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13

抑制剂 & 化合物

7

天然产物

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Cat. No. Product Name Target Signaling Pathways
T20913 Light Green SF Yellowish

Acid Green 5,C.I. Acid Green 5,C.I. 42095

Light Green SF Yellowish (Acid Green 5) 是一种碱性染色剂,可用于动物组织染色,可用于植物组织学中作细胞质和纤维染色。
T8341 QX 314

QX-314

Others Others
QX 314 (Lidocaine N-ethyl bromide) 是一种非膜渗透性阻滞剂,可抑制酸诱导的食管伤害性 C 纤维神经元活化。
TP1696L CGGRGD acetate(1260223-44-6 free base)

Others Others
CGGRGD acetate(1260223-44-6 free base) 是一种以半胱氨酸为 n 端的 RGD 衍生物。 CGGRGD 采用固相多肽合成技术合成,在PCL 纤维表面添加氨基2-氰基苯并噻唑(2-cyanobenzothiazole)(2-cyanobenzothiazole (CBT))进行氨化。
T37744 N-octanoyl-L-Homoserine lactone

C8-HSL,N-octanoyl-L-Homoserine lactone,OHL

Antibacterial Microbiology/Virology
N-octanoyl-L-Homoserine lactone (C8-HSL) 是一种具有扩散性的外源性鼠疫耶尔森菌群体感应分子,可调节LcrV毒力因子,通过参与群体感应控制基因表达,影响细胞代谢。N-octanoyl-L-Homoserine lactone 是用于研究囊性纤维的感染。
T0077 Dantrolene sodium

Lapatinib ditosylate monohydrate,丹曲林钠,Dantrolene sodium salt

Others; Calcium Channel Membrane transporter/Ion channel; Metabolism; Others
Dantrolene sodium (Lapatinib ditosylate monohydrate) salt 是一种骨骼肌松弛药,是一种钙通道蛋白抑制剂,可抑制钙离子从肌浆释放。
T68837 Zelpolib

Zelpolib is a novel DNA polymerase inhibitor, inhibiting DNA replication in assays to assess global DNA synthesis or single-molecule bases by DNA fiber fluorography.
T26376 11-deoxy-PGF2a

11-deoxyPGF2a,11-deoxy PGF2a

11-deoxy-PGF2a, a selective activator of TREK-2 channels, stimulates DRG c-fiber nociceptor K2P currents and limits calcium influx.
T71208 GO-Y078

GO-Y078 is an antiangiogenic curcumin analog which inhibits actin stress fiber formation, thereby resulting in mobility inhibition.
T23697 AL-8417

J1.090.276B,AL8417,(2R)-AL-5898

AL-8417 is an enzyme inhibitor. It acting as an antioxidant, anti-inflammatory, and cytostatic agent. It also has the ability to suppress vitrectomy-induced posterior lens fiber changes.
TP1696 CGGRGD

CGGRGD is a RGD derivative with cysteine as the n-terminal. CGGRGD was synthesized by solid phase peptide synthesis technology, and amino2-cyanobenzothiazole (2-cyanobenzothiazole) (2-cyanobenzothiazole (CBT) was added on the surface of PCL fiber for ammo
T82798 C3bot(154-182) TFA

C3bot(154-182) TFA 是C3 肽类化合物,能够通过促进脊髓损伤后下行纤维束的再生,增强其修复效能。此外,C3bot(154-182) TFA 或许能够促进中枢神经系统损伤后的轴突保护与修复,并有助于功能性恢复。
T28653 S-8510 free base

SB 737552,SB-737552,S8510,SB737552,S-8510,S 8510

S-8510 is a GABA-A receptor inverse agonist. S-8510 selectively potentiated pentylenetetrazol-induced convulsion without affecting minimal electroconvulsive shock- or strychnine-induced convulsion in ddY mice. S-8510 ameliorated memory impairment induced
T82379 FN-A208 fusion peptide

FN-A208 是源自鼠层粘连蛋白 a1 的 A208 与纤连蛋白 (GRGDS) 活性位点和甘氨酸间隔区融合形成的生物活性肽。该肽能形成淀粉样原纤维,并有助于促进肌动蛋白应力纤维的形成,进而介导成纤维细胞附着,显示出其在组织再生和工程生物粘合剂方面的应用潜力。FN-A208 与 IKVAV 受体和整合素发生相互作用,而在 EDTA 存在下,其活性则会被破坏。

