosine HCl
Cat.No: T31931L
Synonym: Gizzerosine HCl(89238-78-8 Free base)
Target: Others
Roflumilast
Cat.No: T1024
Synonym: 罗氟司特,B9302-107,BYK 20869,APTA 2217,BY 217
Target: PDE, RSV
Salbutamol
Cat.No: T1139
Synonym: Albuterol,沙丁胺醇,AH-3365
Target: Adrenergic Receptor
Griseolic acid
Cat.No: T25463
Synonym:
Target:
Indimilast
Cat.No: T32156
Synonym:
Target:
PDE1-IN-4
Cat.No: T63776
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TCO2745 Cyclic AMP

Adenosine 3',5'-cyclophosphate,cAMP,腺苷环磷酸酯,环磷腺苷,Cyclic 3',5'-monophosphate adenosine,3',5'-AMP,Adenosine Cyclophosphate

Others; Endogenous Metabolite Metabolism; Others
Cyclic AMP (cAMP)(Adenosine 3',5'-cyclophosphate) 是有丝分裂信使,可以促进 G1期到 S 期的细胞周期进程。
TN1841 Kushenol A

苦参新醇 A,Leachianone E

cAMP GPCR/G Protein
Kushenol A is a kind of Adenosine 3', 5'-cyclic monophosphate(cAMP)phosphodiesterase inhibitiors, it shows selective alpha-glucosidase inhibitory activity. Kushenol A and kushenol C exhibit inhibitory activity against Sodium-dependent glucose cotransporter 2(SGLT2).
TN4433 Licoarylcoumarin

cAMP; HIV Protease; Antifection GPCR/G Protein; Microbiology/Virology; Proteases/Proteasome
Licoarylcoumarin is a strong inhibitor of adenosine 3',5'-cyclic monophosphate (cAMP) phosphodiesterase. Licoarylcoumarin has antibacterial effects on the VRE strains; it has anti-HIV activity, and it has inhibitory effects on xanthine oxidase.

天然产物

Cyclic AMP
Cat.No: TCO2745
Synonym: Adenosine 3',5'-cyclophosphate,cAMP,腺苷环磷酸酯,环磷腺苷,Cyclic 3',5'-monophosphate adenosine,3',5'-AMP,Adenosine Cyclophosphate
Target: Others, Endogenous Metabolite
Kushenol A
Cat.No: TN1841
Synonym: 苦参新醇 A,Leachianone E
Target: cAMP
Licoarylcoumarin
Cat.No: TN4433
Synonym:
Target: cAMP, HIV Protease, Antifection
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