7
2
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T9530 |
W 36017
|
Others | Others |
W36017 是利多卡因的一种杂质,其阻滞神经活性的pKa 为 7.4。 | |||
T0025 |
Haloperidol
Aloperidin,氟哌啶醇,Serenace,Haldol |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Haloperidol (Serenace) 是一种安定药,是一种dopamine D2 receptor 拮抗剂。 | |||
T4497 |
Amifampridine
3,4-Pyridinediamine,Pyridine-3,4-Diamine,阿米吡啶,3,4-Diaminopyridine |
Others | Others |
Amifampridine (3,4-Diaminopyridine) 可用于罕见肌肉疾病的研究。 | |||
T70224 |
Bupivacaine tartrate
|
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Bupivacaine is a BK/SK, Kv1, Kv3, TASK-2 K Channel and voltage-gated Na channel blocker used as an anesthetic. It maybe neurotoxic at high does, inducing apoptosis in neuroblastoma cells. It acts by binding to the intracellular portion of voltage-gated sodium channels and blocking sodium influx into nerve cells. | |||
T81519 |
Pentapeptide-3
|
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Pentapeptide-3为源自韦氏腹蛇毒素waglerin-1的五肽神经毒素,作为尼古丁乙酰胆碱受体(nAChRs)的竞争性拮抗剂,能够在突触后膜发挥阻滞神经的效果。该化合物具有抗衰老功能,可与其他化妆品肽配合使用。 | |||
TMIH-0086 |
Amifampridine-d3 2HCl
|
||
Amifampridine-d3 2HCl 是 Amifampridine 2HCl 的氘代化合物。Amifampridine 2HCl 的 CAS 号为 54-96-6。Amifampridine 可用于罕见肌肉疾病的研究。 | |||
T61475 |
Ropivacaine mesylate
|
||
Ropivacaine mesylate 是一种高效的钠通道 (sodium channel) 阻断剂,通过可逆性抑制钠离子内流 (sodium ion influx),引致神经纤维脉冲传导阻滞。此外,Ropivacaine 还能抑制 K2P(双孔钾通道)TREK-1,其在 COS-7 细胞膜上的 IC50 值为 402.7 μM。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T4S1876 |
3-Deoxyaconitine
|
Sodium Channel | Membrane transporter/Ion channel |
3-Deoxyaconitine 是一种二萜类生物碱,对钠离子通道有激活作用。 | |||
T2S1727 |
Lycorenine
|
Antifection | Microbiology/Virology |
Lycorenine may produce a decrease in blood pressure as the result of alpha-adrenergic blockade in conjunction with the reduction of the spontaneous sympathetic nerve activity, and produce bradycardia by modifying vagal activity. The development of tachyph |