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79

抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
TP1246L ACTH (22-39) acetate

ACTH (22-39) acetate (37548-29-1 Free base)

Others Others
ACTH (22-39) acetate 是促肾上腺皮质激素 (ACTH) 的片段,在 N 末端的第 3 位和第 15 位含有两个脯氨酸残基。
TP1245L ACTH 4-11 acetate

ACTH 4-11 acetate (67224-41-3 Free base)

Others Others
ACTH 4-11 acetate 是一种促肾上腺皮质激素片段,具有与 α-黑素细胞刺激素 (MSH) 相同的氨基酸序列。 ACTH 4-11 acetate 仅在高剂量时表现出微弱的 MSH 效力。
T7627L Adrenocorticotropic Hormone (ACTH) (4-10) TFA

Adrenocorticotropic Hormone (ACTH) (4-10) TFA(4037-01-8(free base)),Acth (4-10)

Melanocortin Receptor GPCR/G Protein; Neuroscience
Adrenocorticotropic Hormone (ACTH) (4-10) TFA (Acth (4-10)) 是一种有效的黑皮质素 (MC4R) 受体激动剂。
T8231 Adrenocorticotropic Hormone (ACTH) (1-39), human

ACTH (1-39), human,丝拉克肽

Others Others
Adrenocorticotropic Hormone (ACTH) (1-39), human (ACTH (1-39), human) 是黑皮质素受体激动剂。
TP1244L1 Adrenocorticotropic Hormone (ACTH) (1-10), human acetate

Adrenocorticotropic Hormone (ACTH) (1-10), human acetate(2791-05-1 Free base)

Others Others
Adrenocorticotropic Hormone (ACTH) (1-10), human acetate 是促肾上腺皮质激素的一个片段。 Adrenocorticotropic Hormone (ACTH) (1-10), human acetate 仅在 100 和 1000 nM 时具有较弱的 α-MSH 效力。
TP1011L ACTH (1-17) acetate

Melanocortin Receptor GPCR/G Protein; Neuroscience
ACTH (1-17) acetate 是一种有效的人黑皮质素 1 (MC1) 受体激动剂,具有高亲和力 (Ki = 0.21 nM)。
T20482L Acth (1-4) acetate(19405-50-6 free base)

Others Others
Acth (1-4) acetate(19405-50-6 free base) 是 ACTH N 端四肽。
TP1248L ACTH 11-24 acetate(4237-93-8 free base)

Adrenocorticotropic Hormone (11-24) acetate

Melanocortin Receptor GPCR/G Protein; Neuroscience
ACTH 11-24 acetate(4237-93-8 free base) (Adrenocorticotropic Hormone (11-24) acetate) 是促肾上腺皮质激素的片段,可诱导皮质醇释放。 ACTH (11-24) 已被确定为分离的肾上腺细胞中 ACTH (1-39) 和 ACTH (1-10) 的竞争性拮抗剂。
TP1238L ACTH 1-14 acetate(25696-21-3 free base)

Adrenocorticotropic Hormone Fragment 1-14 acetate

Adrenergic Receptor GPCR/G Protein; Neuroscience
ACTH 1-14 acetate(25696-21-3 free base) (Adrenocorticotropic Hormone Fragment 1-14 acetate) 是促肾上腺皮质激素的片段,可调节皮质醇和雄激素的产生。促肾上腺皮质激素 (ACTH),也称为促肾上腺皮质激素,由垂体前叶产生和分泌。作为对生物应激的反应,ACTH 是下丘脑-垂体-肾上腺轴的重要组成部分。
TP1240 Adrenocorticotropic Hormone (ACTH) (18-39), human TFA

CLIP (human) (TFA)

Others Others
Adrenocorticotropic Hormone (ACTH) (18-39), human TFA (CLIP human TFA) 是一种似皮质促素中叶肽,由垂体中叶的促黑素细胞产生。
TP2444 Acth (7-16)NH2

