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Cat. No.	Product Name	Target	Signaling Pathways
T12404	CCK-A receptor inhibitor 1	cholecystokinin	GPCR/G Protein
	CCK-A receptor inhibitor 1 是一种有效的缩胆囊素 A (CCK-A) 受体抑制剂(IC50：340 nM）。CCK-A receptor inhibitor 1 可用于研究与消化系统相关的疾病。
T1052	Proglumide 二丙谷酰胺	cholecystokinin	GPCR/G Protein
	Proglumide (Binoside) 是一种非肽的、口服具有活性的胆囊收缩素(CCK)-A/B 受体拮抗剂。它能够选择性阻断 CCK 在中枢神经系统中的作用。它能够抑制胃分泌，具有保护胃十二指肠粘膜的能力，并表现出抗癫痫和抗氧化活性。
T13260	Gastrin/CCK antagonist 1	cholecystokinin	GPCR/G Protein
	Gastrin/CCK antagonist 1 是一种有效的 gastrin/CCK 拮抗剂，可用于研究代谢系统相关疾病。
TP2204L	CCK Octapeptide, non-sulfated acetate CCK Octapeptide, non-sulfated acetate(25679-24-7 Free base)	cholecystokinin	GPCR/G Protein
	CCK Octapeptide, non-sulfated acetate 是一种合成的胆囊收缩素脱硫酸肽。
TP2419	V-9-M Cholecystokinin nonapeptide V 9 M,Prepro CCK Fragment V-9-M,Val-pro-val-glu-ala-val-asp-pro-met,Cholecystokinin Precursor (24-32),V9M,V-9-M	Beta Amyloid	Neuroscience
	V-9-M Cholecystokinin nonapeptide (Prepro CCK Fragment V-9-M) 是胆囊收缩素(CCK)的前体化合物。胆囊收缩素(CCK)是一种刺激胆囊收缩和胰腺外分泌的脑肠肽，可从狗和猫的小肠中提取的，可以引起胆囊收缩。
T9343	N-Cbz-DL-tryptophan	cholecystokinin	GPCR/G Protein
	N-Cbz-DL-tryptophan 是一种胆囊收缩素受体拮抗剂，可消除离体心脏对 CCK-8 的反应。
T9991	WAY-620645	cholecystokinin	GPCR/G Protein
	WAY-620645 是一种 CCK 拮抗剂，具有抗肿瘤和镇痛活性。
TP1198	Sincalide ammonium SQ19844 ammonium,CCK-8 ammonium,Cholecystokinin octapeptide ammonium	cholecystokinin	GPCR/G Protein
	Sincalide ammonium (CCK-8 ammonium) 是一种有效的氨基酸多肽激素胆囊收缩素 (CCK) 的类似物，是保留了 CCK 的大部分生物活性的活性片段。Sincalide ammonium 促进胆汁的分泌，使胆囊收缩并使 Oddi 的括约肌松弛，从而促进胆汁排入十二指肠。Sincalide ammonium 可通过注射促进胆囊收缩，常用于辅助诊断胆囊、胰腺疾病和胆囊造影术。
TP2500	Cholecystokinin (26-33) free acid CCK (26-33) free acid	cholecystokinin	GPCR/G Protein
	Cholecystokinin (26-33) free acid 是胆囊收缩素 (CCK) 的一部分，是脊椎动物中枢神经系统中存在的 CCKB 型受体的高选择性配体，可诱导大鼠轻度味觉厌恶条件反射。
TQ0062	Nastorazepide Z-360	cholecystokinin	GPCR/G Protein
	Nastorazepide 是一种选择性的、口服有效的1,5-苯并二氮杂环衍生物胃泌素/胆囊收缩素2（CCK-2）受体拮抗剂，具有抗肿瘤的潜能。
TP1197	Sincalide SQ19844,辛卡利特,CCK-8,Cholecystokinin octapeptide	Others	Others
	Sincalide (CCK-8) 是一种速效的胆囊收缩素的氨基酸多肽激素类似物，可在胆囊造影术中静脉使用。它的肝胆生理作用是增加胆汁的分泌，使胆囊收缩并使 Oddi 的括约肌松弛，从而使胆汁排入十二指肠。它是一种通过注射促进胆囊收缩并帮助诊断胆囊和胰腺疾病的药物。
TP1931L1	[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate(96736-12-8 free base)	cholecystokinin	GPCR/G Protein
	[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate ([D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate (96736-12-8 free base)) 是广谱神经肽反向激动剂和拮抗剂。 ghrelin 受体的强效完全反向激动剂(EC50 = 5.2 nM)；减少组成型生长素释放肽受体信号传导。它也是速激肽、缓激肽、CCK 和铃蟾肽受体的拮抗剂。在体外诱导细胞凋亡并抑制癌细胞生长。
T16906	Sograzepide YM-220,Netazepide,YF 476	Others	Others
	Sograzepide is an effective and highly selective Gastrin/CCK-B antagonist (IC50: 0.1 nM), has an inhibitory effect on Gastrin/CCK-A activity (IC50: 502 nM). Sograzepide replaces the specific binding of [125I]CCK-8 to the rat brain, cloned canine, and cloned human Gastrin/CCK-B receptors (Ki: 0.068, 0.62 and 0.19 nM, respectively).
T10707	CCK-B Receptor Antagonist 2	Others	Others
	CCK-B Receptor Antagonist 2 is a potent and orally active antagonist of Gastrin/CCK-B (IC50: 0.43 nM). It also inhibits gastrin/CCK-A activity (IC50: 1.82 μM).
T10055	(Iso)-FK-480 CHEMBL333994	cholecystokinin	GPCR/G Protein
