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Cat. No. Product Name Target Signaling Pathways
T0255 Clomipramine hydrochloride

Clomipramine HCl,Anafranil,盐酸氯米帕明

Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Norepinephrine; GST GPCR/G Protein; Neuroscience; oxidation-reduction
Clomipramine hydrochloride (Anafranil) 是一种5-羟色胺转运体(Ki:0.14 nM)、去甲肾上腺素转运体(Ki:54 nM)和多巴胺转运体(Ki:3 nM)阻断剂。
T21013 Clomipramine

Chlorimipramine,Anafranil,Clomicalm,Anafranil (free base),Clomipramina,氯米帕明

5-HT Receptor GPCR/G Protein; Neuroscience
Clomipramine (Clomicalm) 是一种三环类抗抑郁药,能够有效阻断 5-HT 再摄取 (IC50:1.5 nM) ,可用于研究强迫症 (OCD) 及抑郁症。
T69364 Elzasonan

Elzasonan is a selective 5-hydroxytryptamine 1B receptor antagonist used to treat patients with major depressive disorder and obsessive compulsive disorder.
T68683 Sertraline Free Base

Sertraline Free Base is a Selective Serotonin Reuptake Inhibitor (SSRI). It can treat depression, obsessive-compulsive disorder (OCD), posttraumatic stress disorder (PTSD), premenstrual dysphoric disorder (PMDD), social anxiety disorder, and panic disorder.
T71389 Fluoxetine oxalate

Fluoxetine oxalate is an antidepressant of the selective serotonin reuptake inhibitor (SSRI) class. It is used for the treatment of major depressive disorder, obsessivecompulsive disorder, bulimia nervosa, panic disorder, and premenstrual dysphoric disorder.
T71587 Fluoxetine succinate ester

Fluoxetine succinate ester is an antidepressant of the selective serotonin reuptake inhibitor (SSRI) class. It is used for the treatment of major depressive disorder, obsessivecompulsive disorder, bulimia nervosa, panic disorder, and premenstrual dysphoric disorder.
T68579 Fluvoxamine acid

Fluvoxamine acid is a medication which functions as a selective serotonin reuptake inhibitor (SSRI) and σ1 receptor agonist. Fluvoxamine is used primarily for the treatment of obsessive-compulsive disorder (OCD), and is also used to treat major depressive disorder (MDD), and anxiety disorders such as panic disorder and post-traumatic stress disorder (PTSD).
T60966 UCPH-102

UCPH-102 可用于研究阿尔茨海默病、肌萎缩性侧索硬化症、慢性疼痛和强迫症等,具有良好的血脑通透性。UCPH-102 是高度选择性的 EAAT1抑制剂,IC50值为0.43 μM。UCPH-102 还对 T-ALL 细胞表现出特异性的抗增殖作用。

化合物

Clomipramine hydrochloride
Cat.No: T0255
Synonym: Clomipramine HCl,Anafranil,盐酸氯米帕明
Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Norepinephrine, GST
Clomipramine
Cat.No: T21013
Synonym: Chlorimipramine,Anafranil,Clomicalm,Anafranil (free base),Clomipramina,氯米帕明
Target: 5-HT Receptor
Elzasonan
Cat.No: T69364
Synonym:
Target:
Sertraline Free Base
Cat.No: T68683
Synonym:
Target:
Fluoxetine oxalate
Cat.No: T71389
Synonym:
Target:
Fluoxetine succinate ester
Cat.No: T71587
Synonym:
Target:
Fluvoxamine acid
Cat.No: T68579
Synonym:
Target:
UCPH-102
Cat.No: T60966
Synonym:
Target:
TargetMol Loading
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