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抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T2711 Chembridge-5861528

TCS 5861528

TRP/TRPV Channel Membrane transporter/Ion channel
Chembridge-5861528 (TCS 5861528) 是有效的 TRPA1离子通道阻断剂。
T9263 cim0216

N-(5-methyl-1,2-oxazol-3-yl)-2-phenyl-2-(1,2,3,4-tetrahydroquinolin-1-yl)acetamide

TRP/TRPV Channel Membrane transporter/Ion channel
CIM0216 是选择性的TRPM3激动剂,对 TRPM3 的选择性高于 TRPM1、TRPM2 和 TRPM4-8。它以TRPM3依赖性的方式引起疼痛并唤起感觉神经末梢的神经肽释放,可用于神经源性炎症的相关研究。
T25615 Lanepitant

LY303870,LY-303870,LY 303870

Others Others
Lanepitant (LY303870) 是一种非肽类神经激肽-1(NK-1)拮抗剂,具有镇痛活性,可抑制神经源性硬脑膜炎症,可用于预防偏头痛。
T25616 Lanepitant 2HCl

LY303870 dihydrochloride,LY 303870 dihydrochloride,LY-303870 dihydrochloride,Lanepitant dihydrochloride

Neurokinin receptor GPCR/G Protein; Neuroscience
Lanepitant 2HCl 是一种非肽类神经激肽-1 受体拮抗剂,具有镇痛和抗炎活性。Lanepitant 2HCl 抑制 P 物质与神经激肽-1 受体的结合,抑制神经源性炎症和疼痛传递,可用于研究偏头痛等疼痛性神经病变类疾病。
T27059 CP-122288

CP-122288 is a potent and selective agonist for the 5-HT1B, 5-HT1D and 5-HT1F serotonin receptor subtypes. CP-122288 is potent as an inhibitor of plasma protein extravasation and neurogenic inflammation.
T27915 LY 302148

LY-302148,LY302148

LY 302148 , a 5-HT1F receptor agonist, inhibits neurogenic dural inflammation in guinea pigs. It has potential for migraine therapeutics.
T28516 ReN-1869

NNC-05-1869,NNC 05-1869,NNC-051869,ReN 1869

ReN-1869 is a histamine H1 receptor antagonist. ReN 1869 is active against inflammation and neurogenic pain. ReN-1869 produces potent and selective antinociceptive effects on dorsal horn neurons after inflammation and neuropathy.
T25617 Lanepitant HCl trihydrate

Lanepitant dihydrochloride trihydrate

Lanepitant HCl trihydrate is an effective non-peptide neurokinin-1 receptor antagonist, suppresses neurogenic dural inflammation, and may have a role in migraine therapy.
T76429 Neurokinin Receptor (393-407), rat

Neurokinin Receptor(393-407), rat (SPR393–407) 是一段属于大鼠神经激肽1受体(NK1R)的特定肽。它与P物质(SP)结合后,通过内吞作用迅速被NK1R内化,并循环至质膜。此化合物主要应用于神经源性炎症研究领域。

化合物

Chembridge-5861528
Cat.No: T2711
Synonym: TCS 5861528
Target: TRP/TRPV Channel
cim0216
Cat.No: T9263
Synonym: N-(5-methyl-1,2-oxazol-3-yl)-2-phenyl-2-(1,2,3,4-tetrahydroquinolin-1-yl)acetamide
Target: TRP/TRPV Channel
Lanepitant
Cat.No: T25615
Synonym: LY303870,LY-303870,LY 303870
Target: Others
Lanepitant 2HCl
Cat.No: T25616
Synonym: LY303870 dihydrochloride,LY 303870 dihydrochloride,LY-303870 dihydrochloride,Lanepitant dihydrochloride
Target: Neurokinin receptor
CP-122288
Cat.No: T27059
Synonym:
Target:
LY 302148
Cat.No: T27915
Synonym: LY-302148,LY302148
Target:
ReN-1869
Cat.No: T28516
Synonym: NNC-05-1869,NNC 05-1869,NNC-051869,ReN 1869
Target:
Lanepitant HCl trihydrate
Cat.No: T25617
Synonym: Lanepitant dihydrochloride trihydrate
Target:
Neurokinin Receptor (393-407), rat
Cat.No: T76429
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN6872 Trypsin

Protease-activated Receptor GPCR/G Protein
Trypsin 是一种可从鱼类分离出的丝氨酸蛋白酶,可水解赖氨酸或精氨酸羧基侧蛋白质。Trypsin 具有抗炎活性,可通过 PDCoV 的 S 糖蛋白与 pAPN 的相互作用诱导 PDCoV 感染的细胞膜融合,可激活 PAR2 和 PAR4,促进细胞增殖和分化。Trypsin 可用于促进伤口愈合和研究神经源性炎症。

天然产物

Trypsin
Cat.No: TN6872
Synonym:
Target: Protease-activated Receptor
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