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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T12189 NBDHEX

Apoptosis; Glutathione Peroxidase; Autophagy Apoptosis; Autophagy; Metabolism
NBDHEX 是一种谷胱甘肽 S-转移酶 P1-1 抑制剂,也是晚期自噬抑制剂。它诱导肿瘤细胞凋亡,通过抑制 GST 的催化活性,避免抑制剂被特异性泵从细胞中排出,以及破坏 GSTP1-1和关键信号传导因子之间的相互作用,从而起到抗癌的作用。
T69975 Istaroxime oxalate

Istaroxime, also known as PST-2744, is a positive inotropic agent that mediates its action through inhibition of sodium/potassium adenosine triphosphatase (Na+/K+ ATPase). Na+/K+ ATPase inhibition increases intracellular sodium levels, which reverses the driving force of the sodium/calcium exchanger, inhibiting calcium extrusion and possibly facilitating calcium entry. Additionally, Istaroxime increases intracellular calcium by improving the efficacy by which intracellular calcium triggers sarco...

化合物

NBDHEX
Cat.No: T12189
Synonym:
Target: Apoptosis, Glutathione Peroxidase, Autophagy
Istaroxime oxalate
Cat.No: T69975
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T12313 Ophiobolin B

Others Others
Ophiobolin B is a sesterterpene Helminthosporium oryzae metabolite, inhibits proton extrusion from maize coleoptiles.

天然产物

Ophiobolin B
Cat.No: T12313
Synonym:
Target: Others
TargetMol Loading
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