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Cat. No. Product Name Target Signaling Pathways
T21981 Phthalazinone pyrazole

Aurora Kinase Cell Cycle/Checkpoint; Chromatin/Epigenetic
Phthalazinone pyrazole 是强效、选择性和口服生物可利用的 Aurora-A 激酶抑制剂,IC50值为 0.031 μM。它抑制人胚胎干细胞向肝细胞样细胞分化过程中的上皮间质转化。它还可阻止有丝分裂并随后通过增殖细胞的凋亡抑制肿瘤生长。
T9891 PARP1-IN-8 

N-(3-chlorophenyl)-3-(1-oxo-4-phenylphthalazin-2(1H)-yl)propanamide

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
PARP1-IN-8 (N-(3-chlorophenyl)-3-(1-oxo-4-phenylphthalazin-2(1H)-yl)propanamide) 是PARP1的有效抑制剂(IC50 = 97 nM)。
T0211L Azelastine hydrochloride

Optivar,Azelastine HCl,Allergodil,盐酸氮卓斯汀,Astelin

SARS-CoV; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Azelastine hydrochloride (Astelin) 是一种选择性组胺 1拮抗剂,可研究过敏性鼻炎、哮喘、糖尿病高脂血症和 SARS-CoV-2 。
T36747 HBV-IN-4

HBV-IN-4, a derivative of phthalazinone, functions as a potent, orally active inhibitor of HBV DNA replication, exhibiting an IC50 value of 14 nM. It effectively induces the formation of genome-free capsids, demonstrating significant anti-HBV potency[1].

化合物

Phthalazinone pyrazole
Cat.No: T21981
Synonym:
Target: Aurora Kinase
PARP1-IN-8 
Cat.No: T9891
Synonym: N-(3-chlorophenyl)-3-(1-oxo-4-phenylphthalazin-2(1H)-yl)propanamide
Target: PARP
Azelastine hydrochloride
Cat.No: T0211L
Synonym: Optivar,Azelastine HCl,Allergodil,盐酸氮卓斯汀,Astelin
Target: SARS-CoV, Histamine Receptor
HBV-IN-4
Cat.No: T36747
Synonym:
Target:
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