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4

抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T21454 Nicardipine

Cardene,Dagan,尼卡地平,Antagonil,Flusemide

Calcium Channel Membrane transporter/Ion channel; Metabolism
Nicardipine (Cardene) 是一种二氢吡啶类钙通道阻滞剂,可阻断心脏钙通道,IC50为 1 μM,可用于治疗心绞痛和高血压。
T12633 (R)-Nicardipine

(R)-YC-93 free base

Others Others
(R)-Nicardipine is the less active R enantiomer of Nicardipine. Nicardipine is a blocker of calcium channel(IC50 of 1 μM for blocking cardiac calcium channels).
T1215 Nicardipine hydrochloride

盐酸尼卡地平,RS-69216,Nicardipine HCl,YC-93 Hydrochloride

Calcium Channel; Adrenergic Receptor; AChR; Autophagy Autophagy; GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Neuroscience
Nicardipine hydrochloride (YC-93 Hydrochloride) 是一种钙通道阻滞剂,IC50为 1 μM。它可阻断某些细胞壁中的钙离子并抑制冠状动脉和外周动脉的收缩,从而降低对氧气的需求心肌和减少动脉收缩和痉挛。它在临床上用作脑和冠状血管扩张剂。
T12221 Nicardipine-d3 hydrochloride

盐酸尼卡地平 D3,YC-93 D3

Others Others
Nicardipine D3 hydrochloride is the deuterium labeled Nicardipine hydrochloride.

化合物

Nicardipine
Cat.No: T21454
Synonym: Cardene,Dagan,尼卡地平,Antagonil,Flusemide
Target: Calcium Channel
(R)-Nicardipine
Cat.No: T12633
Synonym: (R)-YC-93 free base
Target: Others
Nicardipine hydrochloride
Cat.No: T1215
Synonym: 盐酸尼卡地平,RS-69216,Nicardipine HCl,YC-93 Hydrochloride
Target: Calcium Channel, Adrenergic Receptor, AChR, Autophagy
Nicardipine-d3 hydrochloride
Cat.No: T12221
Synonym: 盐酸尼卡地平 D3,YC-93 D3
Target: Others
Cat. No. Product Name Target Signaling Pathways
T2142 Yohimbine hydrochloride

盐酸育亨宾,Antagonil,Yohimbine HCl

Adrenergic Receptor GPCR/G Protein; Neuroscience
Yohimbine hydrochloride (Antagonil) 是一种植物生物碱,具有 α-2-肾上腺素能阻断活性。它被用作散瞳药和治疗勃起功能障碍。
TCS2185 Yohimbine

Adrenergic Receptor GPCR/G Protein; Neuroscience
Yohimbine 是一种有效的、相对非选择性的α2 - 肾上腺素能受体拮抗剂,IC50=0.6μM。

天然产物

Yohimbine hydrochloride
Cat.No: T2142
Synonym: 盐酸育亨宾,Antagonil,Yohimbine HCl
Target: Adrenergic Receptor
Yohimbine
Cat.No: TCS2185
Synonym:
Target: Adrenergic Receptor
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