Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0103 |
Dipivefrin hydrochloride
盐酸地匹福林,Dipivefrin HCL |
Adrenergic Receptor; AChR | GPCR/G Protein; Neuroscience |
Dipivefrin hydrochloride (Dipivefrin HCl) 是抗青光眼前体药物,被角膜中的酯酶水解为其活性化合物肾上腺素。 | |||
T9323 |
4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide
4-氨基-6-(三氟甲基)苯-1,3-二磺酰胺,4-Amino-6-(trifluoromethyl)benzene-1,3-d,2,4-Disulfamyl-5-trifluoromethylaniline,2-amino-4-trifluoromethyl-1,5-benzendisulfonamide |
Carbonic Anhydrase | Metabolism |
4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide (4-Amino-6-(trifluoromethyl)benzene-1,3-d) 是一种碳酸酐酶抑制剂,用作潜在的抗肿瘤和抗青光眼药物。 | |||
T1282 |
Carteolol hydrochloride
Arteoptic,Abbott-43326,OPC-1085 hydrochloride,盐酸卡替洛尔,Carteolol HCl,Mikelan |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Carteolol hydrochloride (Abbott-43326) 是一种非选择性的β肾上腺素受体阻断剂。 | |||
T68774 |
Deterenol Free Base
|
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Deterenol Free Base is a beta-adrenoceptor agonist. It is an effective nonmydriatic and nonmiotic hypotensive agent, which can be used in antiglaucoma treatment. | |||
T29707 |
Aganepag ethanediol
AGN-212409,AGN212409 |
||
Aganepag ethanediol 是一种降低眼压的抗青光眼化合物。Aganepag ethanediol 是一种选择性 EP2 受体激动剂。 | |||
T7492 |
Ripasudil free base
K-115 (free base) |
ROCK; Antibacterial | Cell Cycle/Checkpoint; Cytoskeletal Signaling; Microbiology/Virology; Stem Cells |
Ripasudil free base (K-115 (free base)) 是一种ROCK 特异性抑制剂,能够抑制ROCK1和ROCK2的活性,IC50值分别为 51 和 19 nM。 |