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6
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T131543 | Gamabufotalin (Gamabufagin; Gamabufogenin) | ||
Gamabufotalin (Gamabufagin; Gamabufogenin) 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T131543。 | |||
T124283 |
5beta-Hydroxybufotalin
|
||
5beta-Hydroxybufotalin 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124283。 | |||
T10116 | 3-O-Acetylbufotalin | Others | Others |
3-O-Acetylbufotalin is a derivate of bufadienolide with anti-cancer activity. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5A2461 |
Bufotalin
蟾蜍他灵,Bufotaline,蟾毒它灵,蟾蜍他灵 |
Apoptosis; Others; Reactive Oxygen Species | Apoptosis; Immunology/Inflammation; Metabolism; NF-κB; Others |
Bufotalin (Bufotaline) 是一种从蟾酥中分离的类固醇内酯,可诱导癌细胞凋亡,也诱导内质网应激的激活,具有强大的抗肿瘤活性。 | |||
T4A2399 |
Cinobufotalin
华蟾毒它灵,华蟾素 |
IL Receptor; Akt; MRP; P-gp | Cytoskeletal Signaling; Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience; PI3K/Akt/mTOR signaling |
Cinobufotalin 是一种从蟾蜍的皮肤分泌物中提取的强心类固醇或丁二烯内酯。它已被用作强心药,利尿药和止血药,也是潜在的抗肺癌药物。 | |||
T4A2456 |
Gamabufotalin
Gamabufagin,日本蟾蜍毒苷元 |
COX | Immunology/Inflammation; Neuroscience |
Gamabufotalin (Gamabufagin) 是一种蟾蜍甾烯,存在于蟾酥中。它稳定性高,毒性低,被广泛用于癌症的研究。 | |||
T83282 |
5β-Hydroxybufotalin
|
||
5β-Hydroxybufotalin (化合物 6) 是一种来源于中药蟾酥的天然产物,具有有效的抗癌作用,能够抑制癌细胞的生长活性。 | |||
TN1200 |
19-Oxocinobufotalin
|
Others | Others |
19-Oxocinobufotalin 3-adipoylarginine ester shows significant inhibition effect against human hepatocellular carcinoma cell line SMMC-7721 in vitro. | |||
TN1572 |
Desacetylcinobufotalin
|
Others | Others |
Desacetylcinobufotalin has significant antitumor activity through induction apoptosis via mitochondria pathway, it also shows potent cytotoxic activities against HL-60 cell lines. |