Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2350 |
MALT1 inhibitor MI-2
MALT1 inhibitor,MI 2,MI 2 (MALT1 inhibitor) |
MALT | Immunology/Inflammation |
MI 2 (MALT1 inhibitor) 是一种MALT1抑制剂 (IC50=5.84 μM),对动物无毒性。它能够直接与 MALT1 结合,不可逆地抑制蛋白酶功能,并伴有 NF-κB 报告子活性抑制、c-REL 核定位抑制和 NF-κB 靶基因下调。 | |||
T2649 |
Menin-MLL inhibitor MI-2
Menin-MLL Inhibitor,MI2,MI-2,Menin-MLL inhibitor 2,MI 2 |
Apoptosis; Epigenetic Reader Domain; Histone Methyltransferase | Apoptosis; Chromatin/Epigenetic |
Menin-MLL inhibitor MI-2 (MI2) 抑制Menin-MLL 相互作用,IC50为 446±28 nM。 | |||
T22978 | MI-2 (hydrochloride) | Others | Others |
MI-2 (Menin-MLL Inhibitor) is an effective menin-MLL interaction inhibitor (IC50: 446 ± 28 nM). |