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Cat. No. Product Name Target Signaling Pathways
T63480 COX-2-IN-26

COX-2-IN-26 是有效的、口服具有活力的、选择性的 COX-2 抑制剂,能够作用于 COX-1 (IC50: 10.61 μM)、COX-2 (IC50: 0.067 μM)、15-LOX (IC50: 1.96 μM)。COX-2-IN-26 具有抗炎作用,具有胃肠道安全性。
T1185 Rofecoxib

MK 966,罗非昔布,罗非考昔,MK-0966

COX Immunology/Inflammation; Neuroscience
Rofecoxib (MK 966) 是可口服的 COX-2特异性抑制剂,具有抗炎、解热和镇痛特性以及潜在的抗肿瘤特性。在人骨肉瘤细胞和中国仓鼠卵巢细胞中,对人 COX-2 的 IC50值分别为 26 和 18 nM。
T0839 Ketoprofen

酮基布洛芬,RP-19583,酮洛芬

Apoptosis; COX; MRP Apoptosis; Immunology/Inflammation; Neuroscience
Ketoprofen (RP-19583) 是一种非甾体抗炎剂,能够有效地抑制COX 的活性,在人血单核细胞中,对 COX-1 和 COX-2 的IC50值分别为 2 nM 和 26 nM。
T11655 Indomethacin-D4

Indometacin-D4,吲哚美辛-D4

CDK Cell Cycle/Checkpoint
Indomethacin-D4 is a deuterium labeled Indomethacin. Indomethacin is a potent and nonselective inhibitor of COX1 and COX2, with IC50s of 18 nM and 26 nM for human COX-1 and COX-2, respectively, in CHO cells.
T61606 Indomethacin sodium

Indomethacin sodium, a powerful and orally active inhibitor of COX1/2, exhibits IC50 values of 18 nM and 26 nM for COX-1 and COX-2, respectively. Apart from its potent anti-inflammatory effects, this compound possesses notable anticancer and anti-infective activities. Since it has such versatile attributes, it finds useful applicability in cancer, inflammation, and viral infection research [1] [2] [3].

化合物

COX-2-IN-26
Cat.No: T63480
Synonym:
Target:
Rofecoxib
Cat.No: T1185
Synonym: MK 966,罗非昔布,罗非考昔,MK-0966
Target: COX
Ketoprofen
Cat.No: T0839
Synonym: 酮基布洛芬,RP-19583,酮洛芬
Target: Apoptosis, COX, MRP
Indomethacin-D4
Cat.No: T11655
Synonym: Indometacin-D4,吲哚美辛-D4
Target: CDK
Indomethacin sodium
Cat.No: T61606
Synonym:
Target:
TargetMol Loading
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