AChR

An acetylcholine receptor (abbreviated AChR) is an integral membrane protein that responds to the binding of acetylcholine, a neurotransmitter.

Cat. No.	Product Name	CAS No.	Purity
TN2131	Questin 化合物Questin	3774-64-9	98%
TN2131	Questin 是一种从花样黄曲霉中提取出来的抗菌剂，具有抗菌活型，对V. harveyi，V. anguillarum，V. cholerae 和 V. parahemolyticus 具有抑制作用，MIC 值分别为 31.25 µg/mL，62.5 µg/mL，62.5 µg/mL 和 125 µg/mL。Quest...
T17312	(+)-Phenserine 化合物 T17312	116839-68-0	98%
T17312	(+)-Phenserine is a novel selective inhibitor of cholinesterase non-competitive (IC50: 45.3 μM).
T16353	Meseclazone 美西拉宗	29053-27-8	98%
T16353	Meseclazone has anti-inflammatory, analgesic, and antipyretic activity. Meseclazone shows inhibitory potency of secondary phase ADP aggregation.
TN4426	Leojaponin 化合物 TN4426	864817-63-0	98%
TN4426	Leojaponin is a prolyl oligopeptidase (POP) inhibitor. Leojaponin exhibits significant cytoprotective activities against glutamate-induced toxicity at concentrat...
TN3285	8-Hydroxypinoresinol 化合物 TN3285	81426-17-7	98%
TN3285	8-Hydroxypinoresinol has antioxidant activity,it and phillygenin significantly reduce the cell injury by 3-morpholinosydnonimine (SIN-1), a ONOO- generator, may ...
TN4492	Mangostanol 化合物 TN4492	184587-72-2	98%
TN4492	Mangostanol is an acetylcholinesterase (AChE) selective inhibitor.Mangostanol has anti-cancer activity, it shows significant activities against the CEM-SS cell l...
TL0018	Lobelin 化合物 TL0018	90-69-7	98%
TL0018	Inhalation challenge with capsaicin and rapid intravenous injection of Lobelin and alinamin indicated that peripheral c-fiber receptors were involved in the indu...
TN5193	Tubotaiwine 化合物 TN5193	6711-69-9	98%
TN5193	Tubotaiwine shows selective activity against L. infantum. Tubotaiwine and apparicine have affinity for adenosine receptors in the micromolar range and also have ...
T14966	Cimetropium Bromide 西托溴铵	51598-60-8	98%
T14966	Cimetropium Bromide is a mAChR antagonist used for long-term treatment of irritable bowel syndrome.
T12825	Timepidium bromide 化合物 T12825	35035-05-3	98%
T12825	Timepidium bromide is an agent of anticholinergic.
TN3287	8-Lavandulylkaempferol 化合物 TN3287	883859-83-4	98%
TN3287	8-Lavandulylkaempferol exhibits significant inhibitory effects with IC(50) values of 7.10 and 8.11 microM for butyrylcholinesterase and acetylcholinesterase, res...
T12766	RPR121056 化合物 T12766	181467-56-1	98%
T12766	RPR121056 is a Irinotecan metabolite, which is generated by CYP3A4. Irinotecan is an antineoplastic agent that inhibits topoisomerase type I.
TN3550	Buxbodine B 化合物 TN3550	390362-51-3	98%
TN3550	Buxbodine B has weak anti-AChE activity with IC50 values in the range of 10.8-98μM.
T12136	N-0861 racemate 化合物 T12136	121241-87-0	98%
T12136	N-0861 racemate is the racemate of N-0861.
TN3812	Dehydrovomifoliol 化合物 TN3812	39763-33-2	98%
TN3812	Dehydrovomifoliol could be a marker of Polish heather honey. Dehydrovomifoliol exhibits moderate acetylcholinesterase (AChE) inhibitory activities. Dehydrovomifo...
TN4286	Isodunnianol 化合物 TN4286	139726-30-0	98%
TN4286	Isodunnianol exhibits anti-AChE activity with an IC50 value of 13.0 uM; it also exhibits neurite outgrowth-promoting activity at the concentration ranging from 0...
T8306	Epiberberine chloride 表小檗碱氯化物	889665-86-5	98%
T8306	Epiberberine chloride (Epiberberine (chloride)) 是一种从黄连中得到的生物碱，是一种AChE 和BChE 抑制剂，和非竞争性的BACE1抑制剂。它具有抗氧化作用，能够清除 ONOO-，可用于研究阿尔滋海默症和糖尿病。
T19933	GTS-21 化合物GTS-21	148372-04-7	98%
T19933	GTS-21 (DMXB-A) 是一种 α7 nAChR 激动剂。 GTS-21 通过抑制 RA Th1 细胞分化来抑制与类风湿性关节炎相关的炎症。
TN4600	Myrianthic acid 化合物 TN4600	89786-84-5	98%
TN4600	Myrianthic acid shows anticancer activity, it shows inhibitory activities on foam cell formation in human monocyte-derived macrophages induced by acetylated low-...
TN3744	Cyclomorusin 化合物 TN3744	62596-34-3	98%
TN3744	Cyclomorusin exhibits competitive inhibition toward monophenolase activity of mushroom tyrosinase, the IC50 value of 0.092 microM. It evokes the stimulation of s...