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3

抑制剂 & 化合物

3

天然产物

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Cat. No. Product Name Target Signaling Pathways
T0509 Cloxiquine

5-Chloro-8-quinolinol,氯羟喹,Dermofungin,Dermofongin,5-氯-8-羟基喹啉

Antibacterial; Antibiotic; PPAR; Parasite; Antifungal DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Cloxiquine (Dermofongin) 具有抗菌,抗真菌和抗阿米巴虫的作用。它还可通过激活 PPARγ抑制黑素瘤细胞的生长和转移。它可研究结核病和皮肤病。
T25744 Liroldine

Liroldina,HL-707,Liroldinum,HL707,HL 707

Liroldine is a new synthetic agent with antiamoebic activity.
T75640 Thalifendine chloride

Thalifendine chloride 是 Berberine 的一种代谢物,具有抗疟原虫和抗阿米巴虫活性。Thalifendine chloride 对 P. falciparum 和 E. histolytica 作用的 IC50值分别为 7.91 μM 和 116 μM。

化合物

Cloxiquine
Cat.No: T0509
Synonym: 5-Chloro-8-quinolinol,氯羟喹,Dermofungin,Dermofongin,5-氯-8-羟基喹啉
Target: Antibacterial, Antibiotic, PPAR, Parasite, Antifungal
Liroldine
Cat.No: T25744
Synonym: Liroldina,HL-707,Liroldinum,HL707,HL 707
Target:
Thalifendine chloride
Cat.No: T75640
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T3933 Jatrorrhizine

Yatrorizine,neprotin,药根碱

MAO; 5-HT Receptor; Antibacterial; AChE GPCR/G Protein; Metabolism; Microbiology/Virology; Neuroscience
Jatrorrhizine (neprotin) 是一种从黄连中分离得到的生物碱,具有抗菌、抗氧化、抗疟原虫和神经保护活性。它通过抑制 uptake-2 transporter 的活性减少血清素和去甲肾上腺素的摄取。它是一种有口服活性的乙酰胆碱酯酶制剂。
T4912 Jatrorrhizine chloride

盐酸药根碱,Yatrorhizine chloride,Neprotine chloride

Others; 5-HT Receptor; OCT; Antibacterial; AChE GPCR/G Protein; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; Others
Jatrorrhizine chloride (Neprotine chloride) 是从黄连中分离得到的生物碱,具有神经保护、抗菌、抗氧化和抗疟原虫活性。它通过抑制摄取2转运蛋白的活性减少血清素和去甲肾上腺素的摄取。它是具有口服活性的乙酰胆碱酯酶抑制剂。
TN2399 Isoarborinol

Others Others
Isoarborinol has antiamoebic activity

天然产物

Jatrorrhizine
Cat.No: T3933
Synonym: Yatrorizine,neprotin,药根碱
Target: MAO, 5-HT Receptor, Antibacterial, AChE
Jatrorrhizine chloride
Cat.No: T4912
Synonym: 盐酸药根碱,Yatrorhizine chloride,Neprotine chloride
Target: Others, 5-HT Receptor, OCT, Antibacterial, AChE
Isoarborinol
Cat.No: TN2399
Synonym:
Target: Others
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