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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T0977 Medrysone

Gimeracil,6α-Methyl-11β-hydroxyprogesterone,6A-甲基-11B-羟孕酮,甲羟松

Glucocorticoid Receptor; Others Endocrinology/Hormones; Others
Medrysone (6α-Methyl-11β-hydroxyprogesterone) 是局部合成的糖皮质激素,具有代谢、抗炎和抗过敏特性,有潜力用于眼科的眼炎症研究。
T3357 Clascoterone

Cortexolone 17 alpha-propionate,17 alpha-propionate,21-羟基-17-(1-氧代丙氧基)孕甾-4-烯-3,20-二酮,CB-03-01,Cortexolone 17α-propionate

Androgen Receptor Endocrinology/Hormones
Clascoterone (CB-03-01) 是一种新型的局部和外周的雄性激素拮抗剂。

化合物

Medrysone
Cat.No: T0977
Synonym: Gimeracil,6α-Methyl-11β-hydroxyprogesterone,6A-甲基-11B-羟孕酮,甲羟松
Target: Glucocorticoid Receptor, Others
Clascoterone
Cat.No: T3357
Synonym: Cortexolone 17 alpha-propionate,17 alpha-propionate,21-羟基-17-(1-氧代丙氧基)孕甾-4-烯-3,20-二酮,CB-03-01,Cortexolone 17α-propionate
Target: Androgen Receptor
Cat. No. Product Name Target Signaling Pathways
T5040 Medroxyprogesterone

羟孕酮,甲孕酮

Estrogen/progestogen Receptor; Progesterone Receptor Endocrinology/Hormones; Others
Medroxyprogesterone 是一种合成的人孕酮变体,是孕酮受体激动剂,用于治疗肾癌。在兽医实践中用作发情调节剂。
T1429 17α-Hydroxyprogesterone

Hydroxyprogesterone,17-OHP,羟孕酮,17-Hydroxyprogesterone,17α-羟孕酮

Estrogen/progestogen Receptor; Progesterone Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism; Others
17α-Hydroxyprogesterone (17-OHP) 是一种内源性孕激素,其他类固醇激素(包括糖皮质激素,雌激素,和雄激素)生物合成的化学中间体。
T1261 Medroxyprogesterone Acetate

Medroxyprogesterone 17-acetate,Provera,Metigestrona,NSC-26386,醋酸甲羟孕酮,Farlutin,安宫黄体酮,Medroxyprogesterone (acetate)

Glucocorticoid Receptor; Estrogen/progestogen Receptor; Progesterone Receptor; Androgen Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism; Others
Medroxyprogesterone Acetate (Farlutin) 是广泛使用的合成类固醇,与雄激素,孕酮及糖皮质激素受体均有作用。
TCA2511 11Beta-hydroxyprogesterone

Sodium Channel Membrane transporter/Ion channel
The progesterone derivatives 11 alpha- and 11 beta-hydroxyprogesterone are potent inhibitors of 11 beta-hydroxysteroid dehydrogenase (isoforms 1 and 2) in vitro and can confer mineralocorticoid activity on corticosterone in the rat in vivo. 11beta-Hydroxyprogesterone acts as a mineralocorticoid agonist in stimulating Na+ absorption in mammalian principal cortical collecting duct cells.

天然产物

Medroxyprogesterone
Cat.No: T5040
Synonym: 羟孕酮,甲孕酮
Target: Estrogen/progestogen Receptor, Progesterone Receptor
17α-Hydroxyprogesterone
Cat.No: T1429
Synonym: Hydroxyprogesterone,17-OHP,羟孕酮,17-Hydroxyprogesterone,17α-羟孕酮
Target: Estrogen/progestogen Receptor, Progesterone Receptor, Endogenous Metabolite
Medroxyprogesterone Acetate
Cat.No: T1261
Synonym: Medroxyprogesterone 17-acetate,Provera,Metigestrona,NSC-26386,醋酸甲羟孕酮,Farlutin,安宫黄体酮,Medroxyprogesterone (acetate)
Target: Glucocorticoid Receptor, Estrogen/progestogen Receptor, Progesterone Receptor, Androgen Receptor, Endogenous Metabolite
11Beta-hydroxyprogesterone
Cat.No: TCA2511
Synonym:
Target: Sodium Channel
TargetMol Loading
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