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Cat. No. Product Name Target Signaling Pathways
T10729 Cdc7-IN-7

CDK Cell Cycle/Checkpoint
Cdc7-IN-7 (compound I-E) 是一种有效的 Cdc7 激酶抑制剂。
T10727 Cdc7-IN-5

CDK Cell Cycle/Checkpoint
Cdc7-IN-5 是一种有效的 Cdc7 激酶抑制剂。Cdc7 是一种丝氨酸苏氨酸蛋白激酶酶,在细胞周期中对 DNA 复制的启动至关重要。
T23867 Cdc7-IN-7c

Cdc7 inhibitor-7c,Cdc7 inhibitor 7c,Cdc7 IN 7c

CDK Cell Cycle/Checkpoint
Cdc7-IN-7c (Cdc7 inhibitor-7c) 具有抗肿瘤活性,对肝癌,肺癌,肾癌,脑癌,宫颈癌有抑制作用。
T10724 Cdc7-IN-1

CDK Cell Cycle/Checkpoint
Cdc7-IN-1 is a highly selective and ATP competitive inhibitor of Cdc7 kinase (IC50: 0.6 nM at 1 mM ATP). It potently inhibits Cdc7 activity in cancer cells and effectively induces cell death.
T10726 Cdc7-IN-4

Others Others
Cdc7-IN-4 is a potent inhibitor of Cdc7 kinase.
T10725 Cdc7-IN-3

Others Others
Cdc7-IN-3 is a potent inhibitor of Cdc7 kinase.
T3352 XL413

cholecystokinin; Casein Kinase; Pim; CDK Cell Cycle/Checkpoint; Chromatin/Epigenetic; GPCR/G Protein; JAK/STAT signaling; Metabolism; Stem Cells
XL413 是一种口服生物可利用的细胞分裂周期 7 同源物 (CDC7) 激酶抑制剂,具有潜在的抗肿瘤活性,IC50值为 3.4 nM。它对 pMCM 的 EC50值为 118 nM,对 CK2 和 PIM1 的 IC50值分别为 215 和 42 nM。

化合物

Cdc7-IN-7
Cat.No: T10729
Synonym:
Target: CDK
Cdc7-IN-5
Cat.No: T10727
Synonym:
Target: CDK
Cdc7-IN-7c
Cat.No: T23867
Synonym: Cdc7 inhibitor-7c,Cdc7 inhibitor 7c,Cdc7 IN 7c
Target: CDK
Cdc7-IN-1
Cat.No: T10724
Synonym:
Target: CDK
Cdc7-IN-4
Cat.No: T10726
Synonym:
Target: Others
Cdc7-IN-3
Cat.No: T10725
Synonym:
Target: Others
XL413
Cat.No: T3352
Synonym:
Target: cholecystokinin, Casein Kinase, Pim, CDK
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