	(Iso)-FK-480 是一种新型可口服的胆囊收缩素 A（CCK-A）拮抗剂，可用于研究治疗慢性胰腺炎。
T25921	Pbc 264 Pbc264,Pbc-264
	Pbc 264 is a CCK agonist.
T24287	L 365031 L 365,031,L365031,L-365,031,L-365031,L365,031
	L 365031 is a CCK antagonist.
T37205	CCK (26-31) (sulfated)
	CCK (26-31) is an N-terminal fragment of CCK , a peptide hormone found in the intestine and brain that stimulates digestion, mediates satiety, and is involved in anxiety. The sulfated form of CCK (26-31) inhibits binding of [125I]CCK-33 to guinea pig cortical membranes by 21% when used at a concentration of 0.1 mM.
T25139	BC 197 Boc-asp-tyr(SO3H)-ahx-lys-trp-ahx-asp-phe-NH2,BC197,BC-197
	BC 197 is a selective CCK-B agonist.
T26483	A-65186 A65186
	A 65186 is a Type A Cholecystokinin (CCK) receptor antagonist.
T37203	CCK (26-30) (sulfated)
	CCK (26-30) is an N-terminal fragment of CCK , a peptide hormone found in the intestine and brain that stimulates digestion, mediates satiety, and is involved in anxiety. The sulfated form of CCK (26-30) inhibits binding of [125I]CCK-33 to guinea pig cortical membranes by 10% when used at a concentration of 0.1 mM.
T13261	CCK-B Receptor Antagonist 1	Others	Others
	CCK-B Receptor Antagonist 1 is a cholecystokinin B (CCK-B) receptor agonist and has the potential of reducing the secretion of gastric acid.
T26484	A71378 A-71378,A 71378
	A71378 is a high potency, selectivity CCK-A receptors agonist.
T25108	ARL 15849XX ARL15849XX,FPL15849,FPL-15849,FPL 15849,ARL-15849XX
	ARL 15849XX, a CCK-8 analog, is a novel anti-obesity agent.
T13084	Tarazepide	Others	Others
	Tarazepide is a potent and specific antagonist of CCK-A receptor.
T34669	Snf 8906 Snf-8906,Snf8906
	Snf 8906 is a CCK-8 analog.
T29502	A 70874 A-70874,A70874
	A70874 has high selectivity and potency for cholecystokinin (CCK) a receptor.
T27014	CI-1015 CI1015,CI 1015,PD 144598
	CI-1015 is a CCK-B receptor antagonist with oral activity.
T37204	CCK (26-31) (non-sulfated)
	CCK (26-31) is an N-terminal fragment of CCK , a peptide hormone found in the intestine and brain that stimulates digestion, mediates satiety, and is involved in anxiety.
T82732	Cholecystokinin (1-21) CCK-1-21
	Cholecystokinin (1-21)，作为一种胆囊收缩素 (CCK) 片段，能够激活人体脂肪组织的脂肪分解作用。
T28342	PD-149164 PD 149164,PD149164
	PD-149164 is an agonist of the CCK-A receptor.
T23886	Cholecystokinin (27-32)-amide Cholecystokinin (27-32)-NH2
	Cholecystokinin (27-32)-amide is a CCK receptor antagonist.
T32425	Ksg 504 Ksg504,Ksg-504
	Ksg 504 has superior selectivity and affinity to CCK-A receptors and derived from proglumide.
T27900	LY 219057 LY-219057,LY219057
	LY 219057 is a potent, competitive, and specific antagonist of CCK receptor on the exocrine pancreas.
T15101	Devazepide L-364,718,地伐西匹,MK-329	Others	Others
	Devazepide is a competitive and orally active nonpeptide antagonist of cholecystokinin (CCK) receptor (IC50s: 81 pM, 45 pM, and 245 nM for rat pancreatic, bovine gallbladder and guinea pig brain CCK receptors, respectively).
T23946	DA-3934 UNII-J353803KRG
	DA-3934 has a high affinity for gastrin/CCK-B receptors and high selectivity over CCK-A receptors. DA-3934 and its methyl ester derivative inhibited pentagastrin-induced gastric acid secretion in rats in a dose-dependent manner.
