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2

抑制剂 & 化合物

4

天然产物

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Cat. No. Product Name Target Signaling Pathways
T32528 Lacticolorin

Lacticolorin is a phenolic glucoside ester; metabolite of Protea lacticolor Salisb.
T19303 (E/Z)-Methyl mycophenolate

Others Others
Methyl mycophenolate can be used to synthesize mycophenolic acid β-D-glucuronide and phenolic glycosides. (E/Z)-Methyl mycophenolate is a racemic compound of (Z)-Methyl mycophenolate and (E)-Methyl mycophenolate isomers. Methyl mycophenolate is a methyl e

化合物

Lacticolorin
Cat.No: T32528
Synonym:
Target:
(E/Z)-Methyl mycophenolate
Cat.No: T19303
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T9933 Methyl 2,4-dihydroxyphenylacetate

Others Others
Methyl 2,4-dihydroxyphenylacetate 是从 Nigella damascena 种子中分离得到的天然产物,具有选择性的植物毒性作用。
T2784 Ethyl Orsellinate

苷色酸乙酯,山梨酸乙酯,Orsellinic acid ethyl ester

Others; Antibacterial Microbiology/Virology; Others
Ethyl Orsellinate (Orsellinic acid ethyl ester) 是地衣代谢产物,抑制A.salina 的细胞毒性活性,IC50为 495 μM。它是 lecanoric acid 的衍生物,具有抗增殖和抗肿瘤活性。
TL0004 FERULIC ACID METHYL ESTER

阿魏酸甲酯,Methyl ferulate,Methyl 4'-hydroxy-3'-methoxycinnamate

p38 MAPK; Autophagy Autophagy; MAPK
FERULIC ACID METHYL ESTER (Methyl ferulate) 是从大百部中分到的阿魏酸衍生物,具有抗氧化和抗炎作用。在原发性骨髓源性巨噬细胞中,它抑制 COX-2 的表达,降低 p-p38和 p-JNK 的水平。它能够透过细胞膜和血脑屏障,清除自由基,可研究神经退行性疾病。
T3392 Sinapine thiocyanate

P-gp; AChE Membrane transporter/Ion channel; Neuroscience
Sinapine thiocyanate 是萝卜中分离出来的一种生物碱,具有抗炎、抗氧化、抗肿瘤、抗血管生成和放射防护作用。它还是乙酰胆碱酯酶抑制剂,可用于研究阿尔茨海默症,共济失调,重症肌无力和帕金森氏病。

天然产物

Methyl 2,4-dihydroxyphenylacetate
Cat.No: T9933
Synonym:
Target: Others
Ethyl Orsellinate
Cat.No: T2784
Synonym: 苷色酸乙酯,山梨酸乙酯,Orsellinic acid ethyl ester
Target: Others, Antibacterial
FERULIC ACID METHYL ESTER
Cat.No: TL0004
Synonym: 阿魏酸甲酯,Methyl ferulate,Methyl 4'-hydroxy-3'-methoxycinnamate
Target: p38 MAPK, Autophagy
Sinapine thiocyanate
Cat.No: T3392
Synonym:
Target: P-gp, AChE
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