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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T10137 4-Bromo A23187

4-​Bromo A23187

Others Others
4-Bromo A23187 is a halogenated analog of the calcium ionophore A-23187. 4-Bromo A23187 is a calcium modulator and induces apoptosis in different cells.
T75656 Calcimycin hemimagnesium

Calcimycin (A-23187) hemimagnesium,一种具有抗生素功能的独特二价阳离子离子载体(例如钙离子和镁离子),通过提高细胞内钙浓度而诱导Ca2+依赖性细胞死亡。该化合物还能抑制革兰氏阳性细菌和部分真菌生长,同时抑制ATP酶活性并解耦哺乳动物细胞的氧化磷酸化(OXPHOS),触发细胞凋亡(apoptosis)。

化合物

4-Bromo A23187
Cat.No: T10137
Synonym: 4-​Bromo A23187
Target: Others
Calcimycin hemimagnesium
Cat.No: T75656
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T10662L Calcimycin

Antibiotic A-23187,离子载体(钙镁盐混合物),A-23187

Apoptosis; Antibacterial; Antibiotic; Autophagy; Antifungal Apoptosis; Autophagy; Microbiology/Virology
Calcimycin (A-23187) 是抗生素和二价阳离子离子载体。它抑制革兰氏阳性细菌和一些真菌生长,也抑制 ATP 酶的活性并解耦哺乳动物细胞的氧化磷酸化。它通过增加细胞内钙浓度诱导 Ca2+依赖性细胞死亡。
T10662 Calcimycin hemicalcium salt

Antibiotic A-23187 hemicalcium salt,A-23187 hemicalcium salt

Others Others
Calcimycin (A-23187) hemicalcium salt is an antibiotic and a unique divalent cation ionophore (like calcium and magnesium). It induces Ca2+-dependent cell death by increasing intracellular calcium concentration.
T4114 Diffractaic Acid

NSC 5901,地弗地衣酸,NSC 685595

Apoptosis; LTR Apoptosis; Immunology/Inflammation
Diffractaic Acid (NSC 685595) 是松萝的主要成分,具有止痛和解热效果,在各种疾病研究中可作为有效的促凋亡剂。
TN4584 Morolic acid

IL Receptor; COX; HIV Protease Immunology/Inflammation; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Morolic acid and moronic acid have shown sustained antidiabetic and antihyperglycemic action possibly mediated by an insulin sensitization with consequent changes of glucose, cholesterol and triglycerides, in part mediated by inhibition of 11β-HSD 1. Moro

天然产物

Calcimycin
Cat.No: T10662L
Synonym: Antibiotic A-23187,离子载体(钙镁盐混合物),A-23187
Target: Apoptosis, Antibacterial, Antibiotic, Autophagy, Antifungal
Calcimycin hemicalcium salt
Cat.No: T10662
Synonym: Antibiotic A-23187 hemicalcium salt,A-23187 hemicalcium salt
Target: Others
Diffractaic Acid
Cat.No: T4114
Synonym: NSC 5901,地弗地衣酸,NSC 685595
Target: Apoptosis, LTR
Morolic acid
Cat.No: TN4584
Synonym:
Target: IL Receptor, COX, HIV Protease
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