ACTH - (7-16)-amide

Acth (7-16)NH2 exhibits neurotrophic effects.
TP1245 ACTH (4-11)

ACTH 4-11,Adrenocorticotropic Hormone (4-11), human

ACTH (4-11) is a peptide fragment of adrenocorticotropic hormone, a peptide hormone found in the brain that is involved in the biological stress response.
TP1751 ACTH (34-39)

ACTH 34-39

ACTH (34-39) is an adrenocorticotropic hormone fragment.
TP1011 ACTH (1-17)

α1-17-ACTH

ACTH (1-17), an adrenocorticotropin analogue, is a potent human melanocortin 1 (MC1) receptor agonist with a Ki of 0.21 nM. Adrenocorticotropic hormone (ACTH), also known as corticotropin, is produced and secreted by the anterior pituitary gland.
TP1244 Adrenocorticotropic Hormone (ACTH) (1-10), human

ACTH (1-10), human

Adrenocorticotropic Hormone (ACTH) (1-10), human is a fragment of the adrenocorticotropin hormone. It exhibits a weak potency of α-melanocyte stimulating hormone (α-MSH), but only at high doses (100 and 1000 nM).
TP1246 ACTH (22-39)

ACTH 22-39,Adrenocorticotropic Hormone (22-39)

ACTH (22-39) is an adrenocorticotropic hormone (ACTH) fragment and it is the 22-39 sequence of ACTH.
TP1238 ACTH (1-14)

ACTH 1-14,Adrenocorticotropic Hormone Fragment 1-14

ACTH (1-14), a fragment of adrenocorticotropin, governs the production of cortisol and androgens.
T7627 Adrenocorticotropic Hormone (ACTH) (4-10), human

Adrenocorticotropic Hormone (ACTH) (4-10),ACTH (4-10), human,Acth (4-10)

Melanocortin Receptor GPCR/G Protein; Neuroscience
Adrenocorticotropic Hormone (ACTH) (4-10), human 是黑皮质素 4 型受体 (melanocortin 4 receptor, MC4R) 激动剂。
TP1010 ACTH (1-17) (TFA) (7266-47-9 free base)

α1-17-ACTH TFA,ACTH (1-17) (TFA)

ACTH (1-17) TFA is a corticotrophin analogue and an effective human melanocortin 1 (MC1) receptor agonist with Ki value of 0.21 nM.
TP1248 ACTH (11-24)

ACTH 11-24,Adrenocorticotropic Hormone (11-24)

ACTH (11-24) is a fragment of adrenocorticotrophin, induces cortisol release. ACTH (11-24) has been identified as a competitive antagonist of ACTH (1-39) and ACTH (1-10) in isolated adrenal cells.
TP1247 ACTH (1-13)

Adrenocorticotropic Hormone (1-13),ACTH 1-13

ACTH (1-13) is a 13-aa peptide, with cytoprotective effects in the model of ethanol induced gastric lesions in rats.Adrenocorticotropic hormone (ACTH), also known as corticotropin, is produced and secreted by the anterior pituitary gland. ACTH is an impor
T10251 Adrenocorticotropic Hormone (ACTH) (1-39), rat TFA

ACTH (1-39) (mouse, rat) TFA

Others Others
Adrenocorticotropic Hormone (ACTH) (1-39), rat (TFA) is a potent melanocortin 2 receptor (MC2) agonist.
TP1249 Adrenocorticotropic Hormone (ACTH) (1-39), rat

ACTH (1-39) (mouse, rat)

Adrenocorticotropic Hormone (ACTH) (1-39), rat is a potent melanocortin 2 (MC2) receptor agonist.Peptide fragments of ACTH (1-39) were formed during in vitro incubation of the peptide with membrane preparations. ACTH (1-39) were isolated by high pressure
TP1241 Adrenocorticotropic Hormone (ACTH) (18-39), human

