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抑制剂 & 化合物

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Cat. No.	Product Name	Target	Signaling Pathways
T82450	ER proteostasis regulator-1
	ER proteostasis regulator-1 (化合物481) 是高效的内质网蛋白稳态调节剂，其在阿尔茨海默病与糖尿病研究领域显示出潜在应用价值。
T36670	JNJ-67856633	MALT	Immunology/Inflammation
	JNJ-67856633 是口服有效的、选择性的、变构性的 MALT1 protease 抑制剂。在某些情况下，JNJ-67856633可以导致肿瘤停滞。
T69152	Bromopride hydrochloride
	Bromopride hydrochloride is the salt form of Bromopride, a dopamine D2 receptor blocker. Bromopride exerts is a gastrointestinal prokinetic exploited clinically for the management of motor disorders of the upper gastrointestinal tract, including functional dyspepsia, gastric stasis of various origins and emesis.
T64250	Desirudin
	Desirudin (CGP 39393) 是一种凝血酶 (thrombin) 抑制剂，能够抑制血栓形成和静脉淤血性血栓形成。Desirudin 能够用于研究血小板减少症或血小板功能障碍相关。
T63793	Tauro-ω-muricholic acid sodium
	Tauro-ω-muricholic acid sodium (TωMCA sodium) 是一种tauro-α-muricholic acid 的类似物，是来源于肝脏的胆汁酸。Tauro-ω-muricholic acid sodium 能用作早发性新生儿败血症 (EOS) 和胆汁淤积的血清标志物。
T68332	AKI-001
	AKI-001 is a potent Aurora kinase inhibitor, which exhibits low nanomolar potency against both Aurora A and Aurora B enzymes, excellent cellular potency (IC50 < 100 nM), and good oral bioavailability. Phenotypic cellular assays show that both Aurora A and Aurora B are inhibited at inhibitor concentrations sufficient to block proliferation. Importantly, the cellular activity translates to potent inhibition of tumor growth in vivo. An oral dose of 5 mg/kg QD is well tolerated and results in near s...

化合物

ER proteostasis regulator-1

Bromopride hydrochloride

Tauro-ω-muricholic acid sodium

Cat. No.	Product Name	Target	Signaling Pathways
T4S0592	Toddalolactone (+)-Toddalolactone,飞龙掌血内酯,毛两面针素	PAI-1	Metabolism
	Toddalolactone ((+)-Toddalolactone) 是一种Toddalia asiatica 的主要成分，能够抑制重组人纤溶酶原激活物抑制物-1(PAI-1)的活性， IC50=37.31 μM。
T5769	Stachydrine Methyl hygrate betaine,水苏碱,L-stachydrine,Proline betaine,N,N-Dimethyl-L-proline	NF-κB; Endogenous Metabolite	Metabolism; NF-κB
	Stachydrine (N,N-Dimethyl-L-proline) 是中国草本植物益母草的主要成分，具有促进血液循环和消除血瘀的功效。Stachydrine (N,N-Dimethyl-L-proline) 能够抑制NF-κB 信号通路。
TN1000	Solasurine	Others	Others
	Solasurine is a natural product with dissipate blood stasis and detumescence, relieve pain and pull poison.