Cat. No. | Product Name | Target | Signaling Pathways |
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T7277 |
SB 242084
6 - 氯-2,3 - 二氢- 5 -甲基- N - [6 - [(2 - 甲基-3 - 吡啶基)氧] -3 - 吡啶基] - 1H -吲哚- 1 - 酰胺盐酸盐,SB 242084 dihydrochloride hydrate |
5-HT Receptor | GPCR/G Protein; Neuroscience |
SB 242084 是5-HT2C 选择性抑制剂,pKi 值9.0,是一种精神活性药物和研究化学品。 | |||
T6951 |
Pramipexole dihydrochloride hydrate
Pramipexole 2HCl Monohydrate,普拉克索盐酸盐水合物,Mirapex,普拉克索 |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Pramipexole dihydrochloride hydrate (Mirapex) 是选择性的,具有血脑屏障 (BBB) 渗透性的 D2 型多巴胺受体激动剂,对 D2 型受体、D2、D3、D4亚型受体的 Ki 分别为 2.2 nM、3.9 nM、0.5 nM、1.3 nM,可用于研究帕金森综合症和腿多动综合征。 | |||
T10462L |
Bavisant dihydrochloride hydrate
JNJ31001074AAC |
Others | Others |
Bavisant dihydrochloride hydrate (JNJ31001074AAC) is a highly selective, orally active antagonist of the human H3 receptor with a novel mechanism of action, involving wakefulness and cognition, with potential as a treatment for ADHD. in vivo: Mean change | |||
T23210 |
Quinacrine (dihydrochloride hydrate)
Quinacrine (hydrochloride hydrate) (83-89-6 free base) |
Others | Others |
Quinacrine is a compound that is commonly used as an anti-protozoal agent. It inhibits voltage-dependent sodium channels (IC50: 3.3 μM) and suppresses aldehyde oxidase (IC50: 3.3 μM). Quinacrine prevents misfolding of prion protein (EC50: 0.3 μM). As an e | |||
T0788L |
Spectinomycin dihydrochloride pentahydrate
盐酸大观霉素五水合物,Trobicin,Spectogard,Spectinomycin hydrochloride hydrate |
ribosome; Antibacterial; Antibiotic | Microbiology/Virology |
Spectinomycin dihydrochloride pentahydrate (Spectogard) 是一种广谱氨基环糊精抗生素,可以抑制多种革兰氏阳性和革兰氏阴性生物的生长。 | |||
T64151 |
Mibefradil dihydrochloride hydrate
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Mibefradil dihydrochloride hydrate (Ro 40-5967 dihydrochloride hydrate) 是一种长效的钙离子通道拮抗剂。Mibefradil dihydrochloride hydrate 通过对低电压激活 (T) 钙通道的亲和力高于对高电压激活 (L) 钙通道的亲和力来发挥作用。Mibefradil dihydrochloride hydrate 能够降压药。 | |||
T75298 | Cefotiam dihydrochloride hydrate | ||
Cefotiam (SCE-963) dihydrochloride hydrate,一种肠外头孢菌素类抗生素,对革兰氏阳性菌和革兰氏阴性菌展示出广谱活性。 | |||
T22412 |
Quinacrine hydrochloride hydrate
Mepacrine Dihydrochloride Dihydrate,米帕林盐酸盐,Quinacrine Dihydrochloride Dihydrate |
Others | Others |
Quinacrine, a dye of the acridine family, has been widely used as staining agents for DNA and model compounds for intercalators in numerous biophysical studies. It is also an antimalarial drug. | |||
T72105 |
BMS-433771 dihydrochloride hydrate
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BMS-433771 dihydrochloride hydrate 是一种有效的呼吸道合胞病毒 (RSV) 抑制剂,具有口服活性。BMS-433771 dihydrochloride hydrate 对 A 组和 B 组RSV 均有效,EC50均值为 20 nM。BMS-433771 dihydrochloride hydrate 可用于呼吸道疾病的研究。 | |||
T70756 |
KT172
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KT172 是一种 DAGLβ抑制剂,IC50值为 11 nM。KT172 可用于代谢和炎症的研究。 |