ACTH (18-39), human

Adrenocorticotropic Hormone (ACTH) (18-39) is known as the Corticotropin-like Intermediate Lobe Peptide. It stimulates insulin secretion as well as amylase and protein secretion in a dose-dependent manner similar to those of secretin and carbamylcholine.
T20482 Acth (1-4)

(1-4) Corticotropin

Acth (1-4) is the ACTH N-terminal tetrapeptide.
TP1237 ACTH (1-14) TFA (25696-21-3 free base)

Adrenocorticotropic Hormone Fragment 1-14 (TFA),ACTH (1-14) TFA

ACTH (1-14) (TFA) is a polypeptide of corticotrophin, which promotes the release of cortisol.
TP1249L Adrenocorticotropic Hormone (ACTH) (1-39), rat acetate(77465-10-2 Free base)

T80125 ACTH (7-38) (human)

Melanocortin Receptor GPCR/G Protein; Neuroscience
ACTH (7-38) (human) 是 ACTH (1-39) 的第7至第38个氨基酸序列构成的片段。该化合物作为ACTH受体的拮抗剂,又称为促肾上腺皮质激素抑制肽(CIP),它不具有皮质类固醇活性。
TP1242 1-39-Corticotropin (human)(TFA)

Adrenocorticotropic Hormone (ACTH) (1-39), human(TFA)

Adrenocorticotropic Hormone (ACTH) (1-39) human(TFA),a member of the melanocortin family, is a melanocortin receptor agonist. It stimulates production of CS by the adrenals, but melanocortin receptors are also found in the central nervous system (CNS) and
T75979 ACTH (11-24) (acetate)

ACTH (11-24) (acetate) 为促肾上腺皮质激素(ACTH)受体拮抗剂,属于ACTH片段,具有诱导皮质醇释放的功能,适用于中枢神经系统研究。
T83178 ACTH (6-24) (human)

Adrenocorticotropic hormone (6-24)

ACTH (6-24) (human)(腎上腺皮質激素(6-24))是腎上腺皮質激素的片段。該化合物作為ACTH (1-39) 和 ACTH (5-24) 引起的類固醇生成的競爭性抑制劑,具有相應的Kd值分別為13.4和3.4nM。此外,ACTH (6-24) (human) 能夠抑制 hPTH 1-34 所誘導的皮質酮產生以及cAMP的累積。
T75985 ACTH (1-14) (TFA)

ACTH (1-14) (TFA) 是促肾上腺皮质激素的多肽片段,后者能够促进皮质醇的释放。
T80913 Tyr-ACTH (4-9)

Tyr-ACTH(4-9)为行为活性肽,常应用于研究大鼠学习行为的消除。
T75977 ACTH (1-17) (TFA)

ACTH (1-17) TFA 是促肾上腺皮质激素类似物,是一种有效的人黑皮素受体 (human melanocortin 1 (MC1) receptor) 激动剂,Ki 值为 0.21 nM。
T76643 Acetyl-ACTH (3-24) (human, bovine, rat)

Acetyl-ACTH (3-24) (human, bovine, rat) 是原黑色素皮质素 (POMC) 肽的片段。POMC 肽,如促肾上腺皮质激素(ACTH),是α-MSH 的前体,也是 MC-1 受体的激动剂。
T76303 (p-Iodo-Phe7)-ACTH (4-10)

'(p-Iodo-Phe7)-ACTH (4-10)'为垂体前腺产生和分泌的肾上腺皮质激素(ACTH)衍生物,担任黑素皮质素(MC)受体拮抗剂角色,能够抑制α-黑素细胞刺激激素(α-MSH)引发的大鼠过度梳理行为。
T76642 Acetyl-ACTH (2-24) (human, bovine, rat)

Acetyl-ACTH (2-24) (human, bovine, rat) 是原黑色素皮质素 (POMC) 肽的片段。POMC 肽,如促肾上腺皮质激素(ACTH),是α-MSH 的前体,也是MC-1受体的激动剂。
T76595 (Des-His6)-ACTH (1-24) (human, bovine, rat)