化合物

Light Green SF Yellowish
Cat.No: T20913
Synonym: Acid Green 5,C.I. Acid Green 5,C.I. 42095
Target:
QX 314
Cat.No: T8341
Synonym: QX-314
Target: Others
CGGRGD acetate(1260223-44-6 free base)
Cat.No: TP1696L
Synonym:
Target: Others
N-octanoyl-L-Homoserine lactone
Cat.No: T37744
Synonym: C8-HSL,N-octanoyl-L-Homoserine lactone,OHL
Target: Antibacterial
Dantrolene sodium
Cat.No: T0077
Synonym: Lapatinib ditosylate monohydrate,丹曲林钠,Dantrolene sodium salt
Target: Others, Calcium Channel
Zelpolib
Cat.No: T68837
Synonym:
Target:
11-deoxy-PGF2a
Cat.No: T26376
Synonym: 11-deoxyPGF2a,11-deoxy PGF2a
Target:
GO-Y078
Cat.No: T71208
Synonym:
Target:
AL-8417
Cat.No: T23697
Synonym: J1.090.276B,AL8417,(2R)-AL-5898
Target:
CGGRGD
Cat.No: TP1696
Synonym:
Target:
C3bot(154-182) TFA
Cat.No: T82798
Synonym:
Target:
S-8510 free base
Cat.No: T28653
Synonym: SB 737552,SB-737552,S8510,SB737552,S-8510,S 8510
Target:
FN-A208 fusion peptide
Cat.No: T82379
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T12297 Oleuropeinic acid

Others Others
Oleuropeinic acid 是一种抗氧化剂可溶性纤维,存在于橄榄组织中或通过热处理形成,可能是由橄榄苦苷的氧化形成。
T5S1261 Methylophiopogonanone B

Ras GPCR/G Protein; MAPK
Methylophiopogonanone B 是一种高异二氢黄酮,提取自麦冬的根,抗氧化能力强,它通过 Rho 信号传导途径及增加 GTP-Rho 发挥效果。它能够重组肌动蛋白细胞骨架,使细胞形态(如树突收缩、应力纤维形成)发生变化。
T6S0920 2"-O-Galloylhyperin

2”-O-没食子酰基金丝桃苷,2''-O-Galloylhyperin,Q-100605,FT-0689359

Others Others
2"-O-Galloylhyperin (FT-0689359) 是一种分离自Pyrola incarnateFisch. 中的活性化合物,具有抗氧化和抗炎作用,对氧化应激诱导的肝损伤具有肝保护作用。
T17303 α-Cyclodextrin

Alfadex,NSC269470,α-环糊精,NSC 269470,NSC-269470

Others Others
α-Cyclodextrin (Alfadex) 是一种多功能可溶性膳食纤维,可作为纤维原料销售。
TL0018 Lobelin

AChR; Antifection Microbiology/Virology; Neuroscience
Inhalation challenge with capsaicin and rapid intravenous injection of Lobelin and alinamin indicated that peripheral c-fiber receptors were involved in the induction of coughing.
TN5942 Dammarenediol II

达玛烯二醇II,Dammar-24-ene-3,20-diol

Dammarenediol II may have the ability to prevent diabetic microvascular complications, including diabetic retinopathy, it can inhibit vascular endothelial growth factor (VEGF)-induced intracellular reactive oxygen species generation and stress fiber forma
T83231 8-O-4,8-O-4-Dehydrotriferulic acid

8-O-4,8-O-4-Dehydrotriferulic acid 是从皂化后的玉米麸皮不溶性纤维中提取的一种脱氢三阿魏酸。

天然产物

Oleuropeinic acid
Cat.No: T12297
Synonym:
Target: Others
Methylophiopogonanone B
Cat.No: T5S1261
Synonym:
Target: Ras
2"-O-Galloylhyperin
Cat.No: T6S0920
Synonym: 2”-O-没食子酰基金丝桃苷,2''-O-Galloylhyperin,Q-100605,FT-0689359
Target: Others
α-Cyclodextrin
Cat.No: T17303
Synonym: Alfadex,NSC269470,α-环糊精,NSC 269470,NSC-269470
Target: Others
Lobelin
Cat.No: TL0018
Synonym:
Target: AChR, Antifection
Dammarenediol II
Cat.No: TN5942
Synonym: 达玛烯二醇II,Dammar-24-ene-3,20-diol
Target:
8-O-4,8-O-4-Dehydrotriferulic acid
Cat.No: T83231
Synonym:
Target:
TargetMol Loading
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