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12

抑制剂 & 化合物

3

天然产物

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Cat. No. Product Name Target Signaling Pathways
T4990 Cefcapene pivoxil hydrochloride hydrate

Cefcapene Pivoxil Hydrochloride,盐酸头孢卡品酯

Antibacterial; Antibiotic Microbiology/Virology
Cefcapene pivoxil hydrochloride hydrate 是一种头孢菌素的前药,具有口服活性和广谱抗菌活性。它可研究掌跖脓疱病等感染性疾病。
T3497 Ocaperidone

奥卡哌酮,Ocaperidona,R79598

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Ocaperidone (Ocaperidona) 是5-HT2和多巴胺D2的拮抗剂,也是5-HT1A 的激动剂,有安定作用。
T68035 Capeserod

SL-650155,SL-65.0155

5-HT Receptor GPCR/G Protein; Neuroscience
Capeserod 是一种潜在的 5-HT4 receptor(5-羟色胺受体4)激动剂,可用于研究消化系统疾病和神经系统疾病。
T1408 Capecitabine

Xeloda,卡培他滨,Capecitibine,Capiibine,RO 09-1978

Apoptosis; Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Capecitabine (Capecitibine) 是一种可口服的前药,可由胸苷磷酸化酶催化转变为其活性代谢物 Fluorouracil。
T64318 Capecitabine-2',3'-cyclic Carbonate

Others Others
Capecitabine-2',3'-cyclic Carbonate 是一种抗增殖化合物。
TP2385 Ige decapeptide

Immunoglobulin E decapeptide

Ige decapeptide is a peptide.
TP2362 Acetyl decapeptide-3

Rejuline,Ac-tyr-arg-ser-arg-lys-tyr-thr-ser-trp-tyr-NH2

Acetyl decapeptide-3 is a peptide that can stimulate collagen and elastin to increase skin elasticity and increase cell growth and improve healing and repair.
T37371 4(Z),7(Z),10(Z),13(Z),16(Z)-Nonadecapentaenoic Acid

4(Z),7(Z),10(Z),13(Z),16(Z)-Nonadecapentaenoic acid is an unusual polyunsaturated fatty acid (PUFA) generated during the synthesis of docosahexaenoic acid-d5 . While the physiological properties of this compound are not known, dietary intake of n-3 long-chain PUFAs provides potential health benefits.
T68149 tacapenem

Tacapenem 是一种β-内酰胺类抗菌剂。它具有广谱抗菌活性,对β-内酰胺酶具有很高的稳定性。
T131540 Capensin

Capensin 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T131540。
T75714 Decapeptide-12

Decapeptide-12,一个小型寡肽,作为tyrosinase的抑制剂,通过与tyrosinase的C末端残基相互作用(Kd: 61.1 μM)发挥作用。作为mushroom tyrosinase的竞争性抑制剂(IC50: 40 µM),Decapeptide-12有效上调SIRT的转录水平,并能减少黑色素细胞中的黑色素含量,适用于黑色素生成、衰老和炎症的研究。
T26944 Capeserod HCl

SL-65.0155,SL-650155,SL 650155,SL 65.0155

Capeserod HCl, a 5-hydroxytriptamine 4 (5-HT4) receptor agonist, is used potentially for the treatment of Alzheimer's disease.

化合物

Cefcapene pivoxil hydrochloride hydrate
Cat.No: T4990
Synonym: Cefcapene Pivoxil Hydrochloride,盐酸头孢卡品酯
Target: Antibacterial, Antibiotic
Ocaperidone
Cat.No: T3497
Synonym: 奥卡哌酮,Ocaperidona,R79598
Target: Dopamine Receptor, 5-HT Receptor
Capeserod
Cat.No: T68035
Synonym: SL-650155,SL-65.0155
Target: 5-HT Receptor
Capecitabine
Cat.No: T1408
Synonym: Xeloda,卡培他滨,Capecitibine,Capiibine,RO 09-1978
Target: Apoptosis, Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis
Capecitabine-2',3'-cyclic Carbonate
Cat.No: T64318
Synonym:
Target: Others
Ige decapeptide
Cat.No: TP2385
Synonym: Immunoglobulin E decapeptide
Target:
Acetyl decapeptide-3
Cat.No: TP2362
Synonym: Rejuline,Ac-tyr-arg-ser-arg-lys-tyr-thr-ser-trp-tyr-NH2
Target:
4(Z),7(Z),10(Z),13(Z),16(Z)-Nonadecapentaenoic Acid
Cat.No: T37371
Synonym:
Target:
tacapenem
Cat.No: T68149
Synonym:
Target:
Capensin
Cat.No: T131540
Synonym:
Target:
Decapeptide-12
Cat.No: T75714
Synonym:
Target:
Capeserod HCl
Cat.No: T26944
Synonym: SL-65.0155,SL-650155,SL 650155,SL 65.0155
Target:
Cat. No. Product Name Target Signaling Pathways
T6429 Caffeic Acid Phenethyl Ester

Phenylethyl Caffeate,咖啡酸苯乙酯,CAPE

Apoptosis; NF-κB Apoptosis; NF-κB
Caffeic Acid Phenethyl Ester (Phenylethyl Caffeate) 是咖啡酸的苯乙醇酯,是蜂巢蜂胶的生物活性成分。它抑制核转录因子 NF-kappa B 的激活,具有抗肿瘤、细胞保护和免疫调节活性。它抑制 PDGF 诱导的血管平滑肌细胞增殖。
T83660 3(Z),6(Z),9(Z),12(Z),15(Z)-Octadecapentaenoic Acid

C18:5 n-3,C18:5(3Z,6Z,9Z,12Z,15Z),all-cis-3,6,9,12,15-Octadecapentaenoic Acid

3(Z),6(Z),9(Z),12(Z),15(Z)-Octadecapentaenoic acid 是一种在 G. kowalevskii 中发现的微藻 PUFA,常作为微藻和甲藻的化学分类生物标志物使用。
TN4338 Isovouacapenol C

Others Others
Isovouacapenol C是一种天然产物,属于豆科云实属,其产品编号为 TN4338,CAS号为 455255-15-9。Isovouacapenol C可用作对照参考。

天然产物

Caffeic Acid Phenethyl Ester
Cat.No: T6429
Synonym: Phenylethyl Caffeate,咖啡酸苯乙酯,CAPE
Target: Apoptosis, NF-κB
3(Z),6(Z),9(Z),12(Z),15(Z)-Octadecapentaenoic Acid
Cat.No: T83660
Synonym: C18:5 n-3,C18:5(3Z,6Z,9Z,12Z,15Z),all-cis-3,6,9,12,15-Octadecapentaenoic Acid
Target:
Isovouacapenol C
Cat.No: TN4338
Synonym:
Target: Others
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