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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T9347 EAAT2 activator 1

3-[(2-Chloro-6-fluorobenzyl)thio]-6-pyridin-2-ylpyridazine

transporter Metabolism
EAAT2 activator 1 (3-[(2-Chloro-6-fluorobenzyl)thio]-6-pyridin-2-ylpyridazine) 是兴奋性氨基酸转运蛋白 2(EAAT2) 的有效激活剂,以剂量依赖性方式增加 EAAT2 蛋白水平。
T9379 L-Threonic acid magnesium salt

Others Others
L-Threonic acid magnesium salt 可增加老年大鼠和晚期阿尔茨海默病 (AD) 模型小鼠的突触密度和记忆能力。
T26408 A 21960

Ethyl 2-chloroacetoacetate,A21960,A-21960

A 21960 (Ethyl 2-chloroacetoacetate) 能抑制 resolvase 与两个直接重复的 res 位点之间的突触形成,阻断位点特异性重组反应,可用于研究细菌感染。
TP1223L Apamin acetate

Apamine acetate,Apamin acetate(24345-16-2 Free base)

Potassium Channel Membrane transporter/Ion channel
Apamin acetate (Apamine acetate) 是一种具有选择性的 Ca2+ 激活的 K+ (SK) 通道的阻断剂,是在蜂毒素中发现的一种 18 个氨基酸的肽类神经毒素。Apamin acetate 可增强皮质神经元撕裂损伤后的神经突生长和再生。Apamin acetate 具有抗炎和抗纤维化的作用。
T26407 A 20832

A-20832,A20832

A-20832 inhibits resolvase-promoted site-specific recombination postsynaptically at strand cleavage. It does not inhibit resolvase binding to res, as measured by filter binding, or synapse formation. DNase I analysis in the presence of A-20832 indicates t
T76998 Cevostamab

Cevostamab(BFCR4350A; RG6160; RO7187797)为一种人源化IgG1基型双特异性抗体(BsAb),特异性结合多发性骨髓瘤(MM)细胞表面FcRH5的近膜端胞外结构域及T细胞CD3,促进高效的免疫突触形成,增强T细胞对MM肿瘤细胞的杀伤能力。
T35436 (-)-L-threo-PDMP (hydrochloride)

(-)-L-threo-PDMP is an enhancer of ganglioside biosynthesis. The (-)-L-threo-PDMP (1S,2S) isomer is the active stimulatory component of DL-threo-PDMP in contrast to (+)-D-threo-PDMP , which is an inhibitor of glucosylceramide synthetase. (-)-L-threo-PDMP upregulates GM3, GD3, and GQ1b synthase levels, which are glycosyltransferases involved in ganglioside biosynthesis, and increases ganglioside levels in cells. It increases neurite outgrowth and synapse formation in vitro and improves retention ...
T76221 Leptin (116-130)

Leptin(116-130)是一种生物活性的瘦素片段,能促进AMPA受体运输至突触并加强活动依赖性的海马突触可塑性。此外,Leptin(116-130)在抗淀粉样蛋白毒性模型中有效阻止海马突触损伤和神经元细胞死亡,显示出对研究阿尔茨海默病(AD)具有重要潜力。
T35892 Q134R

Q134R

Q134R, a neuroprotective hydroxyquinoline derivative that suppresses nuclear factor of activated T cell (NFAT) signaling. Q134R can across blood-brain barrier. Q134R has the potential for Alzheimer’s disease (AD) and aging-related disorders research[1]. Q134R (1-10 μM) suppresses NFAT signaling, without inhibiting calcineurin activity. Q134R partially inhibits NFAT activity in primary rat astrocytes, but does not prevent calcineurin-mediated dephosphorylation of a non-NFAT target, either in vivo...

化合物

EAAT2 activator 1
Cat.No: T9347
Synonym: 3-[(2-Chloro-6-fluorobenzyl)thio]-6-pyridin-2-ylpyridazine
Target: transporter
L-Threonic acid magnesium salt
Cat.No: T9379
Synonym:
Target: Others
A 21960
Cat.No: T26408
Synonym: Ethyl 2-chloroacetoacetate,A21960,A-21960
Target:
Apamin acetate
Cat.No: TP1223L
Synonym: Apamine acetate,Apamin acetate(24345-16-2 Free base)
Target: Potassium Channel
A 20832
Cat.No: T26407
Synonym: A-20832,A20832
Target:
Cevostamab
Cat.No: T76998
Synonym:
Target:
(-)-L-threo-PDMP (hydrochloride)
Cat.No: T35436
Synonym:
Target:
Leptin (116-130)
Cat.No: T76221
Synonym:
Target:
Q134R
Cat.No: T35892
Synonym: Q134R
Target:
Cat. No. Product Name Target Signaling Pathways
TN2100 Pratensein

红车轴草素,三叶草

Others; NF-κB NF-κB; Others
Pratensein 是黄酮类化合物,能够减少氧化损伤和恢复突触和 BDNF 水平,改善 β-淀粉样蛋白诱导的大鼠认知障碍。

天然产物

Pratensein
Cat.No: TN2100
Synonym: 红车轴草素,三叶草
Target: Others, NF-κB
TargetMol Loading
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