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Cat. No. Product Name Target Signaling Pathways
T1435 Praziquantel

吡喹酮,Pyquiton,Droncit,Biltricide

Calcium Channel; Antibiotic; Parasite Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Praziquantel (Droncit) 是一种外消旋混合物,由 (R)-Praziquantel 和 (S)-Praziquantel 组成。它可研究血吸虫病。
T19527 Praziquantel D11

吡喹酮 D11

Others Others
Praziquantel D11 is the deuterium labeled Praziquantel, and is an agent of anthelmintic.
T12638 (R)-Praziquantel-d11

(R)-吡喹酮 D11,(R)-Praziquantel D11

5-HT Receptor GPCR/G Protein; Neuroscience
(R)-Praziquantel D11 is the deuterium labeled (R)-Praziquantel. (R)-Praziquantel is the active enantiomer of Praziquantel, is a partial the human 5-HT2B receptor agonist
T8818 TC-G 1005

(4-环丙基-3,4-二氢-1(2H)-喹喔啉基)[4-(2,5-二甲基苯氧基)-3-吡啶基]甲酮

GPCR19 GPCR/G Protein
TC-G 1005 是具有口服活性的TGR5选择性激动剂,能够激活 hTGR5 (EC50:0.72 nM)和 mTGR5 (EC50:6.2 nM)。它能够减少小鼠体内葡萄糖水平。

化合物

Praziquantel
Cat.No: T1435
Synonym: 吡喹酮,Pyquiton,Droncit,Biltricide
Target: Calcium Channel, Antibiotic, Parasite
Praziquantel D11
Cat.No: T19527
Synonym: 吡喹酮 D11
Target: Others
(R)-Praziquantel-d11
Cat.No: T12638
Synonym: (R)-吡喹酮 D11,(R)-Praziquantel D11
Target: 5-HT Receptor
TC-G 1005
Cat.No: T8818
Synonym: (4-环丙基-3,4-二氢-1(2H)-喹喔啉基)[4-(2,5-二甲基苯氧基)-3-吡啶基]甲酮
Target: GPCR19
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