首页 工具
登录
购物车

搜索结果

Search Results for " cataplexy "

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T2613 Almorexant

阿莫伦特,ACT 078573

OX Receptor GPCR/G Protein; Neuroscience
Almorexant (ACT 078573) 是一种有效的竞争性食欲素 1 受体 (OX1)/食欲素 2 受体 (OX2) 双重拮抗剂,OX1 和 OX2 的 Ki 值分别为 1.3 和 0.17 nM。
T6155 Almorexant hydrochloride

ACT-078573 hydrochloride,Almorexant HCl

OX Receptor GPCR/G Protein; Neuroscience
Almorexant hydrochloride (ACT-078573 hydrochloride) 是一种有效的竞争性食欲素 1 受体(OX1)/食欲素 2 受体 (OX2) 双重拮抗剂,OX1 和 OX2 的 Ki 值分别为 1.3 和 0.17 nM。
T39229 YNT-185

OX Receptor GPCR/G Protein; Neuroscience
YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R, respectively. Furthermore, YNT-185 effectively alleviates symptoms of narcolepsy-cataplexy in mouse models.
T37112 YNT-185 dihydrochloride

Potent and selective orexin OX2 receptor agonist (EC50 = 28 nM at human OX2 expressed in CHO cells). Displays approximately 100-fold selectivity for OX2 over OX1 (EC50 = 2.75 μM at human OX1 expressed in CHO cells). Depolarizes OX2-expressing histaminergic neurons in mouse brain slices. Increases wake time in wild type mice. Suppresses cataplexy-like symptoms in OX knockout mice. Nagahara et al (2015) Design and synthesis of non-peptide, selective orexin receptor 2 agonists. J.Med.Chem. 58 7931 ...
T78636 Firazorexton hydrate

TAK-994

Firazorexton hydrate (TAK-994)为一种高效的食欲素2型受体(OX2R)激动剂,EC50值为19 nM。在发作性睡病小鼠模型中,该化合物能够有效减少觉醒碎片和猝倒样发作的发生。

化合物

Almorexant
Cat.No: T2613
Synonym: 阿莫伦特,ACT 078573
Target: OX Receptor
Almorexant hydrochloride
Cat.No: T6155
Synonym: ACT-078573 hydrochloride,Almorexant HCl
Target: OX Receptor
YNT-185
Cat.No: T39229
Synonym:
Target: OX Receptor
YNT-185 dihydrochloride
Cat.No: T37112
Synonym:
Target:
Firazorexton hydrate
Cat.No: T78636
Synonym: TAK-994
Target:
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