(Des-His6)-ACTH (1-24) (human, bovine, rat) 是促肾上腺皮质激素 (ACTH) 的类似物。ACTH 是一种由垂体前叶腺产生的多肽激素,调节皮质醇和雄激素的产生。
T76646 Acetyl-ACTH (7-24) (human, bovine, rat)

Acetyl-ACTH (7-24) (human, bovine, rat) 可导致 ACTH 诱发的皮质酮和醛固酮释放显著减少。
T76644 Acetyl-ACTH (4-24) (human, bovine, rat)

Acetyl-ACTH (4-24) (human, bovine, rat) 是原黑色素皮质素 (POMC) 肽的片段。POMC 肽,如促肾上腺皮质激素(ACTH),是α-MSH 的前体,也是 MC-1受体的激动剂。
T76591 (Des-Glu5)-ACTH (1-24) (human, bovine, rat)

(Des-Glu5)-ACTH (1-24) (human, bovine, rat) 是促肾上腺皮质激素 (ACTH) 的类似物。ACTH 是一种由垂体前叶腺产生的多肽激素,调节皮质醇和雄激素的产生。
T76500 ACTH (3-24) (human, bovine, mouse, ovine, porcine, rabbit, rat)

ACTH (3-24) (human, bovine, mouse, ovine, porcine, rabbit, rat) 是ACTH的3-24片段,适用于癌症、免疫疾病、心血管疾病等多种疾病的研究。
T22051 BU 224 hydrochloride

Imidazoline Receptor Neuroscience
BU 224 hydrochloride 是一种选择性的咪唑啉 I(2) 结合位点配体,具有镇痛和抗抑郁样活性。
T24980 5-DACTHF

543U76,5-Deazacyclotetrahydrofolate

5-DACTHF is an inhibitor of glycinamide ribonucleotide transformylase and aminoimidazole ribonucleotide transformylase used as an anti-purine drug.
TP1002L γ-1-MSH, amide acetate (72629-65-3 free base)

γ-1-MSH, amide acetate

Others Others
γ-1-MSH, amide acetate (72629-65-3 free base) 是 ACTH/β-内啡肽 (β-EP) 前体蛋白 N 末端区域的一种推定激素,RIA 使用抗 γ-3-MSH 抗血清对产生 ACTH 的小鼠进行了研究垂体肿瘤细胞,AtT-20/D16v。
TP2221L ANP (1-11), rat acetate

Atrial natriuretic factor (1-11) acetate,ANP (1-11), rat醋酸盐,Atriopeptide (1-11) acetate

Others Others
ANP (1-11), rat acetate (Atrial natriuretic factor (1-11) acetate) 是心房利钠因子之一,是 CRF 刺激的 ACTH 分泌的抑制剂。
T21268L Semax acetate(80714-61-0 free base)

Others Others
Semax acetate(80714-61-0 free base) 是一种合成的促肾上腺皮质激素 (ACTH) 肽类似物,具有神经保护、镇痛和抗焦虑特性。
T36926L Neuropeptide SF (human) aceate

Others Others
Neuropeptide SF (human) aceate 是一种神经肽,可增强心室旁 CRH 的释放并增加血浆中的 ACTH 和皮质酮水平。
TP2082L d[Cha4]-AVP acetate(500170-27-4 free base)

Vasopressin Receptor GPCR/G Protein
d[Cha4]-AVP acetate(500170-27-4 free base) 是一种有效的选择性人血管加压素 V1B 受体激动剂(V1B、V1A、催产素和 V2 受体的 Ki 值分别为 1.2、151、240 和 750 nM)。刺激 ACTH 和皮质酮分泌,并在体内表现出微不足道的血管加压活性。
TP1031 Tetracosactide

Tetracosactrin,替可克肽

Others Others
Tetracosactide (Tetracosactrin) 是一种肾上腺皮质激素 (ACTH) 的类似物,能够刺激肾上腺皮质激素分泌。

