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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T1496 Amiodarone hydrochloride

盐酸胺碘酮,Amiodar,Amiodarone HCl,Nexterone

Potassium Channel; Adrenergic Receptor; Autophagy Autophagy; GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Amiodarone hydrochloride (Amiodarone HCl) 是一种抗心绞痛和 III 类抗心律失常药物,通过抑制钾通道和电压门控钠通道来增加心室和心房肌肉作用的持续时间,可导致心率和血管阻力降低。它通过成纤维细胞中的 ERK1/2和 p38 MAPK 信号传导诱导细胞增殖和肌成纤维细胞分化,可研究室上性和室性心律失常。
T8581 Flecainide hydrochloride

Others Others
Flecainide hydrochloride 是一种用于预防和治疗异常快速心率的药物。这包括室性和室上性心动过速。
T15257 Etripamil

MSP-2017,(-)-MSP-2017

Calcium Channel Membrane transporter/Ion channel; Metabolism
Etripamil (MSP-2017) 是一种短效L 型钙通道拮抗剂,可用于治疗阵发性室上性心动过速的研究。它通过抑制房室结细胞中钙慢通道的钙离子流入,显示房室结传导并延长房室结不应期
T40777 Encainide

Encainide,MJ9067

Encainide (MJ9067), a class IC antiarrhythmic drug, holds potential for research into life-threatening and symptomatic ventricular arrhythmias as well as supraventricular arrhythmias.
T21373 Aprindine hydrochloride

Fiboran,Amidonal,Aprinidine,Aprindin,Aprindine HCl,Aprindina,Fibocil

Aprindine HCl is a Class 1b antiarrhythmic agent used to manage ventricular and supraventricular arrhythmias. In one study, it delayed atrial fibrillation more than digoxin did. It has shown effectiveness when given orally.
T21391 Flecainide

Tambocor,Apocard,Flecainida,Flecainidum

Flecainide acetate is a class Ic antiarrhythmic agent, it is used to treat a variety of cardiac arrhythmias including paroxysmal atrial fibrillation, paroxysmal supraventricular tachycardia, and ventricular tachycardia. It works by regulating the flow of
T71228 Adaprolol maleate

Adaprolol maleate is a beta-blocker and opthalmic which may be used in the treatment of Glaucoma or other ailments of the eye. Adaprolol has marked electrophysiologic effects. Its major action was on sinus node; it prolonged the basic sinus cycle length and had significant effect on intrinsic automaticity as reflected by the prolonged corrected sinus node recovery time and sinuatrial conduction time. There was, also, direct effect on atrial function and AV nodal function. Adaprolol prolonged the...

化合物

Amiodarone hydrochloride
Cat.No: T1496
Synonym: 盐酸胺碘酮,Amiodar,Amiodarone HCl,Nexterone
Target: Potassium Channel, Adrenergic Receptor, Autophagy
Flecainide hydrochloride
Cat.No: T8581
Synonym:
Target: Others
Etripamil
Cat.No: T15257
Synonym: MSP-2017,(-)-MSP-2017
Target: Calcium Channel
Encainide
Cat.No: T40777
Synonym: Encainide,MJ9067
Target:
Aprindine hydrochloride
Cat.No: T21373
Synonym: Fiboran,Amidonal,Aprinidine,Aprindin,Aprindine HCl,Aprindina,Fibocil
Target:
Flecainide
Cat.No: T21391
Synonym: Tambocor,Apocard,Flecainida,Flecainidum
Target:
Adaprolol maleate
Cat.No: T71228
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T8183 Deslanoside

洋地黄,去乙酰西地兰,Desacetyllanatoside C,Deacetyllanatoside C

ATPase; Drug Metabolite Membrane transporter/Ion channel; Metabolism
Deslanoside (Desacetyllanatoside C) 是一种快速作用的强心苷,可抑制Na-K-ATPase 膜泵,导致细胞内钠和钙浓度增加。它用于研究充血性心力衰竭和因折返机制引起的室上性心律失常,并在研究慢性心房颤动时控制心室率。

天然产物

Deslanoside
Cat.No: T8183
Synonym: 洋地黄,去乙酰西地兰,Desacetyllanatoside C,Deacetyllanatoside C
Target: ATPase, Drug Metabolite
TargetMol Loading
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