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Cat. No. Product Name Target Signaling Pathways
T10486 BCI

(E)-BCI

Phosphatase Metabolism
BCI ((E)-BCI) 是双重特异性磷酸酶的变构抑制剂。它特异性抑制 DUSP6和 DUSP1的 EC50分别为 13.3 和 8.0 μM,但不能够抑制 DUSP5。
T23777 BCI-137

BCI137

Others Others
BCI-137 是 Argonaute 2 配体。它通过靶向 MicroRNA 结合域来发挥作用。
T5322 BCI-121

Histone Methyltransferase Chromatin/Epigenetic
BCI-121是一种底物竞争性 SMYD3 抑制剂,可抑制癌细胞的增殖。
T7323 BCI-215

Phosphatase Metabolism
BCI-215 是高效肿瘤细胞选择性的双重特异性磷酸酶DUSP-MKP 抑制剂。它对肿瘤细胞有细胞毒性,但对正常细胞无毒性。
T11139 (E/Z)-BCI

NSC 150117

Apoptosis; Phosphatase Apoptosis; Metabolism
(E/Z)-BCI (NSC-150117) 是一种DUSP6抑制剂,可通过激活 Nrf2 信号和抑制 NF-κB 通路,减弱 LPS 诱导的巨噬细胞炎症和 ROS 生成,具有抗炎活性。
T10486L BCI hydrochloride

(E)-BCI hydrochloride

Others Others
BCI hydrochloride specifically inhibits DUSP6 and DUSP1 with EC50s of 13.3 and 8.0 μM in cells, respectively. BCI hydrochloride does not inhibit DUSP5. BCI hydrochloride is an allosteric inhibitor of dual specificity phosphatase (DUSP).
T28034 MGS-0039

BCI 632,BCI-632,MGS0039,BCI632

MGS-0039 is a group II metabotropic glutamate receptor (mgluR2/3) antagonist. Antidepressant-like action of group II mGlu receptor antagonists does not depend on serotonergic system activation. However, the AMPA receptor seems to play a key role in the an
T28654 Sabcomeline hydrochloride

BCI224,BRL-55473,BCI-224,CEB-2424,SB-202026A,Sabcomeline HCl

Sabcomeline is a selective M1 receptor partial agonist.
T76844 Abciximab

C7E3

Integrin Cytoskeletal Signaling
Abciximab (C7E3) 是一种小鼠/人嵌合单克隆抗体,是一种有效的糖蛋白 IIb/IIIa (glycoprotein IIb/IIIa) 抑制剂。 Abciximab 具有抗血小板聚集和白细胞粘附的作用,通过与糖蛋白 IIb/IIIa、vitronectin 和 Mac-1 受体结合发挥作用。
T18923 BCIP

5-溴-4-氯-3-吲哚基磷酸酯对甲苯胺盐,BCIP p-toluidine salt,X-phosphate p-toluidine salt

Others Others
BCIP (BCIP p-toluidine salt) 是一种显色底物,可用于碱性磷酸酶活性的比色法检测。
T6415 Bismuth Subcitrate Potassium

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Bismuth subcitrate potassium 是针对 12 种幽门螺杆菌菌株的抗生素,MIC50为 8 μg/ml。它用于幽门螺杆菌感染的上胃肠道疾病的研究。
T31223 DCBCI0901

DCBCI-0901,DCBCI 0901

DCBCI0901 is an inhibitor of phosphatidylinositide 3-kinase (PI3K), raptor-mTOR (mTOR complex 1 or mTORC1) and rictor-mTOR (mTOR complex 2 or mTORC2) with potential antineoplastic activity.

化合物

BCI
Cat.No: T10486
Synonym: (E)-BCI
Target: Phosphatase
BCI-137
Cat.No: T23777
Synonym: BCI137
Target: Others
BCI-121
Cat.No: T5322
Synonym:
Target: Histone Methyltransferase
BCI-215
Cat.No: T7323
Synonym:
Target: Phosphatase
(E/Z)-BCI
Cat.No: T11139
Synonym: NSC 150117
Target: Apoptosis, Phosphatase
BCI hydrochloride
Cat.No: T10486L
Synonym: (E)-BCI hydrochloride
Target: Others
MGS-0039
Cat.No: T28034
Synonym: BCI 632,BCI-632,MGS0039,BCI632
Target:
Sabcomeline hydrochloride
Cat.No: T28654
Synonym: BCI224,BRL-55473,BCI-224,CEB-2424,SB-202026A,Sabcomeline HCl
Target:
Abciximab
Cat.No: T76844
Synonym: C7E3
Target: Integrin
BCIP
Cat.No: T18923
Synonym: 5-溴-4-氯-3-吲哚基磷酸酯对甲苯胺盐,BCIP p-toluidine salt,X-phosphate p-toluidine salt
Target: Others
Bismuth Subcitrate Potassium
Cat.No: T6415
Synonym:
Target: Others, Antibacterial, Antibiotic
DCBCI0901
Cat.No: T31223
Synonym: DCBCI-0901,DCBCI 0901
Target:
TargetMol Loading
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