化合物

ACTH (22-39) acetate
Cat.No: TP1246L
Synonym: ACTH (22-39) acetate (37548-29-1 Free base)
Target: Others
ACTH 4-11 acetate
Cat.No: TP1245L
Synonym: ACTH 4-11 acetate (67224-41-3 Free base)
Target: Others
Adrenocorticotropic Hormone (ACTH) (4-10) TFA
Cat.No: T7627L
Synonym: Adrenocorticotropic Hormone (ACTH) (4-10) TFA(4037-01-8(free base)),Acth (4-10)
Target: Melanocortin Receptor
Adrenocorticotropic Hormone (ACTH) (1-39), human
Cat.No: T8231
Synonym: ACTH (1-39), human,丝拉克肽
Target: Others
Adrenocorticotropic Hormone (ACTH) (1-10), human acetate
Cat.No: TP1244L1
Synonym: Adrenocorticotropic Hormone (ACTH) (1-10), human acetate(2791-05-1 Free base)
Target: Others
ACTH (1-17) acetate
Cat.No: TP1011L
Synonym:
Target: Melanocortin Receptor
Acth (1-4) acetate(19405-50-6 free base)
Cat.No: T20482L
Synonym:
Target: Others
ACTH 11-24 acetate(4237-93-8 free base)
Cat.No: TP1248L
Synonym: Adrenocorticotropic Hormone (11-24) acetate
Target: Melanocortin Receptor
ACTH 1-14 acetate(25696-21-3 free base)
Cat.No: TP1238L
Synonym: Adrenocorticotropic Hormone Fragment 1-14 acetate
Target: Adrenergic Receptor
Adrenocorticotropic Hormone (ACTH) (18-39), human TFA
Cat.No: TP1240
Synonym: CLIP (human) (TFA)
Target: Others
Acth (7-16)NH2
Cat.No: TP2444
Synonym: ACTH - (7-16)-amide
Target:
ACTH (4-11)
Cat.No: TP1245
Synonym: ACTH 4-11,Adrenocorticotropic Hormone (4-11), human
Target:
ACTH (34-39)
Cat.No: TP1751
Synonym: ACTH 34-39
Target:
ACTH (1-17)
Cat.No: TP1011
Synonym: α1-17-ACTH
Target:
Adrenocorticotropic Hormone (ACTH) (1-10), human
Cat.No: TP1244
Synonym: ACTH (1-10), human
Target:
ACTH (22-39)
Cat.No: TP1246
Synonym: ACTH 22-39,Adrenocorticotropic Hormone (22-39)
Target:
ACTH (1-14)
Cat.No: TP1238
Synonym: ACTH 1-14,Adrenocorticotropic Hormone Fragment 1-14
Target:
Adrenocorticotropic Hormone (ACTH) (4-10), human
Cat.No: T7627
Synonym: Adrenocorticotropic Hormone (ACTH) (4-10),ACTH (4-10), human,Acth (4-10)
Target: Melanocortin Receptor
ACTH (1-17) (TFA) (7266-47-9 free base)
Cat.No: TP1010
Synonym: α1-17-ACTH TFA,ACTH (1-17) (TFA)
Target:
ACTH (11-24)
Cat.No: TP1248
Synonym: ACTH 11-24,Adrenocorticotropic Hormone (11-24)
Target:
ACTH (1-13)
Cat.No: TP1247
Synonym: Adrenocorticotropic Hormone (1-13),ACTH 1-13
Target:
Adrenocorticotropic Hormone (ACTH) (1-39), rat TFA
Cat.No: T10251
Synonym: ACTH (1-39) (mouse, rat) TFA
Target: Others
Adrenocorticotropic Hormone (ACTH) (1-39), rat
Cat.No: TP1249
Synonym: ACTH (1-39) (mouse, rat)
Target:
Adrenocorticotropic Hormone (ACTH) (18-39), human
Cat.No: TP1241
Synonym: ACTH (18-39), human
Target:
