Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5420 |
Cycloguanil hydrochloride
Chloroguanide Triazine,环氯胍盐酸盐 |
Parasite; Drug Metabolite | Metabolism; Microbiology/Virology |
Cycloguanil hydrochloride (Chloroguanide Triazine) 是抗疟化合物氯胍的活性代谢物。 它作为二氢叶酸还原酶的抑制剂,对于疟原虫和人类形式的 Kis 值分别为 0.3 和 1.5 nM。 | |||
T4382 |
Proguanil hydrochloride
Paludrine hydrochloride,盐酸氯胍,Chlorguanide hydrochloride,Chloroquanil |
Others; Dehydrogenase; DNA/RNA Synthesis; Antifolate; Parasite | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; Others |
Proguanil hydrochloride (Chloroquanil) 是一种双胍类抗疟疾剂,在体内代谢形成环胍。它还是一种二氢叶酸还原酶抑制剂。 | |||
T2549 |
Robenidine hydrochloride
Rasexinium,Dexium,氯苯胍盐酸盐,Robenidine Hydrochoride,Toraxine,盐酸氯苯胍,Nugatex |
Antibacterial; Antibiotic; Parasite | Microbiology/Virology |
Robenidine hydrochloride (Robenidine Hydrochoride) 是一种主要用于家禽的抗球虫剂, 对 MRSA 和 VRE 有抑制活性,其 MIC50值分别为 8.1 和 4.7 μM。 | |||
T0358 |
Aminoguanidine hydrochloride
Imino semicarbazide,Pimagedine hydrochloride,CP-12009-18 tartrate,Hydrazinecarboximidamide,肼甲酰亚胺酰胺一氯化氢(氨基胍盐酸盐),氨基胍盐酸盐,Guanyl hydrazine,Pimagedine |
NOS; NO Synthase | Immunology/Inflammation |
Aminoguanidine hydrochloride (Hydrazinecarboximidamide) 是二胺氧化酶抑制剂,也是一氧化氮合酶抑制剂,可用于糖尿病肾病的研究。 |