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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T126112 | Epiprocurcumenol | ||
Epiprocurcumenol 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126112。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3669 |
Curcumenol
(+)-Curcumenol,莪术醇 |
P450 | Metabolism |
Curcumenol ((+)-Curcumenol) 提取具有药用价值的 Curcuma zedoaria,是高效的 CYP3A4抑制剂(IC50=12.6 μM),具有神经抗肿瘤、保护、抗炎、和保肝的作用。它在 LPS 刺激的 BV-2 小胶质细胞中,抑制 Akt 介导的 NF-κB 活化及 p38 MAPK 信号通路。 | |||
TN3025 | 4-Epi-curcumenol | Others | Others |
4-Epi-curcumenol是一种天然产物,属于姜科姜黄属,其产品编号为 TN3025,CAS号为 350602-21-0。4-Epi-curcumenol可用作对照参考。 | |||
T5S0543 |
Isocurcumenol
|
Apoptosis; Estrogen Receptor/ERR; Reductase | Apoptosis; Endocrinology/Hormones; Metabolism |
Isocurcumenol 是从莪术中分离得到的一种天然产物,是一种ERα抑制剂,对 DLA 和 KB 癌细胞的IC50分别为 99.1 µg/mL 和 178.2 µg/mL,具有抗肿瘤活性。 | |||
TN4320 |
Isoprocurcumenol
|
Others | Others |
Isoprocurcumenol is an inhibitor of Nitric Oxide. | |||
TN4641 |
Neoprocurcumenol
|
Others | Others |
Neoprocurcumenol exerts significant toxicity on mosquito larvae. | |||
TN2102 | Procurcumenol | Others; TNF | Apoptosis; Others |
Procurcumenol is an inhibitor of Nitric Oxide. Procurcumenol and epicurcumenol have inhibitory effects on release of tumor necrosis factor-a (TNF-a). |