Acth (1-4)
Cat.No: T20482
Synonym: (1-4) Corticotropin
Target:
ACTH (1-14) TFA (25696-21-3 free base)
Cat.No: TP1237
Synonym: Adrenocorticotropic Hormone Fragment 1-14 (TFA),ACTH (1-14) TFA
Target:
Adrenocorticotropic Hormone (ACTH) (1-39), rat acetate(77465-10-2 Free base)
Cat.No: TP1249L
Synonym:
Target:
ACTH (7-38) (human)
Cat.No: T80125
Synonym:
Target: Melanocortin Receptor
1-39-Corticotropin (human)(TFA)
Cat.No: TP1242
Synonym: Adrenocorticotropic Hormone (ACTH) (1-39), human(TFA)
Target:
ACTH (11-24) (acetate)
Cat.No: T75979
Synonym:
Target:
ACTH (6-24) (human)
Cat.No: T83178
Synonym: Adrenocorticotropic hormone (6-24)
Target:
ACTH (1-14) (TFA)
Cat.No: T75985
Synonym:
Target:
Tyr-ACTH (4-9)
Cat.No: T80913
Synonym:
Target:
ACTH (1-17) (TFA)
Cat.No: T75977
Synonym:
Target:
Acetyl-ACTH (3-24) (human, bovine, rat)
Cat.No: T76643
Synonym:
Target:
(p-Iodo-Phe7)-ACTH (4-10)
Cat.No: T76303
Synonym:
Target:
Acetyl-ACTH (2-24) (human, bovine, rat)
Cat.No: T76642
Synonym:
Target:
(Des-His6)-ACTH (1-24) (human, bovine, rat)
Cat.No: T76595
Synonym:
Target:
Acetyl-ACTH (7-24) (human, bovine, rat)
Cat.No: T76646
Synonym:
Target:
Acetyl-ACTH (4-24) (human, bovine, rat)
Cat.No: T76644
Synonym:
Target:
(Des-Glu5)-ACTH (1-24) (human, bovine, rat)
Cat.No: T76591
Synonym:
Target:
ACTH (3-24) (human, bovine, mouse, ovine, porcine, rabbit, rat)
Cat.No: T76500
Synonym:
Target:
BU 224 hydrochloride
Cat.No: T22051
Synonym:
Target: Imidazoline Receptor
5-DACTHF
Cat.No: T24980
Synonym: 543U76,5-Deazacyclotetrahydrofolate
Target:
γ-1-MSH, amide acetate (72629-65-3 free base)
Cat.No: TP1002L
Synonym: γ-1-MSH, amide acetate
Target: Others
ANP (1-11), rat acetate
Cat.No: TP2221L
Synonym: Atrial natriuretic factor (1-11) acetate,ANP (1-11), rat醋酸盐,Atriopeptide (1-11) acetate
Target: Others
Semax acetate(80714-61-0 free base)
Cat.No: T21268L
Synonym:
Target: Others
Neuropeptide SF (human) aceate
Cat.No: T36926L
Synonym:
Target: Others
d[Cha4]-AVP acetate(500170-27-4 free base)
Cat.No: TP2082L
Synonym:
Target: Vasopressin Receptor
Tetracosactide
Cat.No: TP1031
Synonym: Tetracosactrin,替可克肽
Target: Others
Cat. No. Product Name Target Signaling Pathways
T8209 Saikosaponin b3

柴胡皂苷b3

Others Others
Saikosaponin b3 是从 Bupleurum falcatum L. 的根中分离得到的。Saikosaponin b3 抑制 ACTH 诱导的脂肪细胞中的脂肪分解并具有镇痛作用。
T8210 Saikosaponin B4

Others Others
Saikosaponin B4 是一种柴胡皂苷,分离自柴胡的根。Saikosaponin B4选择性地抑制 ACTH 诱导的脂解作用。

天然产物

Saikosaponin b3
Cat.No: T8209
Synonym: 柴胡皂苷b3
Target: Others
Saikosaponin B4
Cat.No: T8210
Synonym:
Target: Others
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