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11

抑制剂 & 化合物

4

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T0203	Sumatriptan succinate 舒马普坦琥珀酸盐,GR 43175,琥珀酸舒马曲坦	5-HT Receptor	GPCR/G Protein; Neuroscience
	Sumatriptan succinate (GR 43175) 是一种5-HT1受体激动剂，可作用于偏头疼的急性治疗。
T8414	SNC 80 Snc-80,SNC80,NIH 10815	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	SNC 80 (NIH 10815) 是有效的，高度选择性的非肽类 δ 阿片 (δ-opioid) 受体激动剂，Ki 为1.78 nM，IC50 为 2.73 nM。SNC80 还以 EC50 为 52.8 nM 来选择性激活 HEK293 细胞中的 μ-δ 异聚体。SNC80 具有抗伤害性，抗痛觉过敏和抗抑郁样作用，并可用于多种头痛症的研究。
T26079	RI 61 RI-61,Pro-his-pro-phe-his-leu-phe-val-phe,RI61
	RI 61 (sumatriptan succinate) is utilized in the therapy of migraine, cluster headaches, new daily persistent headache, and cyclic vomiting syndrome.
T60989	Sumatriptan hydrochloride
	Sumatriptan (GR 43175) hydrochloride 可用于研究偏头痛，它是一种口服有效的5-HT1受体激动剂。Sumatriptan hydrochloride 对5-HT1D、5-HT1B 和5-HT1A 受体的 Ki 值分别为 17 nM、27 nM 和 100 nM。
T31671	Erythrityl Tetranitrate Eritrityli tetranitras,Tetranitrato de eritritilo,CHEBI:60072,Tetranitrate d'eritrityle
	Erythrityl Tetranitrate is a vasodilator with general properties similar to nitroglycerin. Like many nitrate esters, ETN acts as a vasodilator, and was the active ingredient in the original "sustained release" tablets, made in the early 50s. Ingesting ETN or prolonged skin contact can lead to absorption and what is known as a "nitro headache".
T60345	Frovatriptan
	Frovatriptan is a highly potent agonist of the 5-HT 1B//D receptors, exhibiting the highest potency among triptan compounds. It possesses prominent cerebroselectivity. Frovatriptan demonstrates efficacy and even superiority in certain endpoints, including when administered during the headache phase of migraine attacks accompanied by aura [1].
T69144	Hexylcaine HCl
	Hexylcaine HCl also called cyclaine or osmocaine, is a short-acting local anesthetic. It acts by inhibiting sodium channel conduction. Overdose can lead to headache, tinnitus, numbness and tingling around the mouth and tongue, convulsions, inability to breathe, and decreased heart function.
T73631	(Rac)-SNC80
	(Rac)-SNC80 是SNC80 的外消旋体。SNC80 (NIH 10815) 是一种有效的，高度选择性的非肽类 δ 阿片 (δ-opioid) 受体激动剂，Ki 为1.78 nM，IC50为 2.73 nM。SNC80 具有抗伤害性，抗痛觉过敏和抗抑郁样作用，并可用于多种头痛症的研究。
T79805	5-HT2 agonist-1 free base	5-HT Receptor	GPCR/G Protein; Neuroscience
	5-HT2 agonist-1 (Compound 24) free base 是一种作用于5-HT2A, 5-HT2B和5-HT2C受体的激动剂，其IC50值分别为10 nM, 8.3 nM和1.6 nM。该化合物主要应用于研究抑郁症、酒精依赖、烟草及可卡因成瘾、炎症、丛集性头痛、创伤后应激障碍(PTSD)、癫痫以及其他中枢神经系统相关疾病。
T70070	Cisapride tartrate
	Cisapride tartrate is chemically related to metoclopramide, but unlike metoclopramide, it does not cross the blood-brain barrier or have antidopaminergic effects. Cisapride is a serotonin-4 (5-HT4) receptor agonist. Cisapride was indicated for the symptomatic treatment of adult patients with nocturnal heartburn due to gastroesophageal reflux disease. The Food and Drug Administration (FDA) in America stopped the marketing of cisapride as of 14th July 2000. They had received at least 341 reports o...
T14614	Biperiden Hydrochloride KL 373 (Hydrochloride),盐酸比哌立登	Others	Others
	Biperiden Hydrochloride (KL 373 Hydrochloride) is an antiparkinsonian agent, which is the selective central M1 cholinoreceptors blocker and it is used for the adjunctive treatment of all forms of Parkinson's disease (postencephalitic, idiopathic, and arte

化合物

Sumatriptan succinate

Cat.No: T0203

Synonym: 舒马普坦琥珀酸盐,GR 43175,琥珀酸舒马曲坦

Target: 5-HT Receptor

Cat.No: T8414

Synonym: Snc-80,SNC80,NIH 10815

Target: Opioid Receptor

Cat.No: T26079

Synonym: RI-61,Pro-his-pro-phe-his-leu-phe-val-phe,RI61

Sumatriptan hydrochloride

Cat.No: T60989

Erythrityl Tetranitrate

Cat.No: T31671

Synonym: Eritrityli tetranitras,Tetranitrato de eritritilo,CHEBI:60072,Tetranitrate d'eritrityle

Cat.No: T60345

Cat.No: T69144

Cat.No: T73631

5-HT2 agonist-1 free base

Cat.No: T79805

Target: 5-HT Receptor

Cisapride tartrate

Cat.No: T70070

Biperiden Hydrochloride

Cat.No: T14614

Synonym: KL 373 (Hydrochloride),盐酸比哌立登

Target: Others

Cat. No.	Product Name	Target	Signaling Pathways
TN2865	(E)-3,4,5-Trimethoxycinnamic acid O-Methylsinapic acid,3,4,5-三甲氧基肉桂酸,3,4,5-Trimethoxy-trans-cinnamic acid,3,4,5-Trimethoxyphenylacrylic acid	Others	Others
	(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) 是一种来自羌活根和根茎的天然产物。
TN1610	Epimagnolin A	Parasite	Microbiology/Virology
	Epimagnolin A 是一种糠醛木脂素，具有中等的抗疟原虫活性，IC50值为5.7 μg/mL。
TN6646	Fargesol
	(-)-Fargesol is a nartural product from the flowers buds of Magnolia fargesii,the dried flower buds of M. fargesii, has been used as therapy for nasal empyema and headache.
T81584	Oxyresveratrol 4-O-β-D-glucopyranoside
	Oxyresveratrol 4-O-β-D-glucopyranoside (化合物 3)，一种从Morus atropurpurea根皮分离的天然产物，具有研究治疗糖尿病、关节炎、风湿、咳嗽及头痛的潜力。

天然产物

(E)-3,4,5-Trimethoxycinnamic acid

Cat.No: TN2865

Synonym: O-Methylsinapic acid,3,4,5-三甲氧基肉桂酸,3,4,5-Trimethoxy-trans-cinnamic acid,3,4,5-Trimethoxyphenylacrylic acid

Target: Others

Cat.No: TN1610

Target: Parasite

Cat.No: TN6646

Oxyresveratrol 4-O-β-D-glucopyranoside

Cat.No: T81584

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