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Search Results for " radiosensitivity "

6

抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
TQ0219 MK-8033

c-Met/HGFR Tyrosine Kinase/Adaptors
MK-8033 是一种新型ATP 竞争性c-Met/Ron 双重抑制剂,对野生型c-Met 的IC50=1 nM,对c-Met N1100Y 的IC50=2.0 nM。
T61189 E7016

GPI 21016

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
E7016 (GPI 21016) (GPI 21016) 是一种口服有效的 PARP 抑制剂。E7016 可以通过抑制 DNA 修复来增强肿瘤细胞在体内外的放射敏感性。
T40066 SENP1-IN-3

SENP1-IN-3

SENP1-IN-3 is a distinct inhibitor of the deSUMOylation protease 1 (SENP1), designed to enhance tumor radiosensitivity.
T40067 SENP1-IN-4

SENP1-IN-4

SENP1-IN-4, a distinct inhibitor of the deSUMOylation protease 1 (SENP1), is designed to enhance tumor radiosensitivity.
T40068 SENP1-IN-1

SENP1-IN-1

SENP1-IN-1 is a distinct inhibitor of the deSUMOylation protease 1 (SENP1), designed to enhance tumor radiosensitivity.
T40069 SENP1-IN-2

SENP1-IN-2

SENP1-IN-2, a distinct inhibitor of the deSUMOylation protease 1 (SENP1), is designed to enhance tumor radiosensitivity.

化合物

MK-8033
Cat.No: TQ0219
Synonym:
Target: c-Met/HGFR
E7016
Cat.No: T61189
Synonym: GPI 21016
Target: PARP
SENP1-IN-3
Cat.No: T40066
Synonym: SENP1-IN-3
Target:
SENP1-IN-4
Cat.No: T40067
Synonym: SENP1-IN-4
Target:
SENP1-IN-1
Cat.No: T40068
Synonym: SENP1-IN-1
Target:
SENP1-IN-2
Cat.No: T40069
Synonym: SENP1-IN-2
Target:
Cat. No. Product Name Target Signaling Pathways
T10021 1-Methylxanthine

Endogenous Metabolite Metabolism
1-Methylxanthine 是咖啡因衍生物,是咖啡因和茶碱 (1,3-二甲基黄嘌呤,TP) 在人体尿代谢产物,能够提高肿瘤细胞的放射敏感性。

天然产物

1-Methylxanthine
Cat.No: T10021
Synonym:
Target: Endogenous Metabolite
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