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Cat. No. Product Name Target Signaling Pathways
T0103 Dipivefrin hydrochloride

盐酸地匹福林,Dipivefrin HCL

Adrenergic Receptor; AChR GPCR/G Protein; Neuroscience
Dipivefrin hydrochloride (Dipivefrin HCl) 是抗青光眼前体药物,被角膜中的酯酶水解为其活性化合物肾上腺素。
T9323 4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide

4-氨基-6-(三氟甲基)苯-1,3-二磺酰胺,4-Amino-6-(trifluoromethyl)benzene-1,3-d,2,4-Disulfamyl-5-trifluoromethylaniline,2-amino-4-trifluoromethyl-1,5-benzendisulfonamide

Carbonic Anhydrase Metabolism
4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide (4-Amino-6-(trifluoromethyl)benzene-1,3-d) 是一种碳酸酐酶抑制剂,用作潜在的抗肿瘤和抗青光眼药物。
T1282 Carteolol hydrochloride

Arteoptic,Abbott-43326,OPC-1085 hydrochloride,盐酸卡替洛尔,Carteolol HCl,Mikelan

Adrenergic Receptor GPCR/G Protein; Neuroscience
Carteolol hydrochloride (Abbott-43326) 是一种非选择性的β肾上腺素受体阻断剂。
T68774 Deterenol Free Base

Deterenol Free Base is a beta-adrenoceptor agonist. It is an effective nonmydriatic and nonmiotic hypotensive agent, which can be used in antiglaucoma treatment.
T29707 Aganepag ethanediol

AGN-212409,AGN212409

Aganepag ethanediol 是一种降低眼压的抗青光眼化合物。Aganepag ethanediol 是一种选择性 EP2 受体激动剂。
T7492 Ripasudil free base

K-115 (free base)

ROCK; Antibacterial Cell Cycle/Checkpoint; Cytoskeletal Signaling; Microbiology/Virology; Stem Cells
Ripasudil free base (K-115 (free base)) 是一种ROCK 特异性抑制剂,能够抑制ROCK1和ROCK2的活性,IC50值分别为 51 和 19 nM。

化合物

Dipivefrin hydrochloride
Cat.No: T0103
Synonym: 盐酸地匹福林,Dipivefrin HCL
Target: Adrenergic Receptor, AChR
4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide
Cat.No: T9323
Synonym: 4-氨基-6-(三氟甲基)苯-1,3-二磺酰胺,4-Amino-6-(trifluoromethyl)benzene-1,3-d,2,4-Disulfamyl-5-trifluoromethylaniline,2-amino-4-trifluoromethyl-1,5-benzendisulfonamide
Target: Carbonic Anhydrase
Carteolol hydrochloride
Cat.No: T1282
Synonym: Arteoptic,Abbott-43326,OPC-1085 hydrochloride,盐酸卡替洛尔,Carteolol HCl,Mikelan
Target: Adrenergic Receptor
Deterenol Free Base
Cat.No: T68774
Synonym:
Target:
Aganepag ethanediol
Cat.No: T29707
Synonym: AGN-212409,AGN212409
Target:
Ripasudil free base
Cat.No: T7492
Synonym: K-115 (free base)
Target: ROCK, Antibacterial
TargetMol Loading
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