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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T0839 Ketoprofen

酮基布洛芬,RP-19583,酮洛芬

Apoptosis; COX; MRP Apoptosis; Immunology/Inflammation; Neuroscience
Ketoprofen (RP-19583) 是一种非甾体抗炎剂,能够有效地抑制COX 的活性,在人血单核细胞中,对 COX-1 和 COX-2 的IC50值分别为 2 nM 和 26 nM。
T35854 9(Z),11(E)-Conjugated Linoleic Acid (sodium salt)

9(Z),11(E)-Conjugated linoleic acid is an isomer of linoleic acid that has been found in beef and milk fat.1It binds to peroxisome proliferator-activated receptor α (PPARα; IC50= 140 nM) and activates the receptor in a reporter assay using COS-1 cells expressing mouse PPARα when used at a concentration of 100 μM.29(Z),11(E)-Conjugated linoleic acid inhibits TNF-α-inducedGLUT4expression and increases insulin-stimulated glucose transport in 3T3-L1 adipocytes.3Dietary administration of 9(Z)11(E)-co...

化合物

Ketoprofen
Cat.No: T0839
Synonym: 酮基布洛芬,RP-19583,酮洛芬
Target: Apoptosis, COX, MRP
9(Z),11(E)-Conjugated Linoleic Acid (sodium salt)
Cat.No: T35854
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T19924 Rhododendrol

Betuligenol,Frambinol,杜鹃醇

Others Others
Rhododendrol (Frambinol) 是一种黑色素合成物,防止雄性小鼠高脂饮食引起的体重升高和增加雄性小鼠白色脂肪细胞的脂肪分解。Rhododendrol 可用作美白/美白化妆品抑制剂。

天然产物

Rhododendrol
Cat.No: T19924
Synonym: Betuligenol,Frambinol,杜鹃醇
Target: Others
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