T32297	Jmv 180 Cck-jmv-180,Jmv-180,Jmv180
	Jmv 180, a CCK analog, can distinguish high-affinity cholecystokinin receptors from low-affinity cholecystokinin receptors.
T25437	Fpl 14294 Fpl-14294,Fpl14294
	Fpl 14294 is a novel CCK-8 agonist with effective intranasal anorectic activity in the rat.
T37206	CCK (27-33) (non-sulfated)
	CCK (27-33) is a C-terminal fragment of CCK , a peptide hormone found in the intestine and brain that stimulates digestion, mediates satiety, and is involved in anxiety. Non-sulfated CCK (27-33) inhibits binding of [3H]naloxone in rat cerebellum membranes (IC50 = 4 uM) and inhibits electrically-stimulated contraction of isolated guinea pig ileum (IC50 = 17 uM), an effect that can be reversed by naloxone. Unlike sulfated CCK (27-33), the non-sulfated form does not reduce exploratory behavior in m...
T39170	Cholecystokinin Octapeptide, desulfated TFA CCK Octapeptide, desulfated TFA,Cholecystokinin Octapeptide, desulfated TFA
	Cholecystokinin Octapeptide, desulfated TFA, is a synthetic octapeptide derived from Cholecystokinin (CCK) that has undergone desulfation.
T62039	L-365260 hemihydrate
	L-365260 hemihydrate 是选择性的、具有口服活性的非肽胃泌素和脑胆囊收缩素受体 (CCK-B) 拮抗剂，Kis 值分别为 1.9 nM 和 2.0 nM。L-365260 hemihydrate 以竞争性方式与豚鼠胃泌素和脑 CCK 受体相互作用。
T25553	Jmv 332 Jmv-332,Jmv332
	Jmv 332 is a cyclic analog of the C-terminal hexapeptide of CCK. It is a CCK/gastrin receptor agonist.
T27774	L-740093 L 740093
	L-740093 is a specific antagonist of CCK-B receptor.
T17274	YM022	CCR	Immunology/Inflammation; Microbiology/Virology
	YM022 is a highly effective and selective gastrin/cholecystokinin (CCK)-B receptor antagonist. YM022 can inhibit gastrin-induced gastric acid secretion and histidine decarboxylase activation in vivo. YM022 shows the Ki values of 68 pM and 63 nM for CCK-B and CCK-A receptor, respectively.
T28331	PD 136450 Cam1189,PD136450,Cam-1189,PD-136450,Cam 1189
	Cholecystokinin type B receptor antagonist PD-136,450 is a partial secretory agonist in the stomach and a full agonist in the pancreas of the rat. Gastrin (cholecystokinin type B (CCK-B)) receptor antagonists may help to elucidate the physiological role o
T15105	Dexloxiglumide	Others	Others
	Dexloxiglumide, an active enantiomer of Loxiglumide, inhibits smooth muscle cell contractions induced by cholecystokinin-octapeptide (CCK-8). It is a selective antagonist of cholecystokinin type A (CCKA) receptors.
T26482	A-57696
	A-57696 is a cholecystokinin antagonist with selective for cortical CCK-B receptors (IC50 = 25 nM).
T25550	Jmv 176 Jmv-176,Jmv176,Boc-tyr(SO3)-nle-psi-(coch2)-gly-trp-nle-asp-phe-NH2
	Jmv 176 is a CCK agonist when first given and becomes a cholecystokinin antagonist after 3-4 hours.
T27772	L-736380 L-736,380,L 736380,L736,380,L 736,380
	L-736380 is a CCK-B receptor antagonist. L-736,380 dose-dependently inhibited gastric acid secretion in anesthetized rats (ID(50), 0.064 mg/kg) and ex vivo binding of [(125)I]CCK-8S in BKTO mice brain membranes (ED(50), 1.7 mg/kg).
T12544	Proglumide hemicalcium	Others	Others
	Proglumide hemicalcium is a antagonist of nonpeptide and orally active cholecystokinin (CCK)-A/B receptors, has antiepileptic and antioxidant activities.

