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6

抑制剂 & 化合物

8

天然产物

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Cat. No. Product Name Target Signaling Pathways
T6582 Mezlocillin Sodium

美洛西林钠,Baycipen

Antibacterial; Antibiotic Microbiology/Virology
Mezlocillin Sodium (Baycipen) 是一种青霉素 β-内酰胺类抗生素,用于治疗由易感染微生物引起的细菌感染。
T7560 Pivmecillinam hydrochloride

美西林盐酸盐,FL-1039 hydrochloride,盐酸匹美西林

Antibacterial; Antibiotic Microbiology/Virology
Pivmecillinam hydrochloride (FL-1039 hydrochloride) 是Mecillinam 的口服活性前药,是一种广谱青霉素抗生素,对革兰氏阴性菌有活性,可用作氨苄青霉素。
T21369 Mecillinam

Amdinocillin,Mecillinamum,Hexacillin,美西林,Coactin,Penicillin HX

Antibacterial Microbiology/Virology
Mecillinam (Hexacillin) 是一种有抗革兰氏阴性菌活性的 β 内酰胺类广谱抗生素。
T29960 Pivmecillinam

美西林,Amdinocillin pivoxil

Amdinocillin pivoxil is a Pivaloyloxymethyl ester of amdinocillin that is well absorbed orally, but broken down to amdinocillin in the intestinal mucosa. It is active against gram-negative organisms and used as for amdinocillin.
T20131 Cevimeline hydrochloride

盐酸西维美林,Cevimeline HCl,Evoxac

Cevimeline HCl is an agonist of cholinergic that binds to muscarinic receptors. Muscarinic agonists in sufficient dosage can enhance the secretion of exocrine glands, such as salivary and sweat glands.
T21119 Cevimeline

AF-102B,西维美林,FKS 508,SNI 2011,HSDB 7286

Cevimeline, a parasympathomimetic and muscarinic agonist, affects M1 and M3 receptors. Cevimeline has been shown to treat dry mouth and Sj gren's syndrome. It is also used to reduce Xerostomia symptoms and increase salivary flow in head and neck cancer survivors after radiotherapy.

化合物

Mezlocillin Sodium
Cat.No: T6582
Synonym: 美洛西林钠,Baycipen
Target: Antibacterial, Antibiotic
Pivmecillinam hydrochloride
Cat.No: T7560
Synonym: 美西林盐酸盐,FL-1039 hydrochloride,盐酸匹美西林
Target: Antibacterial, Antibiotic
Mecillinam
Cat.No: T21369
Synonym: Amdinocillin,Mecillinamum,Hexacillin,美西林,Coactin,Penicillin HX
Target: Antibacterial
Pivmecillinam
Cat.No: T29960
Synonym: 美西林,Amdinocillin pivoxil
Target:
Cevimeline hydrochloride
Cat.No: T20131
Synonym: 盐酸西维美林,Cevimeline HCl,Evoxac
Target:
Cevimeline
Cat.No: T21119
Synonym: AF-102B,西维美林,FKS 508,SNI 2011,HSDB 7286
Target:
Cat. No. Product Name Target Signaling Pathways
T8212 Dichotomitin

Others Others
Dichotomitin 是一种提取自Belamcanda chinensis 根茎中的异黄酮。
T6S1665 Irisflorentin

Others; NO Synthase Immunology/Inflammation; Others
Irisflorentin 是天然存在的异黄酮,是大量存在于 Rhizoma Belamcandae 中的活性成分。它明显抑制了诱导型一氧化氮合酶的转录和翻译以及 NO 产生。
TN2359 Iristectorigenin B

Iristectrigenin B

Liver X Receptor Metabolism
Iristectorigenin B (Iristectrigenin B) 是一种有效的肝脏 X 受体 (LXR) 调节剂,是从 Belamcanda chinensis 中分离的小分子化合物。Iristectrigenin B 可促进巨噬细胞 RAW 1.1 细胞中 ABCA264 和 ABCG7 的表达。
T3862 Irigenin

NF-κB; Integrin Cytoskeletal Signaling; NF-κB
Irigenin 可通过特异性和选择性地阻断 Extra Domain A 域的 C-C 环上α9β1和α4β1整合素结合位点,介导其抗转移作用。可通过增强胃癌细胞中促凋亡分子的表达来敏化 TRAIL 诱导的凋亡,具有抗癌作用。
TN2357 Iristectorigenin A

鸢尾黄酮甲素,鸢尾甲黄素A

Others Others
Iristectorigenin A 是从一种天然异黄酮,分离自B. chinensis 根茎中,具有抗氧化作用。
T3820 Iridin

野鸢尾苷,Lridin

Others Others
Iridin (Lridin) 是抑制异黄酮化合物,从Iris milesii 中提取得到。
TN3738 Cycloartanol

Others Others
Cycloartanol is a natural product from Citrus medica.
TN6524 Irilone

Irilone has immunomodulatory, and α-amylase inhibitory activities, it exhibits the selective inhibition toward CYP3 A4 rather than other major human CYPs. Irilone exhibited prominent antioxidant activities with the IC50 value of 10.46μM. Irilone potentiat

天然产物

Dichotomitin
Cat.No: T8212
Synonym:
Target: Others
Irisflorentin
Cat.No: T6S1665
Synonym:
Target: Others, NO Synthase
Iristectorigenin B
Cat.No: TN2359
Synonym: Iristectrigenin B
Target: Liver X Receptor
Irigenin
Cat.No: T3862
Synonym:
Target: NF-κB, Integrin
Iristectorigenin A
Cat.No: TN2357
Synonym: 鸢尾黄酮甲素,鸢尾甲黄素A
Target: Others
Iridin
Cat.No: T3820
Synonym: 野鸢尾苷,Lridin
Target: Others
Cycloartanol
Cat.No: TN3738
Synonym:
Target: Others
Irilone
Cat.No: TN6524
Synonym:
Target:
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