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Cat. No.	Product Name	Target	Signaling Pathways
T10708	CCR1 antagonist 6	CCR	Immunology/Inflammation; Microbiology/Virology
	CCR1 antagonist 6是一种 CCR1 拮抗剂（IC50 ：3 nM）。
T15253	CCX354 CCR1 antagonist 1,CCX-354,CCX 354	CCR	Immunology/Inflammation; Microbiology/Virology
	CCX354 (CCR1 antagonist 1) 是一种有效的小分子 CCR1 拮抗剂，具有抗炎活性，可用于治疗类风湿关节炎。
T30258	AZD-4818 CCR1 antagonist	CCR	Immunology/Inflammation; Microbiology/Virology
	AZD-4818 (CCR1 antagonist) 是趋化因子CCR1的一种拮抗剂，可用于研究慢性阻塞性肺病。
T77349	CCR1/5/8 activator 1	Phospholipase	Metabolism
	CCR1/5/8 activator 1 是胞质磷脂酶 A 抑制剂，具有抗真菌活性。
T10709	CCR1 antagonist 7	CCR	Immunology/Inflammation; Microbiology/Virology
	CCR1 antagonist 7 (compound 16r) 是CCR1的拮抗剂，IC50值为 4 nM。
T14899	CCR1 antagonist 8	CCR	Immunology/Inflammation; Microbiology/Virology
	CCR1 antagonist 8, a third azaindazole series compound, is a CCR1 antagonist (IC50: 1.8 nM in Ca2+ flux assay).
T10710	CCR1 antagonist 9	CCR	Immunology/Inflammation; Microbiology/Virology
	CCR1 antagonist 9 is an effective and selective CCR1 antagonist (IC50: 6.8 nM in calcium flux assay).
T28072	MLN-3897 AVE9897,AVE 9897,CCR1 antagonist 10,AVE-9897	CCR	Immunology/Inflammation; Microbiology/Virology
	MLN-3897 (CCR1 antagonist 10) 是一种具有口服活性的 CCR1 拮抗剂，对于 125I-MIP-1α 与 THP-1 细胞膜的结合，Ki 为 2.3 nM。 MLN-3897 抑制 Akt 信号转导和 MM 细胞存活和增殖。
T64242	CCR1 antagonist 11 hydrochloride
	CCR1 antagonist 11 hydrochloride (A1B1) 是一种口服具有活力的 CCR1 拮抗剂，能够作用于 hCCR1 (IC50: 0/。03 μM)、mCCR1 (IC50: 0.58 μM)、rCCR1 (IC50: 0.32 μM)。CCR1 antagonist 11 hydrochloride 能够用于研究类风湿性关节炎等相关炎症性疾病。
T11699	J-113863	CCR	Immunology/Inflammation; Microbiology/Virology
	J-113863 是选择性的 CCR1 (CD18)拮抗剂，有抗炎作用，对人和小鼠 CCR1受体的 IC50值分别为 0.9 和 5.8 nM。它是人 CCR3的强效拮抗剂，还是小鼠 CCR3的弱效拮抗剂，IC50分别为 0.58 和 460 nM。
T2375	BX471 BX 471,BX-471,ZK-811752	CCR	Immunology/Inflammation; Microbiology/Virology
	BX471 (BX 471) 是可口服的非多肽 CCR1选择性拮抗剂，Ki 值为 1 nM，对其选择性是对 CCR2、CCR5 和 CXCR4 的 250 倍。
T26861	BMS-817399 BMS817399	CCR	Immunology/Inflammation; Microbiology/Virology
	BMS-817399 是一种具有口服活性的 CCR1 拮抗剂，具有结合亲和力和趋化性抑制效力的 IC50，可用于类风湿性关节炎的研究。
T28072L	MLN-3897 TFA MLN-3897 TFA(1010731-97-1 Free base)	CCR	Immunology/Inflammation; Microbiology/Virology
	MLN-3897 TFA 是一种有效的CCR1 拮抗剂，对 125I-MIP-1α 与 THP-1 细胞膜的结合具有抑制作用。
TQ0283	RS102895	CCR	Immunology/Inflammation; Microbiology/Virology
	RS102895 是一种CCR2拮抗剂，IC50值为 360 nM。
T5384	RS 504393	CCR	Immunology/Inflammation; Microbiology/Virology
	RS 504393 是一种高度选择性的 CCR2 趋化因子受体拮抗剂，作用于人重组 CCR2 和 CCR1 受体，IC50值分别为 89 nM 和大于 100 μM。
T3188	RE-640	CCR; Parasite	Immunology/Inflammation; Microbiology/Virology
	NSC-5844 (RE-640) 是 4-氨基喹啉衍生物，起抗肿瘤和抗疟疾作用。
T14845	BX471 hydrochloride ZK-811752 hydrochloride	Others	Others
	BX471 hydrochloride (ZK-811752 hydrochloride) is a potent, selective non-peptide CCR1 antagonist (Ki: 1 nM for human CCR1). It shows 250-fold selectivity for CCR1 over CCR2, CCR5, and CXCR4.
T23492	UCB 35625	Others	Others
	chemokine CCR1 and CCR3 receptor antagonist
T26849	BMS-457
	BMS-457 is a potent, CCR1-selective antagonist.
T68427	MLN-3897 citrate
	MLN-3897 citrate is a C-C Motif Chemokine Receptor 1 (CCR1) antagonist potentially for the treatment of multiple sclerosis and rheumatoid arthritis.
T31061	CP-481715 CP 481,715,CP-481,715,CP481715,CP481,715
	CP 481715 is an effective selective CCR1 antagonist with potential therapeutic significance for inflammatory diseases.
T73371	BAY-3153
	BAY-3153 是一种选择性的 CCR1(C-C motifchemokine receptor1) 拮抗剂 (humanIC50=3 nM ; ratIC50=11 nM ; miceIC50=81 nM)。
T71905	BX-513 HCl
	BX-513 HCl is a selective CCR1 receptor antagonist.
T12773	RS102895 hydrochloride RS102895盐酸盐	Others; 5-HT Receptor; CCR	GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience; Others
	RS102895 hydrochloride 是一种CCR2拮抗剂，IC50值为 360 nM。
T41016	Vercirnon sodium GSK-1605786 sodium,CCX282-Bsodium,维塞诺钠盐,Traficet-ENsodium
	Vercirnon (GSK1605786A) sodium is an orally bioavailable, selective, and potent antagonist of CCR9 . Vercirnon sodium inhibits CCR9-mediated Ca 2+ mobilization and chemotaxis on Molt-4 cells with IC 50 values of 5.4 and 3.4 nM, respectively. Vercirnon sodium is selective for CCR9 over CCR1-12 and CX3CR1-7 (IC 50 s>10 μM for all). Vercirnon sodium is an equipotent inhibitor of CCL25-directed chemotaxis of both splice forms of CCR9 (CCR9A and CCR9B) with IC 50 values of 2.8 and 2.6 nM, respectivel...
T17274	YM022	CCR	Immunology/Inflammation; Microbiology/Virology
	YM022 is a highly effective and selective gastrin/cholecystokinin (CCK)-B receptor antagonist. YM022 can inhibit gastrin-induced gastric acid secretion and histidine decarboxylase activation in vivo. YM022 shows the Ki values of 68 pM and 63 nM for CCK-B and CCK-A receptor, respectively.

