Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T8236 |
RHC 80267
U-57908 |
Others; Phospholipase; COX; Acyltransferase; AChR | Immunology/Inflammation; Metabolism; Neuroscience; Others |
RHC 80267 (U-57908) 是一种选择性二酰基甘油脂酶(DAGL)抑制剂,对犬血小板的IC50为 4 μM。它抑制COX 活性和磷脂酰胆碱的水解,还抑制胆碱酯酶活性,IC50为 4 μM,增强乙酰胆碱引起的松弛。 |