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3

抑制剂 & 化合物

6

天然产物

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Cat. No. Product Name Target Signaling Pathways
T131543 Gamabufotalin (Gamabufagin; Gamabufogenin)

Gamabufotalin (Gamabufagin; Gamabufogenin) 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T131543。
T124283 5beta-Hydroxybufotalin

5beta-Hydroxybufotalin 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124283。
T10116 3-O-Acetylbufotalin

Others Others
3-O-Acetylbufotalin is a derivate of bufadienolide with anti-cancer activity.

化合物

Gamabufotalin (Gamabufagin; Gamabufogenin)
Cat.No: T131543
Synonym:
Target:
5beta-Hydroxybufotalin
Cat.No: T124283
Synonym:
Target:
3-O-Acetylbufotalin
Cat.No: T10116
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T5A2461 Bufotalin

蟾蜍他灵,Bufotaline,蟾毒它灵,蟾蜍他灵

Apoptosis; Others; Reactive Oxygen Species Apoptosis; Immunology/Inflammation; Metabolism; NF-κB; Others
Bufotalin (Bufotaline) 是一种从蟾酥中分离的类固醇内酯,可诱导癌细胞凋亡,也诱导内质网应激的激活,具有强大的抗肿瘤活性。
T4A2399 Cinobufotalin

华蟾毒它灵,华蟾素

IL Receptor; Akt; MRP; P-gp Cytoskeletal Signaling; Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience; PI3K/Akt/mTOR signaling
Cinobufotalin 是一种从蟾蜍的皮肤分泌物中提取的强心类固醇或丁二烯内酯。它已被用作强心药,利尿药和止血药,也是潜在的抗肺癌药物。
T4A2456 Gamabufotalin

Gamabufagin,日本蟾蜍毒苷元

COX Immunology/Inflammation; Neuroscience
Gamabufotalin (Gamabufagin) 是一种蟾蜍甾烯,存在于蟾酥中。它稳定性高,毒性低,被广泛用于癌症的研究。
T83282 5β-Hydroxybufotalin

5β-Hydroxybufotalin (化合物 6) 是一种来源于中药蟾酥的天然产物,具有有效的抗癌作用,能够抑制癌细胞的生长活性。
TN1200 19-Oxocinobufotalin

Others Others
19-Oxocinobufotalin 3-adipoylarginine ester shows significant inhibition effect against human hepatocellular carcinoma cell line SMMC-7721 in vitro.
TN1572 Desacetylcinobufotalin

Others Others
Desacetylcinobufotalin has significant antitumor activity through induction apoptosis via mitochondria pathway, it also shows potent cytotoxic activities against HL-60 cell lines.

天然产物

Bufotalin
Cat.No: T5A2461
Synonym: 蟾蜍他灵,Bufotaline,蟾毒它灵,蟾蜍他灵
Target: Apoptosis, Others, Reactive Oxygen Species
Cinobufotalin
Cat.No: T4A2399
Synonym: 华蟾毒它灵,华蟾素
Target: IL Receptor, Akt, MRP, P-gp
Gamabufotalin
Cat.No: T4A2456
Synonym: Gamabufagin,日本蟾蜍毒苷元
Target: COX
5β-Hydroxybufotalin
Cat.No: T83282
Synonym:
Target:
19-Oxocinobufotalin
Cat.No: TN1200
Synonym:
Target: Others
Desacetylcinobufotalin
Cat.No: TN1572
Synonym:
Target: Others
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