化合物

CCR1 antagonist 6

Cat.No: T10708

Target: CCR

Cat.No: T15253

Synonym: CCR1 antagonist 1,CCX-354,CCX 354

Target: CCR

Cat.No: T30258

Synonym: CCR1 antagonist

Target: CCR

CCR1/5/8 activator 1

Cat.No: T77349

Target: Phospholipase

CCR1 antagonist 7

Cat.No: T10709

Target: CCR

CCR1 antagonist 8

Cat.No: T14899

Target: CCR

CCR1 antagonist 9

Cat.No: T10710

Target: CCR

Cat.No: T28072

Synonym: AVE9897,AVE 9897,CCR1 antagonist 10,AVE-9897

Target: CCR

CCR1 antagonist 11 hydrochloride

Cat.No: T64242

Cat.No: T11699

Target: CCR

Cat.No: T2375

Synonym: BX 471,BX-471,ZK-811752

Target: CCR

Cat.No: T26861

Synonym: BMS817399

Target: CCR

Cat.No: T28072L

Synonym: MLN-3897 TFA(1010731-97-1 Free base)

Target: CCR

Cat.No: TQ0283

Target: CCR

Cat.No: T5384

Target: CCR

Cat.No: T3188

Target: CCR, Parasite

BX471 hydrochloride

Cat.No: T14845

Synonym: ZK-811752 hydrochloride

Target: Others

Cat.No: T23492

Target: Others

Cat.No: T26849

MLN-3897 citrate

Cat.No: T68427

Cat.No: T31061

Synonym: CP 481,715,CP-481,715,CP481715,CP481,715

Cat.No: T73371

Cat.No: T71905

RS102895 hydrochloride

Cat.No: T12773

Synonym: RS102895盐酸盐

Target: Others, 5-HT Receptor, CCR

Vercirnon sodium

Cat.No: T41016

Synonym: GSK-1605786 sodium,CCX282-Bsodium,维塞诺钠盐,Traficet-ENsodium

Cat.No: T17274

Target: CCR

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