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Cat. No. | Product Name | Target | Signaling Pathways |
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T27794 |
λ-Cyhalothrin
lambda-Cyhalothrin,Karate,λ-氯氟氰菊酯,Icon |
Sodium Channel; Parasite | Membrane transporter/Ion channel; Microbiology/Virology |
λ-Cyhalothrin (Icon) 是广谱的 II 型合成除虫菊酯杀虫剂,含有 α-氰基,用于防治多种害虫。它是一种钠通道神经毒素,靶向中枢神经系统中神经元膜。 | |||
T2390 |
Cevimeline hydrochloride hemihydrate
|
AChR | Neuroscience |
Cevimeline hydrochloride hemihydrate 是乙酰胆碱的奎尼丁衍生物,也是选择性的和口服活性的毒蕈碱型M1和M3受体激动剂。它可穿过血脑屏障,刺激唾液腺分泌,用作口干症的催涎剂。 | |||
T2387 |
Glycopyrrolate
Gastrodyn,Glycopyrronium bromide,Robinul,Glycopyrrolate bromide,格隆溴铵 |
AChR | Neuroscience |
Glycopyrrolate (Glycopyrrolate bromide) 是一种毒蕈碱拮抗剂,在某些胃肠道疾病中用作解痉剂,并与某些麻醉剂一起减少唾液分泌。 | |||
T20713 |
Flonicamid
UNII-9500W2Z53J,N-(cyanomethyl)-4-(trifluoromethyl)nicotinamide |
Others | Others |
Flonicamid (N-(cyanomethyl)-4-(trifluoromethyl)nicotinamide) 是一种吡啶甲酰胺杀虫剂,在食用日本萝卜叶的过程中抑制蚜虫(M.persicae)的唾液分泌和汁液摄入。它对棉蚜、红蚜、巴迪蚜、禾谷蚜和大鼠产生毒性。 | |||
T13615 |
Cinperene
桂哌林,R5046 |
Others | Others |
Cinperene is an atropine-like compound that can block pilocarpine-induced salivation and lacrimation. | |||
T71541 | ASP9133 | ||
ASP9133 is a long-acting muscarinic antagonist (LAMA) which shows more selective inhibition of bronchoconstriction against salivation and more rapid onset of action than tiotropium bromide. | |||
T25912 |
Oxypyrronium bromide
L.D. 3055,Immetropan,LD 3055,LD3055,LD-3055 |
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Oxypyrronium bromide 一种含有季铵的抗胆碱能和解痉剂。在动物模型中,它抑制胃运动、迷走神经刺激或乙酰胆碱静脉注射引起的低血压;鼓索神经刺激引起的流涎和节前颈交感神经刺激引起收缩。 | |||
T36204 |
Methylatropine (nitrate)
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Methylatropine is an antagonist of muscarinic acetylcholine receptors (IC50= <0.1 nM in a radioligand binding assay using isolated porcine brain membranes) and a derivative of atropine .1,2It reduces acetylcholine-induced decreases in blood pressure in rats when administered intravenously with an ED50value of 5.5 μg/kg.2Methylatropine reduces salivation, induces mydriasis, and increases heart rate in dogs.3 1.Schmeller, T., Sporer, F., Sauerwein, M., et al.Binding of tropane alkaloids to nicotin... |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1285 |
Anethole trithione
茴三硫,Anetholtrithion |
Others; AChR | Neuroscience; Others |
Anethole trithione (Anetholtrithion) 是硫杂环胆碱,是一种胆汁分泌刺激剂,可增强唾液分泌并增加 mAChR 受体,用于口干症的研究。 |