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Cat. No. Product Name Target Signaling Pathways
T5420 Cycloguanil hydrochloride

Chloroguanide Triazine,环氯胍盐酸盐

Parasite; Drug Metabolite Metabolism; Microbiology/Virology
Cycloguanil hydrochloride (Chloroguanide Triazine) 是抗疟化合物氯胍的活性代谢物。 它作为二氢叶酸还原酶的抑制剂,对于疟原虫和人类形式的 Kis 值分别为 0.3 和 1.5 nM。
T4382 Proguanil hydrochloride

Paludrine hydrochloride,盐酸氯胍,Chlorguanide hydrochloride,Chloroquanil

Others; Dehydrogenase; DNA/RNA Synthesis; Antifolate; Parasite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; Others
Proguanil hydrochloride (Chloroquanil) 是一种双胍类抗疟疾剂,在体内代谢形成环胍。它还是一种二氢叶酸还原酶抑制剂。
T2549 Robenidine hydrochloride

Rasexinium,Dexium,氯苯胍盐酸盐,Robenidine Hydrochoride,Toraxine,盐酸氯苯胍,Nugatex

Antibacterial; Antibiotic; Parasite Microbiology/Virology
Robenidine hydrochloride (Robenidine Hydrochoride) 是一种主要用于家禽的抗球虫剂, 对 MRSA 和 VRE 有抑制活性,其 MIC50值分别为 8.1 和 4.7 μM。
T0358 Aminoguanidine hydrochloride

Imino semicarbazide,Pimagedine hydrochloride,CP-12009-18 tartrate,Hydrazinecarboximidamide,肼甲酰亚胺酰胺一氯化氢(氨基胍盐酸盐),氨基胍盐酸盐,Guanyl hydrazine,Pimagedine

NOS; NO Synthase Immunology/Inflammation
Aminoguanidine hydrochloride (Hydrazinecarboximidamide) 是二胺氧化酶抑制剂,也是一氧化氮合酶抑制剂,可用于糖尿病肾病的研究。

化合物

Cycloguanil hydrochloride
Cat.No: T5420
Synonym: Chloroguanide Triazine,环氯胍盐酸盐
Target: Parasite, Drug Metabolite
Proguanil hydrochloride
Cat.No: T4382
Synonym: Paludrine hydrochloride,盐酸氯胍,Chlorguanide hydrochloride,Chloroquanil
Target: Others, Dehydrogenase, DNA/RNA Synthesis, Antifolate, Parasite
Robenidine hydrochloride
Cat.No: T2549
Synonym: Rasexinium,Dexium,氯苯胍盐酸盐,Robenidine Hydrochoride,Toraxine,盐酸氯苯胍,Nugatex
Target: Antibacterial, Antibiotic, Parasite
Aminoguanidine hydrochloride
Cat.No: T0358
Synonym: Imino semicarbazide,Pimagedine hydrochloride,CP-12009-18 tartrate,Hydrazinecarboximidamide,肼甲酰亚胺酰胺一氯化氢(氨基胍盐酸盐),氨基胍盐酸盐,Guanyl hydrazine,Pimagedine
Target: NOS, NO Synthase
TargetMol Loading
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