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7

抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T9530 W 36017

Others Others
W36017 是利多卡因的一种杂质,其阻滞神经活性的pKa 为 7.4。
T0025 Haloperidol

Aloperidin,氟哌啶醇,Serenace,Haldol

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Haloperidol (Serenace) 是一种安定药,是一种dopamine D2 receptor 拮抗剂。
T4497 Amifampridine

3,4-Pyridinediamine,Pyridine-3,4-Diamine,阿米吡啶,3,4-Diaminopyridine

Others Others
Amifampridine (3,4-Diaminopyridine) 可用于罕见肌肉疾病的研究。
T70224 Bupivacaine tartrate

Bupivacaine is a BK/SK, Kv1, Kv3, TASK-2 K Channel and voltage-gated Na channel blocker used as an anesthetic. It maybe neurotoxic at high does, inducing apoptosis in neuroblastoma cells. It acts by binding to the intracellular portion of voltage-gated sodium channels and blocking sodium influx into nerve cells.
T81519 Pentapeptide-3

Pentapeptide-3为源自韦氏腹蛇毒素waglerin-1的五肽神经毒素,作为尼古丁乙酰胆碱受体(nAChRs)的竞争性拮抗剂,能够在突触后膜发挥阻滞神经的效果。该化合物具有抗衰老功能,可与其他化妆品肽配合使用。
TMIH-0086 Amifampridine-d3 2HCl

Amifampridine-d3 2HCl 是 Amifampridine 2HCl 的氘代化合物。Amifampridine 2HCl 的 CAS 号为 54-96-6。Amifampridine 可用于罕见肌肉疾病的研究。
T61475 Ropivacaine mesylate

Ropivacaine mesylate 是一种高效的钠通道 (sodium channel) 阻断剂,通过可逆性抑制钠离子内流 (sodium ion influx),引致神经纤维脉冲传导阻滞。此外,Ropivacaine 还能抑制 K2P(双孔钾通道)TREK-1,其在 COS-7 细胞膜上的 IC50 值为 402.7 μM。

化合物

W 36017
Cat.No: T9530
Synonym:
Target: Others
Haloperidol
Cat.No: T0025
Synonym: Aloperidin,氟哌啶醇,Serenace,Haldol
Target: Dopamine Receptor, 5-HT Receptor
Amifampridine
Cat.No: T4497
Synonym: 3,4-Pyridinediamine,Pyridine-3,4-Diamine,阿米吡啶,3,4-Diaminopyridine
Target: Others
Bupivacaine tartrate
Cat.No: T70224
Synonym:
Target:
Pentapeptide-3
Cat.No: T81519
Synonym:
Target:
Amifampridine-d3 2HCl
Cat.No: TMIH-0086
Synonym:
Target:
Ropivacaine mesylate
Cat.No: T61475
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T4S1876 3-Deoxyaconitine

Sodium Channel Membrane transporter/Ion channel
3-Deoxyaconitine 是一种二萜类生物碱,对钠离子通道有激活作用。
T2S1727 Lycorenine

Antifection Microbiology/Virology
Lycorenine may produce a decrease in blood pressure as the result of alpha-adrenergic blockade in conjunction with the reduction of the spontaneous sympathetic nerve activity, and produce bradycardia by modifying vagal activity. The development of tachyph

天然产物

3-Deoxyaconitine
Cat.No: T4S1876
Synonym:
Target: Sodium Channel
Lycorenine
Cat.No: T2S1727
Synonym:
Target: Antifection
TargetMol Loading
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