Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10061 |
(1S,2S)-Bortezomib
Bortezomib,硼替佐米(1S,2S) |
Proteasome | Proteases/Proteasome; Ubiquitination |
(1S,2S)-Bortezomib (Bortezomib) 是 Bortezomib 的对映异构体。 Bortezomib 是一种可逆的选择性蛋白酶体抑制剂,对 20S 蛋白酶体的 Ki 为 0.6 nM。 | |||
T2399 |
Bortezomib
Radiciol,NSC 681239,硼替佐米,MG 341,DPBA,Brotezamide,LDP 341 |
Apoptosis; NF-κB; Proteasome; Autophagy | Apoptosis; Autophagy; NF-κB; Proteases/Proteasome; Ubiquitination |
Bortezomib (LDP 341) 是一种 20S 蛋白酶体抑制剂 (Ki=0.6 nM),具有可逆性和选择性。Bortezomib 具有抗肿瘤活性,可以抑制 NF-κB,可破坏细胞周期、诱导细胞凋亡。 | |||
T67019 |
(S)-3-Phenyl-2-(pyrazine-2-carboxamido)propanoic acid
N-(Pyrazinylcarbonyl)-L-phenylalanine |
Others | Others |
(S)-3-Phenyl-2-(pyrazine-2-carboxamido)propanoic acid 是一种生化试剂,可用于生物研究。 | |||
T7854 |
Bortezomib-pinanediol
|
Proteasome | Proteases/Proteasome; Ubiquitination |
Bortezomib-pinanediol 是一种蛋白酶体抑制剂。是硼替佐米的前药。 |