Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN1266 |
3-O-Methylquercetin
|
IL Receptor; cAMP; PDE | GPCR/G Protein; Immunology/Inflammation; Metabolism |
3-O-Methylquercetin 是分离自植物Rhamnus nakaharai 的天然产物,可抑制总 cAMP 和cGMP-phosphodiesterase (PDE)。它对PDE1、PDE5、PDE 和PDE4的IC50分别是31.9 μM、86.9 μM、18.6 μM 和1.6 μM。 | |||
T2836 |
Isorhamnetin
3-methylquercetin,3'-Methylquercetin,Isorhamnetol,异鼠李素,3'-Methoxyquercetin |
MEK; PI3K; Endogenous Metabolite | MAPK; Metabolism; PI3K/Akt/mTOR signaling |
Isorhamnetin (3-methylquercetin) 是从中草药沙棘中提取的一种类黄酮,可通过抑制MEK1和PI3K 来抑制皮肤癌。 | |||
TN2974 |
3-O-Methylquercetin tetraacetate
|
IL Receptor; TNF; PDE | Apoptosis; Immunology/Inflammation; Metabolism |
Quercetin 3-O-methyl ether is a potent phosphodiesterase (PDE)3/4 inhibitor, it has potential for treating asthma against ovalbumin-induced airway hyperresponsiveness. | |||
T81691 |
Neochilenin
3-O-Methylquercetin 4′-O-glucoside |
||
Neochilenin (3-O-Methylquercetin 4'-O-glucoside) 是一种从蜡菊亚科 (Cactaceae) 分离出的3-O-methylquercetin糖苷。 | |||
T83347 |
3-O-Methylquercetin 4',7-di-β-D-glucopyranoside
|
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3-O-Methylquercetin 4',7-di-β-D-glucopyranoside为一种从尖头瓶尔小草中提取的类黄酮糖苷。 |