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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T38718 Cytarabine triphosphate

Cytarabine triphosphate,Ara-CTP

Cytarabine triphosphate (Ara-CTP), a competitive inhibitor of DNA synthesis and an active metabolite of Cytarabine, exhibits predictive potential for leukemic blasts' chemosensitivity to Cytarabine through intracellular levels.
T1272L Cytarabine hydrochloride

Ara-C hydrochloride,Cytosine Arabinoside hydrochloride

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Cytarabine hydrochloride (Ara-C hydrochloride) 是一种核苷类似物,可导致 S 期细胞周期停滞并抑制DNA 聚合酶。Cytarabine 抑制DNA 合成,IC50为 16 nM。Cytarabine hydrochloride 对HSV 具有抗病毒作用。

化合物

Cytarabine triphosphate
Cat.No: T38718
Synonym: Cytarabine triphosphate,Ara-CTP
Target:
Cytarabine hydrochloride
Cat.No: T1272L
Synonym: Ara-C hydrochloride,Cytosine Arabinoside hydrochloride
Target: DNA/RNA Synthesis
Cat. No. Product Name Target Signaling Pathways
T1272 Cytarabine

阿糖胞苷,Ara-C,Cytosine Arabinoside,Cytosine β-D-arabinofuranoside,Arabinocytidine

Apoptosis; Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis; Endogenous Metabolite; Autophagy; HSV Apoptosis; Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Cytarabine (Ara-C) 是一种核苷类似物,一种 DNA 合成抑制剂 (IC50=16 nM)。Cytarabine 可以抑制 DNA 聚合酶,诱导细胞周期阻滞、细胞自噬和凋亡。Cytarabine 具有抗肿瘤活性。

天然产物

Cytarabine
Cat.No: T1272
Synonym: 阿糖胞苷,Ara-C,Cytosine Arabinoside,Cytosine β-D-arabinofuranoside,Arabinocytidine
Target: Apoptosis, Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis, Endogenous Metabolite, Autophagy, HSV
TargetMol Loading
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