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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10036 |
10β,17β-dihydroxyestra-1,4-dien-3-one
DHED |
Others | Others |
10β,17β-dihydroxyestra-1,4-dien-3-one is a brain-targeting bioprecursor prodrug of the main human estrogen, 17β-estradiol. It alleviates hot flushes in rat models of thermoregulatory dysfunction of the brain. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2S2335 |
Dehydroevodiamine
DHED,去氢吴茱萸碱 |
Others; NF-κB; COX; PGE Synthase; NO Synthase | Immunology/Inflammation; Neuroscience; NF-κB; Others |
Dehydroevodiamine (DHED) 是从吴茱萸中分离出的一种喹唑啉生物碱,可抑制 LPS 诱导的小鼠巨噬细胞中iNOS、COX-2、PGE2和NF-κB 的表达,对豚鼠心室肌细胞具有抗心律失常作用。 | |||
T5721 |
Dehydroevodiamine hydrochloride
|
AChE | Neuroscience |
Dehydroevodiamine hydrochloride 是分离自吴茱萸叶中,能够抑制 AChE。 它能够调节一氧化氮的产生,具有降压和神经保护作用。 |