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Cat. No. Product Name Target Signaling Pathways
T2845 Imperatorin

Ammidin,8-Isoamylenoxypsoralen,欧前胡素,8-Isopentenyloxypsoralene,Marmelosin,Pentosalen

TRP/TRPV Channel; AChR; AChE; NOD Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience; NF-κB
Imperatorin (8-Isopentenyloxypsoralene) 是NO synthesis 和BChE 的抑制剂,IC50分别为 9.2 μmol 和 31.4 μmol。它也是TRPV1的微弱激动剂,EC50为 12.6±3.2 μM。
TN2325 (Z)-Akuammidine

钩吻素丁

Others Others
(Z)-Akuammidine is a natural product
TN3367 Akuammidine

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Akuammidine shows anti-inflammatory and anti-asthmatic properties, it has opioid analgesic activity, it shows a preference for mu-opioid binding sites with Ki values of 0.6, 2.4 and 8.6 microM at mu-, delta- and kappa-opioid binding sites, respectively.

天然产物

Imperatorin
Cat.No: T2845
Synonym: Ammidin,8-Isoamylenoxypsoralen,欧前胡素,8-Isopentenyloxypsoralene,Marmelosin,Pentosalen
Target: TRP/TRPV Channel, AChR, AChE, NOD
(Z)-Akuammidine
Cat.No: TN2325
Synonym: 钩吻素丁
Target: Others
Akuammidine
Cat.No: TN3367
Synonym:
Target: Opioid Receptor
TargetMol Loading
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