化合物

CCK-A receptor inhibitor 1

Cat.No: T12404

Target: cholecystokinin

Cat.No: T1052

Synonym: 二丙谷酰胺

Target: cholecystokinin

Gastrin/CCK antagonist 1

Cat.No: T13260

Target: cholecystokinin

CCK Octapeptide, non-sulfated acetate

Cat.No: TP2204L

Synonym: CCK Octapeptide, non-sulfated acetate(25679-24-7 Free base)

Target: cholecystokinin

V-9-M Cholecystokinin nonapeptide

Cat.No: TP2419

Synonym: V 9 M,Prepro CCK Fragment V-9-M,Val-pro-val-glu-ala-val-asp-pro-met,Cholecystokinin Precursor (24-32),V9M,V-9-M

Target: Beta Amyloid

N-Cbz-DL-tryptophan

Cat.No: T9343

Target: cholecystokinin

Cat.No: T9991

Target: cholecystokinin

Sincalide ammonium

Cat.No: TP1198

Synonym: SQ19844 ammonium,CCK-8 ammonium,Cholecystokinin octapeptide ammonium

Target: cholecystokinin

Cholecystokinin (26-33) free acid

Cat.No: TP2500

Synonym: CCK (26-33) free acid

Target: cholecystokinin

Cat.No: TQ0062

Synonym: Z-360

Target: cholecystokinin

Cat.No: TP1197

Synonym: SQ19844,辛卡利特,CCK-8,Cholecystokinin octapeptide

Target: Others

[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate

Cat.No: TP1931L1

Synonym: [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate(96736-12-8 free base)

Target: cholecystokinin

Cat.No: T16906

Synonym: YM-220,Netazepide,YF 476

Target: Others

CCK-B Receptor Antagonist 2

Cat.No: T10707

Target: Others

Cat.No: T10055

Synonym: CHEMBL333994

Target: cholecystokinin

Cat.No: T25921

Synonym: Pbc264,Pbc-264

Cat.No: T24287

Synonym: L 365,031,L365031,L-365,031,L-365031,L365,031

CCK (26-31) (sulfated)

Cat.No: T37205

Cat.No: T25139

Synonym: Boc-asp-tyr(SO3H)-ahx-lys-trp-ahx-asp-phe-NH2,BC197,BC-197

Cat.No: T26483

Synonym: A65186

CCK (26-30) (sulfated)

Cat.No: T37203

CCK-B Receptor Antagonist 1

Cat.No: T13261

Target: Others

Cat.No: T26484

Synonym: A-71378,A 71378

Cat.No: T25108

Synonym: ARL15849XX,FPL15849,FPL-15849,FPL 15849,ARL-15849XX

Cat.No: T13084

Target: Others

Cat.No: T34669

Synonym: Snf-8906,Snf8906

Cat.No: T29502

Synonym: A-70874,A70874

Cat.No: T27014

Synonym: CI1015,CI 1015,PD 144598

CCK (26-31) (non-sulfated)

Cat.No: T37204

Cholecystokinin (1-21)

Cat.No: T82732

Synonym: CCK-1-21

Cat.No: T28342

Synonym: PD 149164,PD149164

Cholecystokinin (27-32)-amide

Cat.No: T23886

Synonym: Cholecystokinin (27-32)-NH2

Cat.No: T32425

Synonym: Ksg504,Ksg-504

Cat.No: T27900

Synonym: LY-219057,LY219057

Cat.No: T15101

Synonym: L-364,718,地伐西匹,MK-329

Target: Others

Cat.No: T23946

Synonym: UNII-J353803KRG

Cat.No: T32297

Synonym: Cck-jmv-180,Jmv-180,Jmv180

Cat.No: T25437

Synonym: Fpl-14294,Fpl14294

CCK (27-33) (non-sulfated)

Cat.No: T37206

Cholecystokinin Octapeptide, desulfated TFA

Cat.No: T39170

Synonym: CCK Octapeptide, desulfated TFA,Cholecystokinin Octapeptide, desulfated TFA

L-365260 hemihydrate

Cat.No: T62039

Cat.No: T25553

Synonym: Jmv-332,Jmv332

Cat.No: T27774

Synonym: L 740093

Cat.No: T17274

Target: CCR

Cat.No: T28331

Synonym: Cam1189,PD136450,Cam-1189,PD-136450,Cam 1189

Cat.No: T15105

Target: Others

Cat.No: T26482

Cat.No: T25550

Synonym: Jmv-176,Jmv176,Boc-tyr(SO3)-nle-psi-(coch2)-gly-trp-nle-asp-phe-NH2

Cat.No: T27772

Synonym: L-736,380,L 736380,L736,380,L 736,380

Proglumide hemicalcium

Cat.No: T12544

Target: Others

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