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Cat. No. Product Name Target Signaling Pathways
T2381 Abemaciclib

CDK4/6 dual inhibitor,LY2835219

CDK Cell Cycle/Checkpoint
Abemaciclib (LY2835219) 是一种 CDK4/6 的双重抑制剂 (IC50=2/10 nM),具有选择性和特异性。Abemaciclib 具有抗肿瘤活性,被用于治疗晚期或转移性乳腺癌。
T10220 Abemaciclib metabolite M2

Abemaciclib Metabolites M2

CDK Cell Cycle/Checkpoint
Abemaciclib Metabolites M2 is a metabolite of abemaciclib, acts as a potent CDK4 and CDK6 inhibitor (IC50s: 1-3 nM) with anti-cancer activity.
T3111 Abemaciclib methanesulfonate

abemaciclib mesylate,LY2835219,LY2835219 mesylate,LY2835219 (methanesulfonate)

CDK Cell Cycle/Checkpoint
Abemaciclib methanesulfonate (LY2835219) 是一种选择性的CDK4/6抑制剂,能够抑制 CDK4/CDK6 的活性,IC50分别为 2 nM 和 10 nM。
T10738 Abemaciclib metabolite M20

CDK4/6-IN-4,LSN3106726

CDK Cell Cycle/Checkpoint
Abemaciclib metabolite M20 (CDK4/6-IN-4) 是 Abemaciclib 的活性代谢物。 Abemaciclib metabolite M20 是一种特异性 CDK4/6 抑制剂,可用于癌症治疗的相关研究。
T73909 Abemaciclib metabolite M18

LSN3106729

Ligands for Target Protein for PROTAC PROTAC
Abemaciclibmetabolite M18 (LSN3106729) 是一种CDK抑制剂,具有抗肿瘤活性。作为Abemaciclib的代谢物,Abemaciclibmetabolite M18 能与CRBN配体结合,用于设计PROTAC CDK4/6降解剂。
T36967 LSN3106729 hydrochloride

LSN3106729 hydrochloride, the metabolite of Abemaciclib , is a CDK inhibitor with antitumor activity. LSN3106729 hydrochloride and a CRBN ligand have been used to design PROTAC CDK4/6 degrader[1]. [1]. Edward S. Kim, et al. Abemaciclib in Combination with Single-Agent Options in Patients with Stage IV Non-Small Cell Lung Cancer: A Phase Ib Study. [2]. Nathanael Gray, et al. Degradation of cyclin-dependent kinase 4/6 (cdk4/6) by conjugation of cdk4/6 inhibitors with e3 ligase ligand and methods o...

化合物

Abemaciclib
Cat.No: T2381
Synonym: CDK4/6 dual inhibitor,LY2835219
Target: CDK
Abemaciclib metabolite M2
Cat.No: T10220
Synonym: Abemaciclib Metabolites M2
Target: CDK
Abemaciclib methanesulfonate
Cat.No: T3111
Synonym: abemaciclib mesylate,LY2835219,LY2835219 mesylate,LY2835219 (methanesulfonate)
Target: CDK
Abemaciclib metabolite M20
Cat.No: T10738
Synonym: CDK4/6-IN-4,LSN3106726
Target: CDK
Abemaciclib metabolite M18
Cat.No: T73909
Synonym: LSN3106729
Target: Ligands for Target Protein for PROTAC
LSN3106729 hydrochloride
Cat.No: T36967
Synonym:
Target:
TargetMol Loading
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