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Cat. No. Product Name Target Signaling Pathways
T7277 SB 242084

6 - 氯-2,3 - 二氢- 5 -甲基- N - [6 - [(2 - 甲基-3 - 吡啶基)氧] -3 - 吡啶基] - 1H -吲哚- 1 - 酰胺盐酸盐,SB 242084 dihydrochloride hydrate

5-HT Receptor GPCR/G Protein; Neuroscience
SB 242084 是5-HT2C 选择性抑制剂,pKi 值9.0,是一种精神活性药物和研究化学品。
T6951 Pramipexole dihydrochloride hydrate

Pramipexole 2HCl Monohydrate,普拉克索盐酸盐水合物,Mirapex,普拉克索

Dopamine Receptor GPCR/G Protein; Neuroscience
Pramipexole dihydrochloride hydrate (Mirapex) 是选择性的,具有血脑屏障 (BBB) 渗透性的 D2 型多巴胺受体激动剂,对 D2 型受体、D2、D3、D4亚型受体的 Ki 分别为 2.2 nM、3.9 nM、0.5 nM、1.3 nM,可用于研究帕金森综合症和腿多动综合征。
T10462L Bavisant dihydrochloride hydrate

JNJ31001074AAC

Others Others
Bavisant dihydrochloride hydrate (JNJ31001074AAC) is a highly selective, orally active antagonist of the human H3 receptor with a novel mechanism of action, involving wakefulness and cognition, with potential as a treatment for ADHD. in vivo: Mean change
T23210 Quinacrine (dihydrochloride hydrate)

Quinacrine (hydrochloride hydrate) (83-89-6 free base)

Others Others
Quinacrine is a compound that is commonly used as an anti-protozoal agent. It inhibits voltage-dependent sodium channels (IC50: 3.3 μM) and suppresses aldehyde oxidase (IC50: 3.3 μM). Quinacrine prevents misfolding of prion protein (EC50: 0.3 μM). As an e
T0788L Spectinomycin dihydrochloride pentahydrate

盐酸大观霉素五水合物,Trobicin,Spectogard,Spectinomycin hydrochloride hydrate

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Spectinomycin dihydrochloride pentahydrate (Spectogard) 是一种广谱氨基环糊精抗生素,可以抑制多种革兰氏阳性和革兰氏阴性生物的生长。
T64151 Mibefradil dihydrochloride hydrate

Mibefradil dihydrochloride hydrate (Ro 40-5967 dihydrochloride hydrate) 是一种长效的钙离子通道拮抗剂。Mibefradil dihydrochloride hydrate 通过对低电压激活 (T) 钙通道的亲和力高于对高电压激活 (L) 钙通道的亲和力来发挥作用。Mibefradil dihydrochloride hydrate 能够降压药。
T75298 Cefotiam dihydrochloride hydrate

Cefotiam (SCE-963) dihydrochloride hydrate,一种肠外头孢菌素类抗生素,对革兰氏阳性菌和革兰氏阴性菌展示出广谱活性。
T22412 Quinacrine hydrochloride hydrate

Mepacrine Dihydrochloride Dihydrate,米帕林盐酸盐,Quinacrine Dihydrochloride Dihydrate

Others Others
Quinacrine, a dye of the acridine family, has been widely used as staining agents for DNA and model compounds for intercalators in numerous biophysical studies. It is also an antimalarial drug.
T72105 BMS-433771 dihydrochloride hydrate

BMS-433771 dihydrochloride hydrate 是一种有效的呼吸道合胞病毒 (RSV) 抑制剂,具有口服活性。BMS-433771 dihydrochloride hydrate 对 A 组和 B 组RSV 均有效,EC50均值为 20 nM。BMS-433771 dihydrochloride hydrate 可用于呼吸道疾病的研究。
T70756 KT172

KT172 是一种 DAGLβ抑制剂,IC50值为 11 nM。KT172 可用于代谢和炎症的研究。

化合物

SB 242084
Cat.No: T7277
Synonym: 6 - 氯-2,3 - 二氢- 5 -甲基- N - [6 - [(2 - 甲基-3 - 吡啶基)氧] -3 - 吡啶基] - 1H -吲哚- 1 - 酰胺盐酸盐,SB 242084 dihydrochloride hydrate
Target: 5-HT Receptor
Pramipexole dihydrochloride hydrate
Cat.No: T6951
Synonym: Pramipexole 2HCl Monohydrate,普拉克索盐酸盐水合物,Mirapex,普拉克索
Target: Dopamine Receptor
Bavisant dihydrochloride hydrate
Cat.No: T10462L
Synonym: JNJ31001074AAC
Target: Others
Quinacrine (dihydrochloride hydrate)
Cat.No: T23210
Synonym: Quinacrine (hydrochloride hydrate) (83-89-6 free base)
Target: Others
Spectinomycin dihydrochloride pentahydrate
Cat.No: T0788L
Synonym: 盐酸大观霉素五水合物,Trobicin,Spectogard,Spectinomycin hydrochloride hydrate
Target: ribosome, Antibacterial, Antibiotic
Mibefradil dihydrochloride hydrate
Cat.No: T64151
Synonym:
Target:
Cefotiam dihydrochloride hydrate
Cat.No: T75298
Synonym:
Target:
Quinacrine hydrochloride hydrate
Cat.No: T22412
Synonym: Mepacrine Dihydrochloride Dihydrate,米帕林盐酸盐,Quinacrine Dihydrochloride Dihydrate
Target: Others
BMS-433771 dihydrochloride hydrate
Cat.No: T72105
Synonym:
Target:
KT172
Cat.No: T70756
Synonym:
Target:
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